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2-{1-[(4-ethoxyphenyl)methyl]-4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-yl}ethan-1-ol
N-{[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}-N-(prop-2-yn-1-yl)cyclohexanamine
N-(1-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-4-yl}-2-(2-methylphenyl)ethyl)-N-methyl-2-(1H-pyrazol-1-yl)acetamide
ethyl 5-(7-hydroxy-6-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylate
1-({4-[2-hydroxy-3-(morpholin-4-yl)propoxy]-3-methoxyphenyl}methyl)-4-methylpiperidine-4-carbonitrile
N-[furan-2-yl(phenyl)methyl]-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
3-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidine-1-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
2-{5-[1-(2,4-difluoro-3-methoxybenzoyl)piperidin-4-yl]-1H-pyrazol-3-yl}acetic acid
3-[2-(3-fluorophenyl)ethyl]-1-(4-methyl-1,3-thiazole-5-carbonyl)piperidine
2-(1-{[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
N-methyl-N-[(4-phenoxyphenyl)methyl]quinoxaline-5-carboxamide
4-[1-benzyl-5-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]piperazin-2-one
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)propanamide
2-(adamantan-1-yl)-1-[4-hydroxy-4-(pyrrolidin-1-ylmethyl)piperidin-1-yl]ethan-1-one
(4aS,8aR)-1-[2-(cyclohex-1-en-1-yl)ethyl]-6-(dimethyl-1,3-oxazole-4-carbonyl)-decahydro-1,6-naphthyridin-2-one
5-(2-ethylpiperidine-1-carbonyl)-1-[(3-methoxyphenyl)methyl]-N-methyl-N-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
2-({[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(ethyl)amino)ethan-1-ol
1-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
6-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-1,2,3,4-tetrahydroisoquinoline
3-{[1-butyl-3-(furan-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
4-methyl-5-{2-methyl-3-oxo-2,8-diazaspiro[4.5]decane-8-carbonyl}-2-oxo-1,2-dihydropyridine-3-carbonitrile
(1S,4R)-2-{2-[3-(ethoxymethyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}-2-azabicyclo[2.2.1]heptane
ethyl 1-(4-fluorophenyl)-5-({[2-(4-sulfamoylphenyl)ethyl]amino}methyl)-1H-pyrazole-4-carboxylate
2-(3,3-dimethyl-4-phenylpyrrolidin-1-yl)acetamide
2-(4-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1-(thiophen-2-ylmethyl)piperazin-2-yl)ethan-1-ol
4-[4-(1H-imidazol-1-ylmethyl)phenyl]phenol
N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-[7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
2-[4-(carbamoylmethoxy)-3-methylphenyl]-N,N-bis(propan-2-yl)benzamide
6,8-dimethyl-2-[({2-[(pyridin-3-yl)amino]ethyl}amino)methyl]quinolin-4-ol
{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)[(3-methyl-1,2-oxazol-5-yl)methyl]amine
3-benzyl-4-[2-(3-hydroxyazetidin-1-yl)-2-oxoethyl]-1-(3-methylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N,2,3-trimethyl-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}quinoxaline-6-carboxamide
2-(morpholin-4-yl)-N-(5-oxo-1-propylpyrrolidin-3-yl)pyridine-3-carboxamide
2-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-oxo-N-(propan-2-yl)acetamide
1-[(2-fluorophenyl)methyl]-N-(isoquinolin-5-ylmethyl)-N-methylpiperidin-3-amine
N-[3-(4-chlorophenyl)propyl]-1-(methoxymethyl)cyclobutane-1-carboxamide
1-(1-{2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]acetyl}piperidin-4-yl)pyrrolidin-2-one
N-[1-(3-methoxyphenyl)ethyl]-3-(piperidine-1-carbonyl)pyrazine-2-carboxamide
(2S)-2-amino-2-cyclohexyl-1-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
1-(1-{2-methylpyrido[2,3-d]pyrimidin-4-yl}piperidin-4-yl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-(2,3-dihydro-1H-inden-2-yl)-N-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylpiperidin-3-amine
2-(3-oxo-9-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2,9-diazaspiro[5.5]undecan-2-yl)propanoic acid
9-[4-(4-fluorophenyl)-4-oxobutyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-[1-(6-methylpyridine-3-carbonyl)piperidin-4-yl]propanamide
1-(4-methylpiperazine-1-carbonyl)-4-(pyridin-4-yl)-1,4-diazepan-6-ol
(1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)methanol
N-(5-ethyl-1,3,4-thiadiazol-2-yl)-N'-(2-methoxyethyl)-N'-(thiophen-2-ylmethyl)ethanediamide
(2S,4R)-4-amino-1-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(methylamino)acetamide
methyl 4-({1-methyl-2,4-dioxo-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decan-8-yl}methyl)benzoate