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N-[3-(4-{[1-(1,3-thiazol-5-yl)propan-2-yl]amino}piperidin-1-yl)phenyl]-3-(trifluoromethyl)benzamide
4-({3-[4-methoxy-4-(prop-2-en-1-yl)piperidine-1-carbonyl]-1,2-oxazol-5-yl}methyl)morpholine
1-[2-(4-methoxyphenyl)ethyl]-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-6-oxopiperidine-3-carboxamide
1-{1-[1-(2-chloro-5-fluorobenzoyl)piperidin-4-yl]ethyl}-4-methylpiperazine
N-(2H-1,3-benzodioxol-5-ylmethyl)-9-methoxy-3-(4-methyl-2-oxopentanoyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-1-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}ethan-1-one
(2-fluoro-5-{2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}phenyl)methanol
1-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-hydroxy-4-(methylsulfanyl)butan-1-one
methyl[2-methyl-2-(morpholin-4-yl)propyl]{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
4-{[ethyl(pyridin-4-ylmethyl)amino]methyl}-N-(1-methyl-1H-1,2,3-triazol-4-yl)benzamide
4-methyl-2-(1-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperidin-3-yl)-1H-1,3-benzodiazole
[(2S,4R,5R)-4-({[(5-cyclopentylthiophen-2-yl)methyl]amino}methyl)-5-(2-fluorophenyl)-1-methylpyrrolidin-2-yl]methanol
2-({5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-1-(furan-2-yl)ethan-1-ol
N-[1-({[1-(2-methyl-1,3-thiazol-4-yl)ethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-2-phenoxyacetamide
N-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]-6-(3-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
methyl 3-acetamido-5-{[(3-fluorophenyl)methyl]amino}-1-[2-(4-methoxyphenyl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-{1-[4-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]pyrrolidin-2-yl}-4-methyl-1H-1,3-benzodiazole
2-[(5-methylpyrazin-2-yl)methyl]-8-(1H-1,2,4-triazole-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(pyrrolidin-1-yl)-N-[1-(1H-1,2,4-triazol-5-yl)ethyl]benzamide
6-methyl-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
3-[(3S,4R)-3-cyclopropyl-4-(1-methyl-1H-pyrazole-4-amido)pyrrolidin-1-yl]propanoic acid
(2-ethoxy-5-{[2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methyl}phenyl)methyl acetate
N-ethyl-2-{4-[(4-fluorophenyl)methyl]-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl}-N-methylacetamide
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
4-(1-benzyl-1H-imidazol-2-yl)-1-(3-methoxybenzoyl)piperidine
methyl 2-hydroxy-5-[3-(methylcarbamoyl)-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl]benzoate
5-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1,3-dimethyl-1H-pyrazole
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)acetamide
4-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine
N-(1-benzofuran-5-ylmethyl)-1-methyl-N-(pyridin-3-ylmethyl)piperidin-4-amine
ethyl 5-[(4-carbamoylpiperidin-1-yl)methyl]-1-(2,5-dimethylphenyl)-1H-pyrazole-4-carboxylate
N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-3-(1H-pyrazol-1-ylmethyl)benzamide
N-[(1-ethyl-1H-indazol-3-yl)methyl]-1-(oxan-4-yl)piperidine-3-carboxamide
4-fluoro-N-{2-[7-(2-phenylpropyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}benzamide
2-(4-methyl-1,2,5-oxadiazol-3-yl)-N-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}acetamide
N-[1-(5-{[2-(4-fluorophenoxy)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-4-(2-oxopyrrolidin-1-yl)benzamide
9-(dimethoxy-1,3,5-triazin-2-yl)-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane
1-[4-(3-{[(1-benzofuran-2-ylmethyl)amino]methyl}pyridin-2-yl)piperazin-1-yl]ethan-1-one
2-{[2-({2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}carbamoyl)phenyl]amino}acetic acid
5-(2,4-difluorophenoxymethyl)-N-(oxolan-2-ylmethyl)-1H-pyrazole-3-carboxamide
5-methyl-N-[1-(pyridin-3-yl)propan-2-yl]-1-[4-(pyridin-3-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
4-(cyclopropylmethyl)-1-[4-(3-hydroxypyrrolidin-1-yl)pyrimidin-2-yl]piperidine-4-carboxylic acid
4-{[5-(3-cyclohexyl-1H-pyrazol-4-yl)-1,2,4-oxadiazol-3-yl]methyl}morpholine
1-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]-2-(trimethyl-1H-pyrazol-1-yl)ethan-1-one
9-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
4-(hydroxymethyl)-1-[1-(4-methoxyphenyl)cyclopentanecarbonyl]azepan-4-ol
N-[1-(butan-2-yl)-1H-pyrazol-5-yl]-2,6-dimethylquinoline-3-carboxamide
9-methoxy-4-(2-methylpropyl)-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-({5-[(benzyloxy)methyl]-4-phenyl-1H-imidazol-1-yl}methyl)-5-methyl-1,2-oxazole
(4aR,7aS)-1-benzyl-4-{[2-(methylamino)-1,3-thiazol-4-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione