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1-benzyl-3-methyl-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2S)-N-{3-[(4-chlorophenyl)sulfanyl]propyl}-1-(piperidin-4-yl)pyrrolidine-2-carboxamide
6-methyl-2-(1-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidin-2-yl)-1H-1,3-benzodiazole
3-(4-chloro-2-methylbenzoyl)-1-(5-methoxyfuran-2-carbonyl)piperidine
6-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[2-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-2-[3-(trifluoromethyl)phenyl]ethan-1-one
2-ethyl-4-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-6-methylpyrimidine
4-acetyl-N-(4-acetylphenyl)-4-phenylpiperidine-1-carboxamide
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)propyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
3-[1-(4-oxo-3,4-dihydroquinazoline-2-carbonyl)piperidin-3-yl]benzoic acid
1-(methoxymethyl)-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)cyclobutane-1-carboxamide
2-{4-[2-(3-oxo-2,3-dihydro-1H-indazol-2-yl)acetyl]piperazin-1-yl}-N-(propan-2-yl)acetamide
(3aR,7aS)-5-methyl-2-[4-methyl-2-(piperidin-1-yl)pyrimidine-5-carbonyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
[3-(2-phenylethyl)-1-(3-phenylpropyl)piperidin-3-yl]methanol
(2S,4R)-4-amino-1-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-N-methylpyrrolidine-2-carboxamide
5-[(dimethylamino)methyl]-N-{5-[2-(4-methylphenoxy)ethyl]-1,3,4-thiadiazol-2-yl}furan-2-carboxamide
N-[3-(4-{[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]amino}piperidin-1-yl)phenyl]ethane-1-sulfonamide
9-(5-methylpyrazine-2-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]-N-[2-(pyrrolidin-1-yl)ethyl]acetamide
1-benzyl-5-(pyridin-4-ylmethyl)-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
3-[3-({[1-(2,4-dimethoxyphenyl)ethyl](methyl)amino}methyl)-1H-indol-1-yl]propanamide
ethyl 4-(3-phenylpropyl)-1-(1,3-thiazole-5-carbonyl)piperidine-4-carboxylate
1-[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(thiophen-2-yl)ethan-1-one
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-4-(pyridin-2-yl)pyrimidin-2-amine
[4-(6-aminopyridine-3-carbonyl)-1,4-oxazepan-6-yl]methanol
N-(2-methoxyethyl)-N-[(3-methylthiophen-2-yl)methyl]-3-(1H-1,2,4-triazol-1-yl)propanamide
(3aS,6aR)-3-[2-(4-fluorophenyl)ethyl]-5-methanesulfonyl-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(pyridin-3-yl)pyrimidin-2-amine
3-(5-amino-1H-1,2,4-triazol-3-yl)-N-[1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]propanamide
1-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
1-{3-cyclopropyl-5-[2-(phenylamino)pyrimidin-5-yl]-1H-1,2,4-triazol-1-yl}butan-2-ol
{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}(furan-3-ylmethyl)methylamine
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)morpholine-2-carboxamide
[(5-ethylfuran-2-yl)methyl](methyl)[2-(oxan-2-yl)ethyl]amine
N-tert-butyl-2-methyl-3-[2-(pyridin-2-yl)acetamido]benzamide
N-[4-(3-fluorophenyl)phenyl]-1-(1,3-thiazole-5-carbonyl)piperidine-3-carboxamide
4-[3-(hydroxymethyl)-3-(3-phenylpropyl)piperidine-1-carbonyl]pyridin-1-ium-1-olate
2-amino-6-methyl-4-[3-methyl-4-(pyrrolidin-1-yl)phenyl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
(1r,4r)-4-[(6-methylhept-5-en-2-yl)amino]cyclohexan-1-ol
4-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]benzonitrile
6-(3-fluorophenyl)-N-methyl-N-[1-(pyridin-2-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
[(3R,4S)-1-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
8-[(2,5-dimethylphenyl)methyl]-1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1R,5R)-6-(cyclobutylmethyl)-3-(2-ethoxypyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decane
(1R,3S,5S)-8-[3-(2-methoxyphenyl)benzoyl]-8-azabicyclo[3.2.1]octan-3-ol
N-benzyl-N-methyl-3-({[2-(piperidin-1-yl)ethyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
N-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-6-methoxypyridin-2-amine
N-methyl-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]-N-[2-(1H-pyrazol-4-yl)ethyl]acetamide