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1-cyclopentyl-4-[(5-cyclopropyl-4-phenyl-1H-imidazol-1-yl)methyl]pyrrolidin-2-one
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2-(morpholin-4-yl)-N-(propan-2-yl)-2-(pyridin-3-yl)acetamide
N-[2-(3-ethylphenoxy)ethyl]-N-methyl-3-(1H-pyrazol-1-ylmethyl)benzamide
N'-(5-chloro-2-methylphenyl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]propanediamide
(3S,4S)-3-hydroxy-4-(propan-2-yloxy)-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-1-carboxamide
ethyl 1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylate
N-({1-[(8-chloroquinolin-2-yl)methyl]pyrrolidin-3-yl}methyl)-2-methoxyacetamide
3-(2-fluorophenyl)-1-(2-methoxyethyl)-3-[2-oxo-2-(3-phenylpiperidin-1-yl)ethyl]pyrrolidine-2,5-dione
N-[(2-chlorophenyl)methyl]-6-({methyl[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]amino}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-methoxy-4-methyl-1,3-thiazole-5-carboxamide
{[3-(furan-2-yl)phenyl]methyl}[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amine
2-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl](methyl)amino}-2-[4-(propan-2-yloxy)phenyl]acetic acid
N-[(2R,4S,6R)-2-(4-chlorophenyl)-6-(2-methylpropyl)oxan-4-yl]acetamide
2-methyl-4-{4-[4-(trifluoromethyl)piperidine-1-carbonyl]phenyl}butan-2-ol
1-(4-{[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
(3R,9aR)-8-(4-fluorobenzoyl)-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(3S,4R)-1-(1-benzoylpiperidin-4-yl)-4-(3-methylthiophen-2-yl)piperidin-3-ol
5,6-dimethyl-N-(1,2-oxazol-3-ylmethyl)-2-(pyrrolidin-1-yl)pyrimidin-4-amine
2-(3-{2-amino-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridine-5-carbonyl}piperidin-1-yl)acetamide
methyl 3-benzamido-6-{[methyl(oxolan-3-yl)amino]methyl}thieno[2,3-b]pyridine-2-carboxylate
1-methyl-4-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]-1H-indole
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(1H-1,2,4-triazol-3-yl)benzamide
4-(2-fluorophenyl)-2-{4-[4-(2-methoxyethyl)piperazine-1-carbonyl]-5-methyl-1H-pyrazol-1-yl}pyrimidine
N-[(dimethyl-1,3-thiazol-5-yl)methyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
8-(dimethyl-1,3-oxazole-4-carbonyl)-3-hexyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[2-({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}formamido)ethyl]acetamide
1-[4-methyl-2-({2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}amino)pyrimidin-5-yl]ethan-1-one
N-(3,4-dihydro-2H-1-benzopyran-3-yl)-4-(piperidin-1-ylmethyl)benzamide
4-(hydroxymethyl)-N-[(4-methyl-5-oxomorpholin-2-yl)methyl]benzamide
6-cyclopropyl-N-[3-(dimethylamino)-1-phenylpropyl]pyrimidin-4-amine
2-[(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinolin-2-yl]-5-fluoro-N-methylpyrimidin-4-amine
(1R,2S,9S)-11-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
(3E)-1-(4-{4-cyclopropyl-5-[(dimethylamino)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pent-3-en-1-one
3-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-1-(4-ethoxy-2-fluorophenyl)-3-methylurea
3-(but-2-yn-1-yl)-5-{1-[(3-methoxyphenyl)methyl]piperidin-4-yl}-5-(3-phenylpropyl)imidazolidine-2,4-dione
1-[(2-methyl-1H-imidazol-4-yl)methyl]-2-(pyrrolidin-1-ylmethyl)piperidine
4-benzyl-3-(1-ethyl-1H-pyrazol-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-methyl-2-(methylamino)-N-[2-(4-methylmorpholin-2-yl)ethyl]propanamide
6-[4-(4-fluorophenyl)benzoyl]-N-[2-(pyridin-2-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]ethan-1-one
3-{3-[({[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)methyl]-1H-indol-1-yl}propanamide
7-({4-[(pyrimidin-2-yl)amino]piperidin-1-yl}methyl)-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
(2-ethoxy-5-{[2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl}phenyl)methyl acetate
(1S,2S)-2-[(2-amino-5-ethylpyrimidin-4-yl)amino]cyclohexan-1-ol
N-methyl-2-[3-({[3-(2-oxopyrrolidin-1-yl)propyl]carbamoyl}amino)phenyl]acetamide
3,4-dimethoxy-N-{[4-(2-methylphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}benzamide
N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
[(1-butyl-2-cyclobutylmethanesulfonyl-1H-imidazol-5-yl)methyl][2-(diethylamino)ethyl]methylamine
4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-6-(pyrrolidin-1-yl)pyrimidin-2-amine
4-[4-(4-methylpiperazine-1-carbonyl)pyridin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine