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N-[1-(1H-imidazol-1-yl)-3-methylbutan-2-yl]-1-phenyl-1H-1,2,3-triazole-5-carboxamide
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[2-(dimethylamino)-2-(furan-2-yl)ethyl]benzamide
dimethyl(3-{2-[1-(5-methylthiophene-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)amine
1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-2-(3-methylphenoxy)ethan-1-one
N-cyclopropyl-1-{1-[2-(3-hydroxyphenyl)acetyl]piperidin-4-yl}piperidine-3-carboxamide
2-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]pyridine-4-carbonitrile
1-({5-[(4-acetylphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
9-(2,3-difluorobenzoyl)-3,9-diazaspiro[5.6]dodecane
(dicyclopropylmethyl)({[2-methanesulfonyl-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl})methylamine
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1,3-dimethyl-1H-pyrazole-4-carboxamide
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-[4-(3-methoxyphenyl)phenyl]piperidine-3-carboxamide
N'1-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}cyclopropane-1,1-dicarboxamide
7-chloro-2-methyl-4-[(3,4,5-trimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
methyl (2S,4R)-1-[(3-fluorophenyl)methyl]-4-[4-(trifluoromethyl)benzamido]pyrrolidine-2-carboxylate
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-methyl-N-[(1-methylpyrrolidin-2-yl)methyl]acetamide
1-(2,3-dihydro-1-benzofuran-2-carbonyl)-4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
1-ethyl-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
4-benzyl-3-ethyl-1-(pyridine-3-carbonyl)-1,4-diazepan-5-one
(2E)-3-phenyl-1-{4-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}prop-2-en-1-one
{3-oxo-3-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propyl}urea
4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]-N-(dimethyl-1,2-oxazol-4-yl)piperidine-1-carboxamide
N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[2-(2,3-difluoro-6-methoxyphenyl)-1H-imidazol-1-yl]-3-ethoxypropan-2-ol
2-[3-butyl-5-oxo-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-cyclopropylacetamide
N-{2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
2-{3-[3-methyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]pyrrolidin-1-yl}-5-(trifluoromethyl)pyridine
8-(3-cyclopropyl-1,2-oxazole-5-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(3aR,6aS)-5-methyl-N-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-2-carboxamide
5-{1-[(2-methyl-1H-indol-3-yl)methyl]piperidin-4-yl}-5-(2-phenylethyl)imidazolidine-2,4-dione
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-6-(methoxymethyl)-N-methylpyrimidin-4-amine
4-[4-hydroxy-4-(pyridin-3-yl)piperidine-1-carbonyl]-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
N-(1H-1,3-benzodiazol-2-ylmethyl)-2-[1-cyclopropyl-3-(4-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide
methyl 4-({1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}carbamoyl)butanoate
1-[(1R,5S,6R)-6-{[(2-methoxyethyl)(thiophen-2-ylmethyl)amino]methyl}-3-azabicyclo[3.1.0]hexan-3-yl]ethan-1-one
2-{3-[(3-chlorophenyl)methoxy]phenyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
2-(5-fluoro-2-methoxyphenyl)pyridine-4-carbonitrile
3,5-dimethyl-1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)-1H-1,2,4-triazole
1-[6-(2,3-dihydro-1-benzofuran-7-yl)pyridine-3-carbonyl]-4-(pyrimidin-2-yl)-1,4-diazepane
3-{1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}phenol
N-(4-{[1-(4-fluoro-3-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}phenyl)acetamide
N-[(1-cyclopropyl-5-oxopyrrolidin-3-yl)methyl]-N'-(3,5-dimethylphenyl)propanediamide
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)acetamide
2-(5-ethylfuran-2-yl)-1-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-1H-imidazole
4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-methyl-N-(thiophen-2-ylmethyl)benzamide
1-{2-[1-(2,3-dimethylphenyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]ethyl}-4-methylpiperazine
1-[4-(4-{[cycloheptyl(ethyl)amino]methyl}-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-2-methylpropan-1-one
(3R,4R)-4-(4-methylpiperazin-1-yl)-1-[4-(piperidin-1-yl)benzoyl]piperidin-3-ol
N-methyl-N-(oxan-4-yl)-5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine