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5-(2,6-difluorophenoxymethyl)-N-[1-(naphthalen-1-yl)ethyl]-1,2-oxazole-3-carboxamide
1-{[6-(4-chlorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-3-methoxypiperidine
3-[(2-fluorophenyl)methyl]-1-methyl-6-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
(2E)-1-[3-(5-methyl-2-{[2-(morpholin-4-yl)ethyl]sulfanyl}pyrimidin-4-yl)piperidin-1-yl]-3-(pyridin-3-yl)prop-2-en-1-one
4-[(1-{[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methyl]morpholine
6-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-2-carbonitrile
{3-[(4-fluorophenyl)methyl]-1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidin-3-yl}methanol
1-methyl-2-oxo-8-(5,6,7,8-tetrahydroquinolin-2-yl)-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-(2-{3-[1-(2-hydroxyethyl)-1H-pyrazol-3-yl]phenyl}phenyl)ethan-1-one
(3aS,6aR)-5-(2-ethoxyacetyl)-3-[3-(4-methoxyphenyl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
5-acetyl-N,2,4-trimethyl-N-(quinolin-5-ylmethyl)-1H-pyrrole-3-carboxamide
(4aR,8aS)-6-(adamantan-2-yl)-1-{[3-(trifluoromethyl)phenyl]methyl}-decahydro-1,6-naphthyridin-2-one
N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-1H-pyrazole-3-carboxamide
methyl N-{2-[(4aS,7aR)-4-(2-methoxyethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-2-oxoethyl}carbamate
methyl (2S,4R)-4-(quinoline-2-amido)-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxylate
4-(2-methyl-1H-imidazol-1-yl)-1-[(2E)-3-(1-methyl-1H-pyrazol-4-yl)prop-2-enoyl]piperidine-4-carboxylic acid
1-{2-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}pyrrolidin-2-one
8-[3-(dimethylamino)propyl]-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[3-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]-3-[2-(pyrrolidine-1-sulfonyl)ethyl]urea
5-{[3-(4-methyl-3-phenylpiperazine-1-carbonyl)-1,2-oxazol-5-yl]methoxy}isoquinoline
3-[(3R,4S)-1-[(4-fluoro-3-methylphenyl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
N-(4-{4-[(2-methoxyethyl)amino]piperidin-1-yl}phenyl)-5-phenylpentanamide
2-{4-[(2-ethylphenyl)methyl]-2-oxopiperazin-1-yl}benzonitrile
2-{[(2S,4S)-2-[4-(adamantan-2-yl)piperazine-1-carbonyl]-4-[(4-methoxyphenyl)sulfanyl]pyrrolidin-1-yl]methyl}-4-methoxyphenol
N-methyl-3-propanamido-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)benzamide
(3S,4R)-4-(3-fluorophenyl)-1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]pyrrolidine-3-carboxylic acid
4-(4-{[(4-chlorophenyl)(pyridin-4-yl)methyl]amino}piperidin-1-yl)-N-cyclopentylbenzamide
5-ethyl-4-[4-(4-methylphenyl)piperazin-1-yl]pyrimidin-2-amine
1-[(3-chlorothiophen-2-yl)methyl]piperidin-3-ol
1-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
1,5-dimethyl-2-({4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}methyl)-1H-indole
1-(2-phenoxyethyl)-4-(5-propyl-1,3,4-oxadiazol-2-yl)piperazine
2-{5-[2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)ethyl]-1-[(4-fluorophenyl)methyl]-1H-1,2,4-triazol-3-yl}acetamide
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(pyrazin-2-yl)propanamide
3-[4-(2-fluorophenoxy)piperidine-1-carbonyl]-2,8-diazaspiro[4.5]decane
2-methoxy-N-[7-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-1-(2-phenylethyl)-1H-1,3-benzodiazol-5-yl]acetamide
8-fluoro-2-{[(2S)-2-(morpholine-4-carbonyl)pyrrolidin-1-yl]methyl}quinolin-4-ol
(3S,9aR)-8-[(2-methoxyphenyl)methyl]-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[(3-acetylphenyl)methyl]-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
3-(2-chlorophenyl)-1-[2-(dimethylamino)ethyl]-3-{2-[4-(2-hydroxyethyl)piperazin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
5-{[3-(2,3-dimethoxyphenyl)pyrrolidin-1-yl]methyl}-3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazole
N-ethyl-4-oxo-N-[(2E)-3-phenylprop-2-en-1-yl]-4H-chromene-2-carboxamide
N-[(3-chlorophenyl)methyl]-3-[1-(2-methylpyridine-3-carbonyl)piperidin-4-yl]propanamide
1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-hydroxypropan-1-one
N,3,6-trimethyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
N-(cyclohex-1-en-1-ylmethyl)-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
2-(cyclohex-1-en-1-yl)-N-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]methyl}acetamide
2-(2-{[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}phenoxy)ethan-1-ol
2-[4-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1-(3-phenylpropyl)piperazin-2-yl]ethan-1-ol
2-(1-{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}pyrrolidin-2-yl)pyridine