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2-({[(3-ethoxyphenyl)methyl](2-hydroxyethyl)amino}methyl)-4-fluorophenol
N-[2-(4-fluorophenyl)-2-hydroxyethyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
5-cyclobutanecarbonyl-3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
6-methoxy-3-{[methyl({[2-(methylamino)pyrimidin-5-yl]methyl})amino]methyl}-1,2-dihydroquinolin-2-one
N-{3-oxo-3-[1-(propan-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]propyl}methanesulfonamide
8-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decane
6-[(2R,3R)-2-hydroxy-3-(1H-imidazol-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]pyridine-3-carboxamide
1-{[3-(4-chlorophenyl)-1-(2-hydroxybutyl)-1H-1,2,4-triazol-5-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-cyclopentyl-1-(cyclopropylmethyl)-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-methyl-6-{9-methyl-3,9-diazaspiro[5.6]dodecan-3-yl}pyrimidin-4-amine
1-methyl-8-(2-phenylethyl)-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2S,4S)-4-amino-N-methyl-1-(5-methylpyridine-3-carbonyl)pyrrolidine-2-carboxamide
6-[2-(4-methanesulfonylphenyl)-1H-imidazol-1-yl]-1H-indazole
2-{9-[(2S)-2-hydroxy-3-phenylpropanoyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
3-{1-[2-(4-acetylphenoxy)acetyl]piperidin-4-yl}-1-(pyrrolidin-1-yl)propan-1-one
1-{7-[(4-acetylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-(naphthalen-1-yl)ethan-1-one
[(5-{1-[(4-chloro-2-fluorophenyl)methyl]piperidin-4-yl}-4-ethyl-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
[(3R,4R)-1-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
4,4,4-trifluoro-N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)butanamide
N-(6-methylpyridin-3-yl)-3-[(3-oxopiperazin-1-yl)methyl]benzamide
ethyl 1-{[2-(methoxycarbonyl)-3-(4-methylbenzamido)thieno[2,3-b]pyridin-6-yl]methyl}piperidine-4-carboxylate
(4S,6R)-6-methyl-N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-2-sulfanylidene-1,3-diazinane-4-carboxamide
2-{[4-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}ethan-1-ol
(3aR,6aR)-2-[(3-fluoro-4-methoxyphenyl)methyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amine
4-[3-(oxolan-3-yl)-5-(1H-pyrazol-4-yl)-1H-1,2,4-triazol-1-yl]benzonitrile
N-{1-[(4-fluorophenyl)methyl]-7-[4-(1-hydroxypropyl)piperidine-1-carbonyl]-1H-1,3-benzodiazol-5-yl}-2-methoxyacetamide
1-cyclohexyl-N-[(2-ethyl-4-methyl-1,3-thiazol-5-yl)methyl]piperidine-4-carboxamide
1-ethyl-5-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-3-(propan-2-yl)-1H-pyrazole
5-(2-methoxy-4-methylbenzoyl)-3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-[(3-methoxyphenyl)methyl]-1-propyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-{1-[2-(4-fluorophenyl)acetyl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
4-{[5-(hydroxymethyl)furan-2-yl]methyl}-6-[(3-methoxyphenyl)methoxy]-1-(2-methylpropyl)-1,4-diazepan-2-one
1-[2-(1-{3-[4-(dimethylamino)phenyl]propanoyl}piperidin-4-yl)ethyl]pyrrolidin-2-one
8-chloro-N-(1,4-dioxan-2-ylmethyl)-2-(furan-2-yl)quinoline-4-carboxamide
4-(furan-3-carbonyl)-6-[(3-methoxyphenyl)methoxy]-1-(2-phenylethyl)-1,4-diazepan-2-one
1-[(3-methoxyphenyl)methyl]-5-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazole
4-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(quinolin-5-yl)piperazine-1-carboxamide
6-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]quinazolin-4-amine
N-cyclopentyl-6-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)pyridine-3-carboxamide
N-[(3S,4R)-1-(3-fluoropyridine-4-carbonyl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
3-[3-(4-methyl-1,3-thiazol-2-yl)propyl]-1-[3-methyl-4-(2-oxopyrrolidin-1-yl)phenyl]urea
ethyl 4-(1-{[(4-phenyloxan-4-yl)methyl]carbamoyl}-6-azaspiro[2.5]octan-6-yl)piperidine-1-carboxylate
2-{1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carbonyl}-2-azaspiro[4.4]nonane
2-({2-amino-6-[4-fluoro-2-(trifluoromethyl)phenyl]pyrimidin-4-yl}amino)ethan-1-ol
3-(hydroxymethyl)-1-[4-(3-methylphenoxy)benzoyl]piperidin-3-ol
1'-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-({1-[3-(4-hydroxyphenyl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-yl}methyl)benzoic acid
ethyl 4-oxo-5-phenoxy-1-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,4-dihydropyridine-3-carboxylate
1'-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]