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1-{2-[4-(5-chloro-2-methylphenyl)piperazin-1-yl]-2-oxoethyl}-3-methoxy-1,2-dihydropyridin-2-one
N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]quinoline-2-carboxamide
methyl 9-(cyclopentyloxy)-3-(1H-indol-3-ylmethyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
7-methoxy-N-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-[1-(3,5-dimethylfuran-2-carbonyl)piperidin-3-yl]-1-(4-methylpiperazin-1-yl)propan-1-one
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
4-(4-methyl-1,3-oxazole-5-carbonyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{2-[4-(4-fluorophenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]ethyl}-5-methylthiophene-2-carboxamide
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-[(2-hydroxyethyl)(methyl)amino]pyridine-3-carboxamide
4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)-1-[(2-methoxyphenyl)methyl]piperidine
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-6-oxo-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
2-[(prop-2-en-1-yl)amino]-N-[1-(pyridin-4-yl)propan-2-yl]benzamide
1-[(4aR,8aS)-6-[2-(4-methoxyphenyl)acetyl]-decahydro-1,6-naphthyridin-1-yl]-2-(4-methylphenoxy)ethan-1-one
4-{[4-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1-(propan-2-yl)-1H-pyrazole
8-(2-methylpyrimidin-4-yl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-[(3S,4R)-4-(morpholin-4-yl)-1-(naphthalen-1-ylmethyl)piperidin-3-yl]-N-(propan-2-yl)propanamide
3-hydroxy-1-(2-methoxyethyl)-3-{[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]methyl}piperidin-2-one
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(2,5-dimethylbenzoyl)piperidine
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-5-methyl-1,3-oxazole-4-carboxamide
methyl 1-[(3S,5S)-1-(adamantan-2-yl)-5-{[2-(1H-indol-3-yl)ethyl]carbamoyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
1-(4,7-dimethylquinazolin-2-yl)-N-[(1R)-1-(4-methoxyphenyl)ethyl]piperidine-4-carboxamide
1-(4-{[4-(5-methylpyrimidin-4-yl)piperidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
4-(propan-2-yl)-6-(3-{[4-(propan-2-yl)phenyl]amino}piperidine-1-carbonyl)pyrimidin-2-amine
3-(4-methoxy-3,5-dimethylbenzoyl)piperidine
N-[(3-methoxyphenyl)methyl]-4-(4-methylphenyl)-5-(pyrimidin-5-yl)pyrimidin-2-amine
(3S,4S)-4-(morpholin-4-yl)-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-ol
N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-2-(2,2,6,6-tetramethylpiperidin-4-yl)acetamide
2-{1-[(5-methylfuran-2-yl)methyl]-4-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperazin-2-yl}ethan-1-ol
(5S,9aS,9bS)-5-(2,1,3-benzothiadiazol-5-yl)-2-[(3-chlorophenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-(furan-2-ylmethyl)-4-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}piperidine
N-(1-{7-[(2-ethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)furan-2-carboxamide
4-({1-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]pyrrolidin-3-yl}methyl)benzoic acid
1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine
6-tert-butyl-2-[4-(1,4-oxazepan-4-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-methyl-1,5-diazatricyclo[5.2.2.02,6]undecane
4-(5-{[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]methyl}thiophen-2-yl)-2-methylbut-3-yn-2-ol
ethyl 2-(4-{[4-(pyridin-4-yl)piperazine-1-carbonyl]amino}phenyl)acetate
(2R,3S,6R)-5-(dimethyl-1,3-thiazole-5-carbonyl)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-acetyl-3-[(3R,4S)-3-amino-4-(4-methoxyphenyl)pyrrolidine-1-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N-methyl-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
4-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-6-methyl-1-(2-methylphenyl)piperazin-2-one
3-(2-fluorophenyl)-3-phenyl-N-[2-(pyridin-3-yl)ethyl]propanamide
N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
4-[2-(2-methoxyethyl)piperidine-1-carbonyl]-2-methyl-1H-1,3-benzodiazole
(3aR,7aS)-5-methyl-2-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}-2,3,3a,4,7,7a-hexahydro-1H-isoindole
7-[(2,3-difluorophenyl)methyl]-2-(pyrazin-2-yl)-2,7-diazaspiro[4.5]decane
4-(2-fluoro-5-methylphenyl)-6-methylpyrimidin-2-amine
9-[(2-fluoro-4-methylphenyl)methyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
8-[4-(hydroxymethyl)benzoyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one