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3-chloro-4-{[1-(furan-3-ylmethyl)piperidin-4-yl]oxy}-N-(2-methoxyethyl)benzamide
4-{[1-(cyclohexylmethyl)-2-methanesulfonyl-1H-imidazol-5-yl]methyl}morpholine
1-[(4-hydroxyquinolin-2-yl)methyl]-N-[4-(1H-pyrazol-5-yl)phenyl]piperidine-3-carboxamide
1-[(3S,4S)-3-[benzyl(methyl)amino]-4-hydroxypyrrolidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
2-({[(3R,4R)-1-(2,3-dichlorobenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(ethyl)amino)ethan-1-ol
1-(naphthalen-1-ylmethyl)-N-[3-(pyridin-3-yloxy)propyl]-1H-1,2,3-triazole-4-carboxamide
2-[3-({methyl[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]amino}methyl)phenyl]-3,4,5,6,7,8-hexahydroquinazolin-4-one
2-({ethyl[(1-methylpyrrolidin-3-yl)methyl]amino}methyl)benzoic acid
N-(1H-pyrazol-3-yl)-5-{1-[2-(pyridin-2-yl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
N-[(2R,3R)-1'-(1,5-dimethyl-1H-pyrazole-3-carbonyl)-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
1-{3-[4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
5-{[7-(cyclopropylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
8-(6-methylpyridine-3-carbonyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
1-methyl-1'-[3-(2-oxo-1,2-dihydropyridin-1-yl)propanoyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
1-[3-(thiophen-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyrrolidine
2-[3-cyclopropyl-5-(methanesulfonylmethyl)-1H-1,2,4-triazol-1-yl]pyridine
(3S,5R)-N3-(6-methylpyridin-3-yl)-N5-[2-(2-oxoimidazolidin-1-yl)ethyl]piperidine-3,5-dicarboxamide
N-[1-(propan-2-yl)-1H-pyrazol-4-yl]-2-[2-(pyridin-2-yl)ethyl]piperidine-1-carboxamide
N-[4-(furan-2-yl)butan-2-yl]-4-(4-methylphenoxy)piperidine-4-carboxamide
4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]-N-(1-methyl-1H-1,3-benzodiazol-5-yl)piperidine-1-carboxamide
3-[2-(2,2-diphenylethyl)morpholine-4-carbonyl]pyridin-1-ium-1-olate
N-[2-chloro-4-(2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamido)phenyl]propanamide
3-tert-butyl-1-({1-[(1-ethenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}methyl)urea
2-[2,5-dioxo-3-phenyl-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]-N-(oxolan-2-ylmethyl)-N-propylacetamide
2-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl](methyl)amino}-2-(2-methoxy-5-methylphenyl)acetic acid
N-[3-(6-methyl-1,3-benzoxazol-2-yl)propyl]-5-(oxolan-2-yl)thiophene-2-carboxamide
1-methyl-5-[2-(3-phenylpyrrolidin-1-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]-1-[7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-2-yl]ethan-1-one
N-{1-[7-(2-cyclopentylacetyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-2-methylpropyl}oxolane-3-carboxamide
2-(carbamoylamino)-N,3-dimethyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}butanamide
methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}amine
(2S,4S)-1-[(4-chlorophenyl)methyl]-N-ethyl-4-{[(4-methoxy-3-methylphenyl)methyl]amino}pyrrolidine-2-carboxamide
5-fluoro-2-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
2-{[5-(2-cyanophenyl)furan-2-yl]methyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-{1-oxo-1-[4-(2-phenylethyl)piperidin-1-yl]propan-2-yl}methanesulfonamide
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(2,3-dimethyl-1H-indole-7-carbonyl)pyrrolidin-3-yl]methanol
7-(oxan-4-yl)-2-[2-(1H-1,2,3-triazol-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
6-fluoro-2-({2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}methyl)quinolin-4-ol
4-acetyl-N-cyclopentyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)benzamide
1-{1-[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]piperidin-4-yl}azepane
2-[1-(3-methylbut-2-en-1-yl)-4-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}piperazin-2-yl]ethan-1-ol
1-[2-methoxy-5-({[2-(pyridin-3-yl)ethyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
[(3S,5R)-1-[5-(methoxymethyl)furan-2-carbonyl]-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
2-cyclopropyl-N-ethyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}-6-oxo-1,6-dihydropyrimidine-5-carboxamide
2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}-1-[7-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
4-{1-methyl-3-[3-(1-methyl-1H-pyrazol-5-yl)phenyl]-1H-1,2,4-triazol-5-yl}morpholine
4-(cyclopropylmethyl)-3-(propan-2-yl)-1-[3-(pyridin-4-yl)-1H-pyrazole-5-carbonyl]-1,4-diazepan-5-one
(4aS,8aR)-6-[2-(propan-2-yloxy)acetyl]-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
1-[(2,6-difluorophenyl)methyl]-N-[2-(2,4-dimethoxyphenyl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-[1-(2-chlorophenyl)-5-oxopyrrolidin-3-yl]-6-methylimidazo[1,2-a]pyridine-2-carboxamide