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methyl (2S)-2-({1-[(2,6-difluorophenyl)methyl]-1H-1,2,3-triazol-4-yl}formamido)-3-methylbutanoate
3-({1-[(4-methylpiperazin-1-yl)methyl]cyclopropyl}methyl)-1-[3-(methylsulfanyl)phenyl]urea
N-[2-(dimethylamino)ethyl]-4-(quinolin-3-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-(propan-2-yl)-1-[(1s,4s)-4-(2-phenoxypropanamido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-[1-(2-phenylethyl)piperidin-3-yl]cyclopent-1-ene-1-carboxamide
1-{1,3-dioxo-2-[(trimethyl-1H-pyrazol-4-yl)methyl]-2,3-dihydro-1H-isoindol-4-yl}-N-[1-(furan-2-yl)ethyl]-N-methylpiperidine-4-carboxamide
5,7-dimethyl-N-[2-(piperidin-1-yl)butyl]pyrido[2,3-d]pyrimidin-4-amine
2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}-N-[2-(pyridin-3-yl)ethyl]acetamide
N-[1-(3,5-difluorophenyl)cyclopropyl]-4-(4H-1,2,4-triazol-4-yl)benzamide
ethyl 1-[2-(4-methoxyphenyl)ethyl]-5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1,9-dimethyl-4-{[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
5-[(2-fluoro-5-methoxyphenyl)methyl]-5-(3-{4-[(2-fluorophenyl)methyl]-1,4-diazepan-1-yl}-3-oxopropyl)pyrrolidin-2-one
N-[(3-methyl-1-benzofuran-2-yl)methyl]-6-(piperidin-3-yl)pyrimidin-4-amine
1-(2-cyclopropylacetyl)-4'-(3,3-dimethylbutyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
{[4-(3-methoxyphenyl)-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(methyl)(quinolin-8-ylmethyl)amine
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-6-methyl-2-(methylsulfanyl)pyrimidine
5-[(1,3-benzothiazol-2-ylmethyl)amino]-N,N-dimethyl-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(4aS,8aR)-N-(3-methyl-1,2,4-thiadiazol-5-yl)-decahydroisoquinoline-2-carboxamide
3-{5-[(2-fluorophenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1-(pyrrolidin-1-yl)propan-1-one
1-{3,5-dimethyl-4-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-1H-pyrrol-2-yl}ethan-1-one
1-(2-amino-5-butyl-6-methylpyrimidin-4-yl)-4-(1H-imidazol-1-ylmethyl)piperidin-4-ol
N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-1-methyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3-{[(2R)-oxolan-2-ylmethyl]sulfamoyl}benzamide
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(4-methoxy-3-methylphenyl)methyl]-N-(thiophen-3-ylmethyl)pyrrolidine-2-carboxamide
2-(oxolan-2-ylmethyl)-9-[2-(pyridin-2-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
3-(2,4-difluorophenyl)-6-(oxolane-2-carbonyl)-1-(pyridin-2-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-[(2-fluorophenyl)methyl]-3-hydroxy-3-{[(1-methylpiperidin-4-yl)amino]methyl}piperidin-2-one
N-(1-{4-[(1-benzothiophen-2-ylmethyl)(methyl)carbamoyl]phenyl}-1H-pyrazol-4-yl)furan-3-carboxamide
3,5-dimethoxy-N-{[7-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)benzamide
(3R,4R)-3-cyclopropyl-1-[5-fluoro-4-(methylamino)pyrimidin-2-yl]-4-methylpyrrolidin-3-ol
[(3R,4R)-1-[3-(3-fluorophenyl)benzoyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
1-(5-cyclopropyl-1,2-oxazole-3-carbonyl)-3-(4-phenylbenzoyl)piperidine
(3S,4R)-N,N-dimethyl-4-(4-methylphenyl)-1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-amine
N-{[7-chloro-5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-methyl-3-phenyl-1,2-oxazole-4-carboxamide
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-3-hydroxy-4-methoxybenzamide
4-[1-(2-methyl-1,3-benzothiazol-6-yl)-1H-1,2,4-triazol-5-yl]oxane-4-carbonitrile
N-(1-cycloheptylpiperidin-3-yl)-2-(6-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
4-[(4-methoxy-2,3,6-trimethylphenyl)methyl]-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
2-[methyl({[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl})amino]-6-(trifluoromethyl)pyridine-3-carboxamide
5-[(4-benzylpiperidin-1-yl)methyl]-N-methyl-N-(2-methylprop-2-en-1-yl)-1,2-oxazole-3-carboxamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-3-(3-methoxyphenyl)-N-methyl-1H-pyrazole-4-carboxamide
5-(1-benzofuran-2-yl)-N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-1,2,4-triazin-3-amine
6-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1,3-benzothiazole
2-amino-4-[5-(1H-pyrazol-3-yl)thiophen-2-yl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
3-(2,3-dihydro-1H-isoindol-2-yl)-1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)propan-1-one
N-[3-(furan-2-yl)propyl]-7-(oxolan-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
dimethyl(2-{2-[1-(quinoxaline-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)amine
2-(1H-indol-3-yl)-1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide