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N-({4-[(4-fluorophenyl)methoxy]phenyl}methyl)-4-(1H-pyrazol-1-yl)-N-(pyridin-3-ylmethyl)benzamide
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
(2S,4R)-4-({[4-(benzyloxy)phenyl]methyl}amino)-1-[(3-chlorophenyl)methyl]-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
8-(5-cyclobutyl-3-methyl-1H-1,2,4-triazol-1-yl)quinoline
3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-{2-[(1,3-thiazol-2-yl)carbamoyl]ethyl}propanamide
3-({1-[6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidin-4-yl}oxy)pyridine
N-(1-{1-[4-(piperidin-1-ylmethyl)benzoyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
2-{4-[5-(ethylsulfanyl)thiophene-2-carbonyl]morpholin-3-yl}acetic acid
4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(5-methylthiophene-2-carbonyl)piperidine
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]urea
N-(5-chloro-2-methoxyphenyl)-3-[1-(2-methyl-1H-pyrrole-3-carbonyl)piperidin-3-yl]propanamide
N-(2-methoxyethyl)-1-{1-[4-methyl-6-(methylamino)pyrimidin-2-yl]piperidin-4-yl}piperidine-3-carboxamide
1-{1-[(2,5-dimethylphenyl)methyl]piperidin-4-yl}-N-(2-hydroxyethyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide
1-benzoyl-N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]piperidin-4-amine
5-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]quinoxaline
6-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}pyridine-3-carboxylic acid
N-(3-hydroxypropyl)-1-{[5-(pyrimidin-2-ylsulfanyl)furan-2-yl]methyl}piperidine-3-carboxamide
(4aR,7aS)-4-(3-hydroxy-4-methylbenzoyl)-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-3-(morpholin-4-ylmethyl)piperidin-2-one
1-(3-cyanophenyl)-3-[2-(dimethylsulfamoyl)ethyl]urea
3-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]propanamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-2-(3-hydroxypiperidin-1-yl)acetamide
1-(2-ethylpyridine-4-carbonyl)-4-(3-phenylpropyl)-1,4-diazepane
3-{2-[3-(2-methylpropyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-1,2,4-triazol-5-amine
{1-cyclohexyl-3-[(2,4-difluorophenyl)methyl]piperidin-3-yl}methanol
3-chloro-N-(2-methoxyethyl)-4-{[1-(2-oxopropanoyl)piperidin-4-yl]oxy}benzamide
N-{4-[2-(dimethylamino)ethoxy]-1-(4-fluorophenyl)-1H-indazol-3-yl}-1-methylcyclopropane-1-carboxamide
N-[1-benzyl-4-(morpholin-4-yl)-1H-indazol-3-yl]-2-propoxyacetamide
3-({2-[1-(2-chlorophenyl)-1H-1,2,4-triazol-5-yl]ethyl}(methyl)amino)-1λ6-thiolane-1,1-dione
2-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-N-methylacetamide
2-(phenoxymethyl)-5-[2-(trifluoromethyl)pyrrolidine-1-carbonyl]pyrimidin-4-ol
1-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(pyridin-3-yl)propan-1-one
4-(1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-yl)-1-(2-methylpropyl)piperidine
N-{3-[2-(dimethylcarbamoyl)ethyl]phenyl}-8-methyl-9-oxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
2-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-2,8-diazaspiro[4.5]decane
[(2-tert-butylpyrimidin-5-yl)methyl](methyl)[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]amine
N-(2-hydroxyethyl)-N-methyl-1-(1-{[4-(trifluoromethoxy)phenyl]methyl}piperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide
2-(4-{4-[(3-methylphenyl)methyl]-3-oxopiperazine-1-carbonyl}phenoxy)acetamide
(2S,4S)-4-amino-1-(2,3-dihydro-1-benzofuran-5-carbonyl)-N-methylpyrrolidine-2-carboxamide
{1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-3-(2-phenoxyethyl)piperidin-3-yl}methanol
(3R,4S)-1-[5-(methoxymethyl)thiophene-2-carbonyl]-3,4-dimethylpiperidin-4-ol
N-(3-ethylphenyl)-3-[4-(pyridin-4-yl)piperazin-1-yl]propanamide
2-(1,3-thiazol-2-yl)-1-(1,3-thiazol-4-ylmethyl)piperidine
(2S,4S)-4-[(adamantan-2-yl)amino]-1-(2,3-dihydro-1H-inden-2-yl)-N,N-diethylpyrrolidine-2-carboxamide
methyl[(5-methylfuran-2-yl)methyl][(3-phenyloxolan-3-yl)methyl]amine
2-{[4-(2,3-difluoro-4-methylphenyl)-1H-1,2,3-triazol-1-yl]methyl}-4,6-dimethylpyrimidine
2-amino-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-6-(trimethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
1-(2-methylfuran-3-carbonyl)-4-(thiophen-2-ylmethyl)-1,4-diazepane
2-ethyl-4-methyl-N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}-1,3-oxazole-5-carboxamide