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1-(2-phenylethyl)-3-(1,3-thiazol-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3R,5R)-1-(2-methylpropyl)-3-(pyrrolidin-1-ylmethyl)-5-(pyrrolidine-1-carbonyl)piperidine
N-[4-(2-fluorophenoxy)phenyl]-1-[(trimethylpyrazin-2-yl)methyl]piperidine-4-carboxamide
5-ethyl-6-methyl-N4-[3-(3-methyl-1H-pyrazol-1-yl)propyl]pyrimidine-2,4-diamine
1-[7-(1-benzothiophen-3-yl)-9-(pyridin-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(1,3-benzoxazol-2-yl)propan-1-one
2-(4-butyl-2,3-dioxopiperazin-1-yl)-N-cyclohexyl-2-phenylacetamide
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-{3-[(pyridin-3-yl)amino]propyl}acetamide
2-(2,5-difluorophenyl)-2-(4-propyl-1,4-diazepan-1-yl)acetic acid
1-[(5-chloro-2,3-dimethoxyphenyl)methyl]-3-(pyrrolidine-1-carbonyl)piperidine
3-[(3R,4S)-1-[3-(dimethylamino)pyrazin-2-yl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
7-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}cyclopentanecarboxamide
1-(3,4-dimethylphenyl)-N-[(3-methoxyphenyl)methyl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-[2-(4-methoxyphenyl)phenyl]-1-(1H-pyrrole-3-carbonyl)piperidine-3-carboxamide
1-(3,3-dimethylbutanoyl)-N-[3-(4-fluorophenyl)phenyl]piperidine-3-carboxamide
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-(1,3-thiazol-2-ylmethyl)-decahydro-2,7-naphthyridine-2-sulfonamide
(1-{3-[(pyrimidin-4-yl)amino]propyl}piperidin-3-yl)methanol
(2S)-2-cyclohexyl-2-{[2-(ethylamino)pyrimidin-5-yl]formamido}acetic acid
methyl(1H-pyrazol-3-ylmethyl)(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)amine
2-{1-[(3-cyanophenyl)methyl]piperidin-2-yl}acetamide
5-(2,5-dimethylfuran-3-yl)-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-1,2,4-triazin-3-amine
2,5-difluoro-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}benzamide
1-{4-[(2-chloro-4,5-dimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-3-methylbutan-1-ol
(2R)-N-[(2-methoxyphenyl)methyl]-N-(pyridin-4-ylmethyl)pyrrolidine-2-carboxamide
methyl (2R,4S)-4-hydroxy-1-(pyridine-3-carbonyl)piperidine-2-carboxylate
1-[3-(oxan-4-yl)-1-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]-6-azaspiro[2.5]octane
3-ethyl-4-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}piperazin-2-one
8-methoxy-2-[4-(pyridin-3-ylmethyl)piperazin-1-yl]quinoline
N-{[1-(4-ethenylbenzoyl)piperidin-3-yl]methyl}naphthalene-1-carboxamide
6-fluoro-4-[3-(1H-pyrazol-5-yl)piperidine-1-carbonyl]-1,2-dihydroquinolin-2-one
N-{1-[1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2,2-dimethylpropanamide
2-ethoxy-5-[2-(propan-2-yl)pyrimidin-4-yl]benzoic acid
N-{1-[1-(2-methylpropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-phenylbutanamide
N-{4-[2-hydroxy-3-(2-methylphenoxy)propanamido]-2-methylphenyl}pentanamide
(2S)-N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-acetamido-4-(methylsulfanyl)butanamide
1-(2-{3-[4-(methylsulfanyl)benzoyl]piperidine-1-carbonyl}phenyl)ethan-1-one
3-{2-amino-4-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-6-methylpyrimidin-5-yl}propanoic acid
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-3-(2-methyl-1H-imidazol-1-yl)propanamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-9-methoxy-3-(3-methylbenzoyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-(3,3-dimethylbutanoyl)-4'-[(1-methyl-1H-imidazol-5-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-(1H-pyrazol-4-yl)-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]benzamide
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,3,6-trifluorobenzamide
3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-1-[(4-methoxyphenyl)methyl]urea
N-[1-(butan-2-yl)-3-methyl-1H-pyrazol-5-yl]-2-[4-(9H-purin-6-yl)-1H-pyrazol-1-yl]acetamide
(3aR,5R,6S,7aS)-2-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-octahydro-1H-isoindole-5,6-diol
2-benzyl-4-{[4-(pyrimidin-2-yloxy)phenyl]methyl}morpholine
2-[({[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}(methyl)amino)methyl]-3,4-dihydroquinazolin-4-one
5-[(2-chlorophenyl)methyl]-3-(cyclopropylmethyl)-5-{1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
5-(methoxymethyl)-N-({7-[(4-methoxynaphthalen-1-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)furan-2-carboxamide
1-[2-(4-methylphenyl)quinoline-4-carbonyl]azetidine-2-carboxylic acid