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2-[5-(4-fluorophenyl)-2H-1,2,3,4-tetrazol-2-yl]-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}acetamide
2-ethyl-4-methyl-N-[1-(morpholin-4-ylmethyl)cyclopentyl]-1,3-oxazole-5-carboxamide
1-[1-(6-{2-azaspiro[4.4]nonan-2-yl}pyridine-3-carbonyl)piperidin-3-yl]-3-methylbutan-1-one
N-(cyclohexylmethyl)-4-hydroxy-2-phenylpyrimidine-5-carboxamide
N-[3-({[3-(4-methylpiperazin-1-yl)propyl]carbamoyl}amino)phenyl]cyclopentanecarboxamide
2-methyl-2-[4-(morpholin-4-yl)-2-[(oxan-4-ylmethyl)amino]pyrimidin-5-yl]propanoic acid
1-[4-(6-hydroxy-1,4-oxazepane-4-carbonyl)-3,5-dimethyl-1H-pyrrol-2-yl]ethan-1-one
2,7,8-trimethyl-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]quinoline-4-carboxamide
N-methyl-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]-5-propyl-1,2-oxazole-3-carboxamide
2-(2,3-difluoro-6-methoxyphenyl)-1-[(1-ethyl-1H-imidazol-2-yl)methyl]-1H-imidazole
2-{[2-(1-{6-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl)-1H-imidazol-1-yl]methyl}pyridine
[(3R,4R)-4-(piperidin-1-ylmethyl)-1-(thiophene-2-carbonyl)pyrrolidin-3-yl]methanol
(2S,4R)-1-[(3-ethoxy-4-hydroxyphenyl)methyl]-N-(2-methyl-1,3-benzothiazol-5-yl)-4-(pyridin-2-ylsulfanyl)pyrrolidine-2-carboxamide
1-[(4-chlorophenyl)methyl]-5-(thiomorpholine-4-carbonyl)piperidin-2-one
7-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
4,6-dimethyl-3-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
3-{2-[7-(2-chlorobenzamido)-1,2,3,4-tetrahydroisoquinolin-2-yl]-2-oxoethyl}-1,2,3-oxadiazol-3-ium-5-olate
ethyl 4-{6-[2-(2-phenyl-1,3-thiazol-4-yl)acetyl]-6-azaspiro[2.5]octane-1-carbonyl}piperazine-1-carboxylate
2-{[1-benzyl-3-(morpholine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-3-methylquinoxaline
2-methyl-N-{1-[1-(pyrimidin-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
2-(morpholin-4-yl)-1-[4-(2-phenylpyrimidin-4-yl)piperidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
1-{1-[(1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}ethan-1-ol
(2R,3S,6R)-3-phenyl-5-(3-propyl-1H-pyrazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(3-fluorobenzoyl)-2,8-diazaspiro[4.5]decan-3-one
1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-4-(3-phenylpropyl)-1,4-diazepane
2-[1-(1-cyclopentanecarbonylpiperidin-4-yl)-1H-1,2,3-triazol-4-yl]propan-2-ol
2-{2-[1-tert-butyl-3-(furan-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1-methylpiperidine
3-(3-hydroxy-3-methylbutyl)-N-{[4-(hydroxymethyl)oxan-4-yl]methyl}benzamide
4-(1-methyl-1H-pyrazol-4-yl)-1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,2,3,6-tetrahydropyridine
3-({[(3,4-dimethoxyphenyl)methyl]amino}methyl)-7-fluoro-N,N-dimethylquinolin-2-amine
4-{[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,4-triazol-5-yl]methyl}-1λ6-thiane-1,1-dione
1-cyclohexyl-4-{3-[(4-methylpiperidin-1-yl)methyl]imidazo[1,2-a]pyridine-2-carbonyl}piperazine
2-[(6-chloropyridin-3-yl)methyl]-2,7-diazaspiro[4.5]decane
N-{1-[1-(dimethyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-methoxybenzamide
1-(5-methoxy-2-methylphenyl)-3-[3-(methylsulfanyl)propyl]urea
2-[1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-4-methyl-1H-1,3-benzodiazole
ethyl 1-(cyclohex-3-ene-1-carbonyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
3,4-dimethyl-N-[(5-methyl-2-{3-[3-(pyridin-3-yl)propanamido]phenyl}-1,3-oxazol-4-yl)methyl]benzamide
{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)[(1-methylpyrrolidin-2-yl)methyl]amine
2-(4-methyl-1,3-thiazole-5-carbonyl)-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decane
5-[(2-methylphenyl)methyl]-1-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(4-{[(3R,4S)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]methyl}phenyl)ethan-1-one
2-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-(2-methylpropyl)-2-oxoacetamide
1-{1-ethyl-5-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}pyrrolidine
N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2-(pyridin-2-ylsulfanyl)propanamide
4-{1-[(trimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}benzoic acid
3-(dimethyl-1H-1,2,4-triazol-1-yl)-N,2-dimethyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
N,2,8-trimethyl-N-[1-(1,3-thiazol-5-yl)ethyl]quinoline-4-carboxamide
1-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(4-fluorophenoxy)ethan-1-one