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methyl (2S,4S)-4-(furan-2-amido)-1-[(3-methoxyphenyl)methyl]pyrrolidine-2-carboxylate
7-(2-methylphenyl)-4-(morpholine-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(2-chloro-5-fluorophenyl)-3-cyclopropyl-3-[(trimethyl-1H-pyrazol-4-yl)methyl]urea
3-(3,5-dimethylphenyl)-N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)propanamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-2,3,6-trimethylquinoline-4-carboxamide
2-(4-chlorophenyl)-2-hydroxy-1-(4-phenyl-1,4-diazepan-1-yl)ethan-1-one
2-[1-cyclohexyl-4-({3-[3-(dimethylamino)propoxy]phenyl}methyl)piperazin-2-yl]ethan-1-ol
4-[(1R,5S)-3,8-diazabicyclo[3.2.1]octane-8-carbonyl]-2,6,8-trimethylquinoline
8-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2-{[5-(1-methoxypropyl)-4-phenyl-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
2-(furan-2-yl)-1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}pyrrolidine
N-(2-{4-[3-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}ethyl)acetamide
N-benzyl-N-ethyl-3-(3-hydroxyazetidin-1-yl)propanamide
N-[(3,5-dimethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-2-(methylamino)pyridine-4-carboxamide
2-(1-methyl-3-oxopiperazin-2-yl)-N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}acetamide
5-[1-(1H-imidazol-1-ylmethyl)cyclopropyl]-1-(2-phenylethyl)-1H-1,2,4-triazole
3,3-dimethyl-1-(5-methyl-1,2-oxazole-4-carbonyl)-4-(morpholin-4-ylmethyl)piperidin-4-ol
4-(4-{methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl)benzamide
(1S,2R)-2-{methyl[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]amino}cyclohexan-1-ol
3-({4-[2-(2-methylphenyl)-1,3-thiazol-5-yl]-1H-1,2,3-triazol-1-yl}methyl)-1λ6-thiolane-1,1-dione
4-(azocan-1-yl)-N,5-dimethyl-N-(propan-2-yl)thieno[2,3-d]pyrimidine-6-carboxamide
2-ethoxy-4-[1-(oxan-4-yl)-4-phenyl-1H-imidazol-5-yl]phenol
N-(1-benzothiophen-2-ylmethyl)-1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide
2-(4-methoxyphenyl)-5-(2-propoxyethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N-butyl-3-[(3-hydroxyazetidin-1-yl)methyl]-N-methylimidazo[1,2-a]pyridine-2-carboxamide
N-(2-chlorophenyl)-4-[4-(2-hydroxyethyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
3-[(4-fluoro-3-methoxyphenyl)methyl]-9-methoxy-10-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
N-({1-[(5-ethylpyridin-2-yl)methyl]piperidin-3-yl}methyl)-3-methylbut-2-enamide
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetic acid
1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-4-(thiophene-2-carbonyl)piperazine
3-{3-methyl-5-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazol-5-yl]-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
2-cyclohexyl-N-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]-1,3-benzoxazole-6-carboxamide
1-[(4aR,8aR)-4a-hydroxy-7-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
5-{2-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(2-{3-[ethyl(pyridin-4-ylmethyl)amino]piperidine-1-carbonyl}phenyl)ethan-1-one
3,3-dimethyl-1-[(3S,4R)-1-{2-[methyl(pyridin-4-ylmethyl)amino]acetyl}-4-(propan-2-yl)pyrrolidin-3-yl]urea
N-methyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-2-(phenylamino)pyrimidine-5-carboxamide
1-[3-(furan-2-yl)-3-phenylpropyl]-2-(4-methyl-1H-imidazol-5-yl)-1H-imidazole
2-amino-6-(furan-2-yl)-4-(quinolin-4-yl)pyridine-3-carbonitrile
(1R,5R)-6-(1H-indol-5-ylmethyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
2-{5-[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]-4-phenyl-1H-imidazol-1-yl}acetamide
4-{3-[(5-oxo-1-phenylpyrrolidin-3-yl)amino]propoxy}benzamide
1-[9-benzyl-1-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]ethan-1-one
2-({[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}(thiophen-3-ylmethyl)amino)butan-1-ol
N-[(2,4-dihydroxyphenyl)methyl]-2-(dimethylamino)-2-(4-methylphenyl)acetamide
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-4-sulfamoylbenzamide
1-[(4-tert-butylphenyl)methyl]-4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperazine
1-cyclobutanecarbonyl-4-[2-(furan-2-yl)pyrrolidine-1-carbonyl]piperidine
N-cyclopropyl-1-(1-{thieno[3,2-d]pyrimidin-4-yl}piperidin-4-yl)piperidine-3-carboxamide