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N-(adamantan-2-ylmethyl)-6-({methyl[1-(trimethyl-1H-pyrazol-4-yl)ethyl]amino}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
N-{1-[(3-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-4-oxo-3,4-dihydroquinazoline-2-carboxamide
2-[4-(1H-pyrazol-1-yl)phenyl]-2-[4-(thiophen-3-ylmethyl)piperazin-1-yl]acetic acid
{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[(3-methylthiophen-2-yl)methyl]amine
4,4,4-trifluoro-1-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]butan-1-one
1-methyl-3-(naphthalen-2-ylmethyl)-8-(oxan-4-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-cyclopropyl-4-[(2-methylprop-2-en-1-yl)oxy]-N-(1,3-thiazol-2-ylmethyl)benzamide
2-(1-methyl-1H-imidazol-2-yl)-1-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}piperidine
(1R,2S)-2-{1-benzyl-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}-N-methylcyclohexane-1-carboxamide
8-benzoyl-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-3-azaspiro[5.5]undecan-9-amine
N-{3-[4-({[5-(methoxymethyl)thiophen-2-yl]formamido}methyl)-5-methyl-1,3-oxazol-2-yl]phenyl}-1-methylpiperidine-3-carboxamide
benzyl N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}carbamate
N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine
1-(4-{[2-(cycloheptanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}piperazin-1-yl)ethan-1-one
6-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrole-2-carbonyl]-2-(4-fluorophenyl)imidazo[1,2-a]pyridine
(2S,4S)-4-amino-1-(5-phenyl-1,2-oxazole-3-carbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-(cyclopropylmethyl)-2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
2-[(6-{[(4-fluorophenyl)methyl](methyl)amino}pyridazin-3-yl)oxy]-1-{4-[(3-fluorophenyl)methyl]-1,4-diazepan-1-yl}ethan-1-one
3-(3-methoxy-1,5-dimethyl-1H-pyrazol-4-yl)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-1-propylurea
N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}-3-phenoxypropanamide
1-(2-methoxyethyl)-3-(2-methoxyphenyl)-3-{2-[4-(2-methylphenyl)piperazin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
3-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-3,9-diazaspiro[5.5]undecane
N-({6-[4-(methylsulfanyl)phenyl]pyridin-3-yl}methyl)acetamide
5-fluoro-2-{5-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-1,3-benzodiazole
2-fluoro-N-{[4-(2-methylpropoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)benzamide
1-[5-(methoxymethyl)thiophene-2-carbonyl]-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-(methoxymethyl)-N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-1H-pyrazole-4-carboxamide
1-[3-methoxy-4-(pyrrolidin-1-yl)phenyl]-2-(oxolan-3-yl)-1H-imidazole
methyl 1-({6-chloro-4-[(2-methoxyethyl)amino]quinazolin-2-yl}methyl)piperidine-2-carboxylate
1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethan-1-amine
3-(2-methoxyethyl)-1-[4-methyl-6-(methylamino)pyrimidin-2-yl]piperidine-3-carboxylic acid
1-[2-methyl-1-(pyrrolidin-1-yl)propan-2-yl]-3-(3-phenyl-1,2,4-thiadiazol-5-yl)urea
4-{5-[({1-[(2-fluorophenyl)methyl]piperidin-3-yl}(methyl)amino)methyl]thiophen-2-yl}-2-methylbut-3-yn-2-ol
2-ethoxy-6-{[3-(2-hydroxyethyl)-4-(thiophen-2-ylmethyl)piperazin-1-yl]methyl}phenol
5-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-N-methyl-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)-2-(trifluoromethyl)benzamide
(2E)-N-[1-(4-methyl-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]-3-(thiophen-2-yl)prop-2-enamide
2-{2-[3-(oxolan-2-ylmethyl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-1,3-benzodiazole
1-cyclohexanecarbonyl-N-(4-fluorophenyl)piperidin-3-amine
1-methyl-2-(morpholin-4-yl)-N-[1-(1,3-thiazol-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
1-{4-[({[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}(2-methoxyethyl)amino)methyl]thiophen-2-yl}ethan-1-one
3-methyl-4-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
1-(4-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)-3-phenylpropan-1-ol
(5-{[({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}-2-(propan-2-yloxy)phenyl)methanol
(2S,4R)-4-amino-N-methyl-1-{2-methyl-3-[(pyridin-2-ylmethyl)amino]benzoyl}pyrrolidine-2-carboxamide
4-(3-methyl-1H-pyrazole-5-carbonyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[1-(5-methoxypyrimidin-2-yl)piperidin-4-yl]-3-methylbutan-1-ol
1-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-2-ethoxyethan-1-one
9-(2,8-dimethylquinoline-3-carbonyl)-1,4,9-triazaspiro[5.5]undecan-5-one