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2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxy-N-methyl-N-[(4-methylphenyl)methyl]benzamide
1-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-4-(morpholine-4-carbonyl)-1,4-diazepan-6-ol
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-{[(pyridin-3-ylmethyl)amino]methyl}piperidin-2-one
(3-ethyl-1-{[2-(ethylamino)pyrimidin-5-yl]methyl}piperidin-3-yl)methanol
(1R,5S)-6-methyl-3-[(3-phenyl-1,2-oxazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
(3R,4R)-4-ethyl-1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]piperidine-3,4-diol
1-ethyl-5-[(3-phenoxyazetidin-1-yl)methyl]-1H-1,2,4-triazole
1-[1-(2-methylpropyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
{[(3S,4R)-1-(4-fluoro-3-methoxybenzoyl)-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
(2R,6R)-4-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-10-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-{4-[(dimethyl-1,3-thiazol-5-yl)methyl]piperazin-1-yl}pyrimidine
1-[3-({[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)propyl]pyrrolidin-2-one
N,N-diethyl-1-[(1s,4s)-4-(5-methyl-3-phenyl-1,2-oxazole-4-amido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
6-[(3-fluorophenyl)methoxy]-1-(2-phenylethyl)-4-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}-1,4-diazepan-2-one
5-benzyl-1-(3-methoxyphenyl)-4-[(3E)-pent-3-enoyl]piperazin-2-one
methyl 2-(tert-butylsulfamoyl)-6-{[3-(trifluoromethyl)phenyl]methyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-[4-(4-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]-1-methylimidazolidin-2-one
3-(6-chloropyridin-3-yl)-1-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]urea
1-(4-{4-[2-(methylsulfanyl)pyrimidin-4-yl]piperazin-1-yl}piperidin-1-yl)butan-1-one
4-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}-1,4-oxazepan-5-one
methyl (2S)-3-methyl-2-[(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}phenyl)formamido]butanoate
{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}[1-(2-methoxyphenyl)ethyl]methylamine
N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]cyclopent-1-ene-1-carboxamide
4-[(3,5-dimethoxyphenyl)methyl]-3-[2-oxo-2-(pyrrolidin-1-yl)ethyl]piperazin-2-one
2-amino-N-[1-(butan-2-yl)-1H-pyrazol-5-yl]-6-(2-methylpropyl)pyrimidine-4-carboxamide
2,3-dimethyl-N-[7-oxo-5-(4-propylpiperazine-1-carbonyl)-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]benzamide
3-{2-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
N-[3-(1H-imidazol-2-yl)propyl]-6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
4-({4-[(4-methoxyphenyl)methyl]-3-oxopiperazin-1-yl}methyl)-1,5-dimethyl-1H-pyrrole-2-carbonitrile
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-3-[5-(thiophen-2-yl)-1,3,4-thiadiazol-2-yl]urea
N-{[1-(3-phenylpropyl)pyrrolidin-3-yl]methyl}methanesulfonamide
N-(1-{1-[(3,4-dimethoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide
1-(carbamoylmethyl)-N-methyl-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]piperidine-4-carboxamide
2-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-[1-(3-hydroxybenzoyl)piperidin-4-yl]propanamide
5-{[4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]methyl}-2-methoxypyridine
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)acetamide
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
1-methyl-3-{2-oxo-2-[4-(thiophen-2-ylmethyl)piperazin-1-yl]ethyl}-3-(4-phenylphenyl)pyrrolidine-2,5-dione
4-(2,2-diphenylethyl)piperazine-2-carboxylic acid
N-[(7-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]-3-(pyridin-3-yl)propanamide
5-(2,4-dimethoxypyrimidin-5-yl)-2-methylquinoline
2-(4-butyl-2,3-dioxopiperazin-1-yl)-N-[(5-methylthiophen-2-yl)methyl]-2-phenylacetamide
[(4aS,8aR)-6-(5-methyl-2-phenylfuran-3-carbonyl)-decahydro-1,6-naphthyridin-4a-yl]methanol
N-[(1R,2R)-2-hydroxycyclohexyl]-N-propyl-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
{1-[(1-benzyl-1H-imidazol-5-yl)methyl]-3-propylpiperidin-3-yl}methanol
2-(adamantan-1-yl)-N-{[1-(prop-2-en-1-yl)pyrrolidin-3-yl]methyl}acetamide
3-[2-(2-fluorophenoxy)pyridin-3-yl]-1-(piperidin-4-ylmethyl)urea
3-{2-[(2-methoxyethyl)[(3-methylthiophen-2-yl)methyl]amino]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
(1R,2S,9R)-11-[2-(1H-1,3-benzodiazol-1-yl)acetyl]-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one