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1-{1-[(ethylcarbamoyl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(5-methyl-1,2-oxazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
[(2,3-dimethoxyphenyl)methyl][2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]amine
N-{5-[(5S,9aS,9bS)-2-[(2-methoxyphenyl)methyl]-1-oxo-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-5-yl]thiophen-2-yl}acetamide
2,2-dimethyl-5-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]thiomorpholin-3-one
N-[(4-methoxyphenyl)methyl]-N-{[7-(methylsulfanyl)-2-(thiophen-2-yl)quinolin-3-yl]methyl}propanamide
4-benzyl-1-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}pyrrolidin-2-one
4-[(5-fluoro-2-methylphenyl)methyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-(2-methyl-4-{4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
4-[4-({4-[(2-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenyl]but-3-yn-1-ol
2-[benzyl({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)amino]ethan-1-ol
4-methyl-N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)-1,2,3-thiadiazole-5-carboxamide
1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(methylsulfanyl)propan-1-one
1-(4-benzylpiperazin-1-yl)-3-{1-[(3,4-difluorophenyl)methyl]piperidin-3-yl}propan-1-one
5-[2-methyl-6-(trifluoromethyl)quinolin-4-yl]pyridin-3-amine
(5-{[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]methyl}-2-ethoxyphenyl)methanol
1-(cyclopropylmethyl)-5-(1H-1,2,4-triazole-5-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
2-{3-ethoxy-4-[(2-methylprop-2-en-1-yl)oxy]phenyl}-1H-imidazole
4-(3-hydroxy-3-methylbutyl)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}benzamide
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-2-oxo-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)acetamide
3-[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-4,5,6,7-tetrahydro-1-benzofuran-4-one
{[2-(difluoromethoxy)phenyl]methyl}({1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
3-(2-methoxyphenyl)-N-{1-[2-(1,2-oxazolidin-2-yl)-2-oxoethyl]-1H-pyrazol-4-yl}propanamide
6-[(5-chloro-2-hydroxyphenyl)methyl]-N-(2-methyl-1,3-benzothiazol-5-yl)-6-azaspiro[2.5]octane-1-carboxamide
6-(3-fluorophenyl)-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-6-oxo-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
2-{4-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-1-(3-methylbutyl)piperazin-2-yl}ethan-1-ol
2-[methyl(pyridin-3-ylmethyl)amino]-1-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
1-(2-chloroprop-2-en-1-yl)-6,7-dimethoxy-3-({[(trimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-1,2-dihydroquinolin-2-one
3-[2-(dimethylamino)ethyl]-5-[(3-fluorophenyl)methyl]-5-{1-[2-(1-methyl-1H-pyrrol-3-yl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
N-[4-(4-aminopyridin-3-yl)phenyl]-2-methylpropanamide
3,4,7-trimethyl-N-({1-[(4-methylpiperazin-1-yl)methyl]cyclopropyl}methyl)-1H-indole-2-carboxamide
2-(2-methoxyethoxy)-1-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]ethan-1-one
4-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}morpholine
4-(1-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)morpholine
ethyl 4-[1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperazine-1-carboxylate
2-(1-benzylpiperidin-4-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(3aR,6aS)-N-(1H-1,2,3-benzotriazol-5-yl)-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-2-carboxamide
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}({[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl})(oxolan-2-ylmethyl)amine
2-(1-butyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}acetamide
5-{5-[(4-methylpiperazin-1-yl)methyl]pyridin-2-yl}pyridin-2-amine
(2S)-2-[4-(4-fluoro-3-methoxyphenyl)-1H-1,2,3-triazol-1-yl]-3-(4-hydroxyphenyl)propanoic acid
4-(2-{6-chloro-[1,2,4]triazolo[4,3-a]pyridin-3-yl}-2-methylpropyl)morpholine
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-3-ethoxy-4-(prop-2-en-1-yloxy)benzamide
[(2,3-dimethoxyphenyl)methyl]({[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})amine
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(3-chlorophenyl)methyl]-4-{[(3-fluorophenyl)methyl]amino}pyrrolidine-2-carboxamide
7-cyclopropanecarbonyl-N-[4-(pyridin-2-yl)butyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-(4-fluorophenyl)-4-(oxane-4-carbonyl)-1,4-diazepane
N-[(1-cyclopentylpiperidin-4-yl)methyl]-3-(2-oxopyrrolidin-1-yl)-N-(pyridin-3-ylmethyl)propanamide
1-(4-{[(pyridin-3-ylmethyl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol