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N-[3-(1H-imidazol-1-yl)propyl]-3-[(oxolan-3-yl)sulfamoyl]benzamide
6-[4-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]-1-methyl-1H-indole
3-(cyclopentylsulfamoyl)-N-[(dimethyl-1,2-oxazol-4-yl)methyl]benzamide
(3S,4S)-4-(4-fluorophenyl)-1-(5-methyl-1H-indole-2-carbonyl)piperidin-3-ol
(2R,3R,6R)-5-{imidazo[1,2-a]pyrimidine-2-carbonyl}-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(1H-1,3-benzodiazol-2-ylmethyl)-2-[4-(1,3-benzothiazol-2-yl)-2-[(dimethylamino)methyl]phenoxy]acetamide
1-[1'-(3,5-dimethylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
2,2-dimethyl-1-(4-phenylazepan-1-yl)butan-1-one
N-cyclopropyl-1-[1-(6-ethylpyrimidin-4-yl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
[(3R,4R)-1-[2-(dimethylamino)benzoyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
N-(3,4-dimethoxyphenyl)-1-(2,3-dimethylquinoxaline-6-carbonyl)piperidin-3-amine
methyl 8-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-1-ethoxy-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-N'-(4-methylphenyl)propanediamide
7-fluoro-3-methyl-2-{4-[1-(morpholin-4-yl)ethyl]piperidine-1-carbonyl}-1H-indole
N-{2-[2-(methylcarbamoyl)ethyl]phenyl}-2-phenylmorpholine-4-carboxamide
N-methyl-2-(1-oxo-1,2-dihydrophthalazin-2-yl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)acetamide
1-{1-[1-(6-phenylpyridazin-3-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}ethan-1-ol
3-[1-(2H-1,3-benzodioxol-4-ylmethyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)propanamide
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N,6-dimethyl-2-[(2-methylphenyl)methyl]-4-oxo-1-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3-carboxamide
2-[3-(propan-2-yl)-5-[1-(1H-pyrazol-1-yl)propyl]-1H-1,2,4-triazol-1-yl]pyridine
2-(2-chloro-4-fluorophenyl)-1-[4-(2-methoxybenzoyl)piperazin-1-yl]ethan-1-one
2-butyl-5-chloro-4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}-1H-imidazole
3-chloro-N-cyclopentyl-4-{[1-(2-hydroxypropanoyl)piperidin-4-yl]oxy}benzamide
methyl 5-[(5-methyl-2-phenyl-1,3-oxazol-4-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
1-methyl-4-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-2-phenylpiperazine
3-(1-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1H-1,2,3-triazol-4-yl)piperidine
1-[3-(methylsulfanyl)propyl]-3-[3-(propan-2-yloxy)benzoyl]piperidine
{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}(methyl)[(5-methyl-1,2-oxazol-3-yl)methyl]amine
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-({[2-(furan-2-yl)ethyl]amino}methyl)-3-hydroxypiperidin-2-one
2-(4-{[2-(cyclopentyloxy)phenyl]methyl}-1-(propan-2-yl)piperazin-2-yl)ethan-1-ol
N-butyl-1-cyclohexyl-4-oxo-5-[4-(pyridin-4-ylmethyl)piperazine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
5-{3-[(4aS,8aR)-decahydroisoquinolin-2-yl]-3-oxopropyl}-5-(naphthalen-2-ylmethyl)pyrrolidin-2-one
N-(furan-2-ylmethyl)-5-{[(3-methoxyphenyl)methyl]amino}-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}-4-(oxolane-2-carbonyl)-1,4-diazepane
N4-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N2,N2,N4,5,6-pentamethylpyrimidine-2,4-diamine
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-[4-(1-benzothiophen-3-yl)-2-(morpholin-4-ylmethyl)phenoxy]acetamide
5-ethyl-2,3-dimethyl-N-(piperidin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
2-{8-methylimidazo[1,2-a]pyridin-3-yl}-1-[4-(pyrimidin-2-yloxy)piperidin-1-yl]ethan-1-one
2-methyl-N-[5-(6-methyl-9H-purin-9-yl)pyridin-2-yl]propanamide
2-[2-(2,6-difluoro-4-methoxyphenyl)-1H-imidazol-1-yl]ethan-1-ol
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-amine
1-{4-[2-(3-methoxyphenyl)-1-[methyl(pyridin-3-ylmethyl)amino]ethyl]piperidin-1-yl}-2-(1-methyl-1H-pyrrol-3-yl)ethan-1-one
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-3-(1-methyl-1H-pyrazol-4-yl)propanamide
5-{3-[(4-fluorophenyl)methoxy]azetidine-1-carbonyl}-3-(2-methylpropyl)-1,2-oxazole
(2S,4R)-4-(cycloheptylamino)-N-methyl-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
1-ethyl-5-[3-(2-fluorophenoxy)azetidine-1-carbonyl]-3-(2-methylpropyl)-1H-pyrazole
N-ethyl-5-(3-fluorophenoxymethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-3-carboxamide
2-{4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-(1-methylpiperidin-4-yl)piperazin-2-yl}ethan-1-ol
N-[(4-fluorophenyl)methyl]-N-(3-methoxypropyl)-1,2-oxazole-3-carboxamide
N-[(2R,4R,6S)-2-cyclohexyl-6-(6-methoxypyridin-3-yl)oxan-4-yl]acetamide