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1-(4-{[2-(4-chlorophenyl)pyrimidin-5-yl]methyl}-1,4-diazepan-1-yl)-2-methoxyethan-1-one
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
3-{5-[(2-ethyl-1-benzofuran-3-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}pyridine
N-methyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-(4-{2-[(1-benzylpyrrolidin-3-yl)carbamoyl]ethyl}piperidin-1-yl)acetic acid
1-(2-methoxyphenyl)-3-(1-{1-[3-(methylsulfanyl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
4-{[5-(2-fluorophenyl)furan-2-yl]methyl}-N,N-dimethylpiperazine-1-sulfonamide
8-(2-aminoacetyl)-3-{2-[cyclohexyl(methyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(1S,5S)-3-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-6-methyl-3,6-diazabicyclo[3.2.2]nonane
8-(furan-2-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
N-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-propylpropanamide
1-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}-2-(morpholin-3-yl)ethan-1-one
1-cyclopentyl-4-[1-(2-methoxyphenyl)-1H-1,2,4-triazol-5-yl]pyrrolidin-2-one
(3aR,6aS)-5-(2,3-dihydro-1-benzofuran-7-carbonyl)-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(1H-imidazol-2-ylmethyl)-3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-butyl-5-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]pyrazine-2-carboxamide
1-[3-(aminomethyl)phenyl]-3-{[1-(hydroxymethyl)cyclobutyl]methyl}-3-methylurea
4-{[5-(hydroxymethyl)furan-2-yl]methyl}-1-(propan-2-yl)-6-{[4-(trifluoromethoxy)phenyl]methoxy}-1,4-diazepan-2-one
1-[1-(2-fluorophenyl)cyclopropanecarbonyl]-1,4-diazepane-6-carboxylic acid
1-[4-({methyl[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)thiophen-2-yl]ethan-1-one
1-(cyclohex-1-ene-1-carbonyl)-N-(3,4-dimethoxyphenyl)piperidin-3-amine
8-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
(1R)-1-[3-cyclopropyl-1-(1-propyl-1H-1,3-benzodiazol-2-yl)-1H-1,2,4-triazol-5-yl]butane-1,4-diamine
{3-ethyl-1-[2-(methylamino)pyridine-4-carbonyl]piperidin-3-yl}methanol
2-methoxy-1-[1'-(5-methyl-1,3-oxazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
N2-[1-(4,6-dimethylpyrimidin-2-yl)piperidin-4-yl]-N1-(3-methylpyridin-4-yl)ethane-1,2-diamine
2-[1-(2-propyl-1,3-thiazole-4-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
3-ethyl-8-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
methyl 4-(2-ethylpyrimidine-5-carbonyl)piperazine-1-carboxylate
2-(4-chlorophenyl)-2-{2-[1-(propan-2-yl)piperidin-4-yl]acetamido}acetic acid
3-(3-fluoro-4-phenylbenzoyl)-1-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidine
4-(2-{1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperidin-2-yl}ethyl)phenol
2-(4-acetylphenoxy)-N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]acetamide
4-(1H-imidazol-2-ylmethyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
1-[3-(2-methyl-5-propylpyrimidin-4-yl)phenyl]ethan-1-one
3-methyl-8-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N2,N2,5,6-tetramethyl-N4-[3-(1H-1,2,4-triazol-1-yl)propyl]pyrimidine-2,4-diamine
4-[(1,3-diphenyl-1H-pyrazol-4-yl)methyl]-7-(pyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-3-(pyridin-4-yl)propanamide
1-ethyl-3-[(3-methoxyphenyl)methyl]-8-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(3,4-dimethyl-6-oxo-1,6-dihydropyridazin-1-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
5-{[(3,5-difluorophenyl)methyl]amino}-N,N-dimethyl-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(2,6-difluoro-4-methoxybenzoyl)-3-(2-ethylphenoxy)azetidine
2-(dimethylamino)-4-methyl-N-[1-(4-methylphenyl)cyclopropyl]pyrimidine-5-carboxamide
N-[3-(3-{[4-(2,3-dimethylphenyl)piperazin-1-yl]methyl}phenoxy)propyl]propanamide
2-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-N,N-dimethylpyridine-3-carboxamide
6-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyrimidin-4-amine