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(4aR,8aR)-7-[4-(benzyloxy)butyl]-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-carboxamide
N-ethyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-4-(1H-pyrazol-1-yl)benzamide
5-{4-hydroxy-1-[(2E)-2-methylbut-2-en-1-yl]piperidin-4-yl}-N-methyl-N-(quinolin-6-ylmethyl)-1-benzofuran-2-carboxamide
methyl 3-{[(3-fluorophenyl)formamido]methyl}-5-(2-methoxybenzamido)benzoate
8-({2-oxo-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-3-yl}methyl)-1,3-dioxa-8-azaspiro[4.5]decan-2-one
2-ethyl-4-phenyl-9-(1H-pyrazole-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[2-(4-ethylpiperazin-1-yl)ethyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-[3-oxo-1-(pyridin-3-ylmethyl)piperazin-2-yl]-N-[2-(thiophen-2-yl)ethyl]acetamide
N-cyclopropyl-2-(1,2,3,4-tetrahydroisoquinolin-5-yl)pyridine-4-carboxamide
N-({3-[(3-fluorophenyl)methoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
N-(oxan-2-ylmethyl)-5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-amine
3-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}propanoic acid
2-{1-[2-(phenoxymethyl)-1,3-oxazole-4-carbonyl]piperidin-2-yl}pyridine
[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl](methyl){[2-(methylsulfanyl)pyrimidin-5-yl]methyl}amine
1-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
N-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
N-(adamantan-1-ylmethyl)-N-methyl-2-(1-methyl-3-oxopiperazin-2-yl)acetamide
1-[(5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)amino]propan-2-ol
4-[2-(3,4-dihydro-2H-1,4-benzoxazin-4-yl)-2-oxoethyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-[3-(2,6-dimethylphenoxy)azetidin-1-yl]-2-{2-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
1-{4-[3-({[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]amino}methyl)pyridin-2-yl]piperazin-1-yl}ethan-1-one
3-[(4-{4-cyclopropyl-5-[(dimethylamino)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]phenol
N-[(3S,5S)-1-cyclopentanecarbonyl-5-(ethylcarbamoyl)pyrrolidin-3-yl]-6-methylpyridine-3-carboxamide
N-(3-cyclopentylpropyl)-4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-methylbenzamide
{[5-(1H-imidazol-4-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}(methyl)[(5-methylthiophen-2-yl)methyl]amine
N-[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]-6-(2-methylphenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-{2-[2-(2-fluorophenyl)acetamido]ethyl}-N-(thiophen-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
4-(cyclohexylmethyl)-11-(4-propylpiperazin-1-yl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-[(1R)-1-(4-methoxyphenyl)ethyl]-1-(4,6,7-trimethylquinazolin-2-yl)piperidine-4-carboxamide
N,4-dimethyl-N-[(5-methylthiophen-2-yl)methyl]-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
N-benzyl-2-[1-cyclopentyl-3-(3-fluorophenyl)-2,5-dioxopyrrolidin-3-yl]-N-(2-hydroxyethyl)acetamide
(2,1,3-benzothiadiazol-5-ylmethyl)[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]methylamine
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-1-(propan-2-yl)piperidine-4-carboxamide
N-{4-[3-(diethylamino)propanamido]phenyl}-4-methylbenzamide
5-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}-N-phenylpyrimidin-2-amine
{5H,6H,7H,8H,9H,10H-cyclohepta[b]indol-2-ylmethyl}[(1-ethyl-1H-imidazol-2-yl)methyl]amine
1-cyclopentyl-4-[5-(2,5-dimethylphenyl)-4-methyl-1H-imidazol-2-yl]pyrrolidin-2-one
2-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propanamide
3-[(2,3-dimethoxyphenyl)methyl]-5-methyl-5-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}imidazolidine-2,4-dione
2-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-2-azatricyclo[6.3.1.04,12]dodeca-1(12),4,6,8,10-pentaen-3-one
N-({1-[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidin-3-yl}methyl)acetamide
3-(3-chlorophenyl)-3-(2-hydroxyphenyl)-N-methyl-N-(2-methylprop-2-en-1-yl)propanamide
{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}[(2-methoxyphenyl)methyl](prop-2-en-1-yl)amine
N-cyclopropyl-N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-2,1,3-benzothiadiazole-4-sulfonamide
1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-3-(pyrrolidin-1-yl)piperidine
5-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane-4-carbonyl}-2-(propan-2-yl)-3,4-dihydropyrimidin-4-one
1-{4-[4-(pyrazin-2-yl)piperazine-1-carbonyl]phenyl}imidazolidine-2,4-dione
5-methyl-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-1,2-oxazole-3-carboxamide
4-(3-chloropyridin-2-yl)-1H-indole
methyl (2S,4S)-1-[(2-ethoxyphenyl)methyl]-4-[3-(4-fluorophenyl)benzamido]pyrrolidine-2-carboxylate