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N-methyl-5-(3-methyl-1,2,4-oxadiazol-5-yl)-N-(pyrimidin-4-ylmethyl)pyridin-2-amine
methyl({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}){[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
2-{[1-(4-methoxy-2,3-dimethylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-imidazole
N-[2-(2-fluorophenyl)ethyl]-5-[4-hydroxy-1-(2-methylpropyl)piperidin-4-yl]-1-benzofuran-2-carboxamide
1-[4-({3-[2-(methoxymethyl)piperidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)phenyl]ethan-1-one
N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
{2-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]quinolin-3-yl}methanol
3-({4-benzyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)-5-tert-butyl-1H-pyrazole
4-[3-(1,3-benzothiazol-2-yl)propanoyl]piperazine-2-carboxylic acid
{3-[(3-chlorophenyl)methyl]-1-(quinoline-8-sulfonyl)piperidin-3-yl}methanol
N-(2-methoxyethyl)-6-[2-(3-methoxyphenyl)pyrrolidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
2-[2-(1-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}piperidin-3-yl)-1H-imidazol-1-yl]acetamide
N,N-dimethyl-5-(5-phenyl-1,2-oxazole-3-carbonyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}cycloheptanecarboxamide
5-oxo-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
N-[4-(3-methylphenyl)phenyl]-1-[2-(1H-pyrazol-1-yl)acetyl]piperidine-4-carboxamide
N-[(3-ethenylphenyl)methyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
(4aS,7aR)-1-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-4-(2-methoxyacetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-cyclopropanecarbonyl-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)piperidine-4-carboxamide
1-(2-{1-oxa-7-azaspiro[3.5]nonan-7-yl}-2-oxoethyl)-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
ethyl 1-(cyclopropylmethyl)-5-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-(4-methoxyphenyl)-N-methyl-1H-pyrazole-3-carboxamide
3-{5-methylthieno[2,3-d]pyrimidin-4-yl}-1H-pyrazole
2-{4-[(1S,4S)-5-benzyl-2,5-diazabicyclo[2.2.1]heptane-2-carbonyl]-1H-1,2,3-triazol-1-yl}ethan-1-amine
8-(2-hydroxybenzoyl)-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{[2-(diethylamino)pyridin-3-yl]methyl}-3,4-dihydro-2H-1-benzopyran-2-carboxamide
N-[1-(furan-2-yl)ethyl]-N-methyl-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-1H-pyrazole-3-carboxamide
N-(1-{7-benzyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)-2-methoxyacetamide
1-[7-(3,6-dimethylpyrazin-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]but-3-en-1-one
N-{1-[(4-methylphenyl)methyl]cyclopropyl}-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
2-[2-(dimethylamino)ethyl]-9-[(3-methyl-1,2-oxazol-5-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-N-{3-[(4-methylphenyl)sulfanyl]propyl}imidazo[1,2-a]pyridine-6-carboxamide
1-(2-fluoro-4-methylbenzoyl)-4-phenoxypiperidine-4-carboxylic acid
ethyl 4-(cyclopropylmethyl)-1-[3-(2-methyl-1H-1,3-benzodiazol-1-yl)propanoyl]piperidine-4-carboxylate
6-(4-{[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-9H-purine
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2,4-dimethyl-1,3-oxazole-5-carboxamide
(3R,4S)-1-(3-chloro-2-fluorobenzoyl)-4-propylpyrrolidin-3-amine
N-[1-(4-fluorophenyl)propyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
N-{[1-(1H-indol-3-ylmethyl)piperidin-3-yl]methyl}-2,3-dimethoxybenzamide
3-cyclopropyl-N-[1-(3-fluorophenyl)-4-(morpholin-4-yl)-1H-indazol-3-yl]propanamide
4-[4-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2-methylquinoline
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
2-benzyl-N-(pyridin-3-yl)-1,3-thiazole-4-carboxamide
3-(furan-3-ylmethyl)-7,11-dimethyl-3,7,11-triazaspiro[5.6]dodecane
(2R,3S)-2-amino-3-methyl-1-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]pentan-1-one
4-(1-{4-[6-(thiomorpholin-4-yl)pyridazin-3-yl]phenyl}ethyl)morpholine
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-methyl-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
5-(azocane-1-carbonyl)-N-[1-(furan-2-yl)ethyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
methyl 5-[3-(naphthalene-2-carbonyl)piperidin-1-yl]-5-oxopentanoate
1-methyl-N-[(4-phenyloxan-4-yl)methyl]-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine