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N-({3-[3-(1H-pyrazol-3-yl)phenyl]phenyl}methyl)propanamide
3-{[(4-chlorophenyl)methyl]amino}-N-(4-methoxyphenyl)-5-(methylsulfamoyl)benzamide
N-[(4-ethylphenyl)methyl]-N-methyl-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
1-{1-[6-(aminomethyl)-2-methylpyrimidin-4-yl]piperidin-4-yl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
4-(1H-imidazol-4-ylmethyl)-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
2,4-dimethoxy-N-({4-[(3-phenylpropyl)amino]quinazolin-2-yl}methyl)benzene-1-sulfonamide
N-[(3R,4S)-4-cyclopropyl-1-[1-(2-fluorophenyl)piperidin-4-yl]pyrrolidin-3-yl]acetamide
[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl](methyl)[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]amine
1-{1-ethyl-5-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-4-phenylpiperazine
2-[4-(1,1-dioxo-4,5-dihydro-1λ6-thiophen-2-yl)-1H-pyrazol-1-yl]-N-(1-propyl-1H-1,2,3-triazol-4-yl)acetamide
1-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-4,4,4-trifluorobutan-1-one
1-[3-(3-hydroxy-3-methylbutyl)benzoyl]piperidin-4-ol
N-[(2R,4R,6S)-2-(4-fluoro-3-methoxyphenyl)-6-[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]oxan-4-yl]acetamide
4-[(4aR,8aR)-4a-hydroxy-7-(2-methoxyacetyl)-decahydro-2,7-naphthyridin-2-yl]-1-phenylbutan-1-one
4-[2-oxo-2-(3-propoxypiperidin-1-yl)ethyl]-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
N-{[2-(dimethylamino)-8-methylquinolin-3-yl]methyl}-N-[2-(dimethylamino)ethyl]-2-methoxybenzamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-3-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propanamide
(3R,4S)-1-[(5-ethylthiophen-2-yl)sulfonyl]-4-propylpyrrolidin-3-amine
1-[(2-aminopyridin-3-yl)methyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
8-cyclopropanecarbonyl-2-(3-methyl-1,2-oxazole-5-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl](ethyl)(1,3-thiazol-2-ylmethyl)amine
1-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propan-1-one
5-methyl-5-phenyl-1-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}piperidin-2-one
2-(3-hydroxypropyl)-9-(5-phenyl-1,3,4-thiadiazol-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
3-benzyl-1-methyl-8-(thiophen-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[2-(trifluoromethoxy)phenyl]-1H-pyrazolo[3,4-d]pyrimidin-6-amine
N-(1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-3-yl)acetamide
1-[cyclohexyl(methyl)amino]-3-[2-methoxy-4-({[2-(1-methylpiperidin-4-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
3-(2,3-dihydro-1H-inden-2-yl)-8-[(1-methyl-1H-indol-3-yl)methyl]-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{4-[3-(6-methoxynaphthalene-2-carbonyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
(1S,5R)-3-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propanoyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}acetamide
2-methyl-5-{2-[3-(methylsulfanyl)phenyl]phenyl}-1,3,4-oxadiazole
methyl[(1-phenyl-1H-pyrazol-4-yl)methyl]{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
[1-(4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzoyl)piperidin-2-yl]methanol
(1-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}pyrrolidin-3-yl)methanamine
6-[(diethylamino)methyl]-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
3-(1-{[2-(5-methylfuran-2-yl)phenyl]methyl}piperidin-4-yl)-1-(morpholin-4-yl)propan-1-one
7-(2-methylphenyl)-9-(oxolan-3-ylmethoxy)-4-(quinolin-8-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-(phenoxymethyl)-N-(3-phenylpropyl)-1,2-oxazole-3-carboxamide
(5S,9aS,9bS)-2-[(3-methoxyphenyl)methyl]-5-(3-methyl-1-propyl-1H-pyrazol-4-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-(phenylsulfanyl)-1-{4-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
(4aR,8aR)-7-(7-chloroquinolin-4-yl)-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-carboxamide
1-benzoyl-2-{3-[(2-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}piperidine
(1R,5R)-N,N-dimethyl-6-(4-phenoxybutanoyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-(2-fluorophenyl)-3-[1-(oxan-4-yl)piperidin-3-yl]propanamide
5-(methoxymethyl)-N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]furan-2-carboxamide
N-(1-{7-[(4-fluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-methoxybenzamide
2-methoxy-N-(3-{[(piperidin-4-ylmethyl)carbamoyl]amino}phenyl)acetamide
N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide