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2-{4-[(4-ethoxyphenyl)methyl]-1-(propan-2-yl)piperazin-2-yl}ethan-1-ol
N,N-dimethyl-4-({1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidin-3-yl}formamido)butanamide
N-[2-(pyridin-3-ylformamido)ethyl]oxane-2-carboxamide
N1,N1-dimethyl-N3-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]piperidine-1,3-dicarboxamide
N-methyl-2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
2-phenoxy-N-{[8-(pyridin-4-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
(3R,4R)-3-cyclobutyl-N-[(4-fluorophenyl)methyl]-3-hydroxy-4-methylpyrrolidine-1-carboxamide
N-ethyl-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-(methylamino)pyridine-3-carboxamide
(1S,3R)-N-cyclohexyl-3-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamido]cyclopentane-1-carboxamide
3-({3-azaspiro[5.5]undecan-9-yl}amino)-1-[4-(propan-2-yl)piperazin-1-yl]propan-1-one
[7-(1H-1,3-benzodiazol-6-yl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methanamine
(2S)-2-({[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amino)propanamide
methyl 5-{[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}-3-(oxolane-2-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-[(2S)-2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl]-2-(pyridin-4-yl)pyrimidine
(2S,4S)-4-{[(4-fluorophenyl)methyl]amino}-N-(propan-2-yl)-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
N-[(5-fluoro-2-methylphenyl)methyl]-1,3-dimethyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-[1-(1-{[2-(difluoromethoxy)phenyl]methyl}piperidin-4-yl)ethyl]morpholine
1-[(2S)-2-(3-ethyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]-3-(3-hydroxyquinoxalin-2-yl)propan-1-one
1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine
methyl 5-(2-{[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]carbamoyl}piperidin-1-yl)-5-oxopentanoate
4-(1H-imidazol-1-yl)-1-(pyrrolidine-1-carbonyl)piperidine-4-carboxylic acid
1-(2-methoxybenzoyl)-4-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}piperazine
3-{1-[(2-methoxyphenyl)methyl]-1H-pyrazol-5-yl}-1-[2-(piperidin-1-yl)ethyl]urea
2-[(4-methoxyphenyl)methyl]-4-(thiophene-3-carbonyl)morpholine
(2S)-1-(piperidin-4-yl)-N-[(4-sulfamoylphenyl)methyl]pyrrolidine-2-carboxamide
7-methoxy-5-(1-methyl-1H-pyrazol-4-yl)-1-benzofuran-2-carboxylic acid
3-(5-chloro-4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}-1-methyl-1H-pyrazol-3-yl)-5-methyl-1,2-oxazole
N6-benzyl-N5-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N5-methyl-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
1-[(4-chlorophenyl)methyl]-N-(1H-indol-4-ylmethyl)-6-oxopiperidine-3-carboxamide
N-methyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-2-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-4-yl)acetamide
3-(2-methoxyethyl)-6-phenyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(oxan-4-ylmethyl)acetamide
3-({[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl](methyl)amino}methyl)-N-(pyridin-2-yl)benzamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-5-[1-(2,3-dihydro-1H-inden-2-yl)-1H-pyrazol-3-yl]-4-methyl-1,3-thiazol-2-amine
2-(2-chlorophenyl)-N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
5-[1-(2-cyclopentylacetyl)piperidin-4-yl]-5-(pyridin-3-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-[4-(methylsulfanyl)phenyl]ethan-1-one
1-benzyl-4-[2-(1H-pyrazol-1-yl)benzoyl]piperazine
[4-(2-phenoxyethyl)-1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl]methanol
N-[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-2,7,8-trimethylquinoline-4-carboxamide
1-{4-[(1-cyclopentylpiperidin-4-yl)oxy]-3-methoxybenzoyl}azepane
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
5-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine-2-carbonitrile
6-{[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
3-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl}-3-(4-methoxyphenyl)-1-methylpyrrolidine-2,5-dione
1-{1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
2-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-1-(morpholin-4-yl)ethan-1-one
1,5-dimethyl-4-{7-oxo-1H,5H,6H,7H,8H-pyrido[3,2-f]indazol-5-yl}-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
N-methyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1,2,3,4-tetrahydronaphthalen-1-amine
6-methyl-2-{[3-(1-phenylcyclopropyl)-1-propyl-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydropyridazin-3-one