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N-{2-[4-(dimethylamino)phenyl]ethyl}-4-methylpyrimidine-5-carboxamide
9-[(3-chloro-4-fluorophenyl)methyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N,N-diethyl-2-{4-[(2S)-4-methyl-2-phenylpiperazine-1-carbonyl]-1H-1,2,3-triazol-1-yl}acetamide
4-[(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)amino]pyrimidine-5-carboxylic acid
(2S)-2-hydroxy-2-phenyl-1-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidine
4-{5-cyclopropyl-1-[4-(3-fluoro-4-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}morpholine
(2-{2-[1-(1H-indazole-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
5-(1-benzofuran-2-yl)-3-[3-(2,3-dimethoxyphenyl)pyrrolidin-1-yl]-1,2,4-triazine
N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-N-(2-hydroxyethyl)-N-methyl-5-(propan-2-yl)-1H-pyrazole-4-carboxamide
2-(dimethylamino)-N-(3-methoxypropyl)-N-(1-methylpiperidin-4-yl)-6-(thiophen-2-yl)pyridine-3-carboxamide
2-(4-methoxyphenoxy)-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]acetamide
2-{4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl}benzonitrile
3-fluoro-4-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
4-[5-(cyclopent-2-en-1-ylmethyl)-3-cyclopropyl-1H-1,2,4-triazol-1-yl]-2-methylpyridine
N-[1-(methoxymethyl)cyclopentyl]-6-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide
N-(3-acetylphenyl)-2-(2-phenylethyl)morpholine-4-carboxamide
2-(2-methoxyethyl)-8-(2,4,5-trimethylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
5-[(cyclopropylmethyl)amino]-1-ethyl-N-(furan-2-ylmethyl)-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
ethyl 5-{[2-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-5-oxopyrrolidin-1-yl]methyl}furan-2-carboxylate
3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-N-{[1,2,4]triazolo[4,3-a]pyridin-8-yl}propanamide
ethyl 4-[(4-methoxyphenyl)methyl]-1-(5-methyl-1,2-oxazole-3-carbonyl)piperidine-4-carboxylate
1-(2-phenoxyethyl)-4-(3,3,3-trifluoro-2-methylpropyl)piperazine
4-[1-(5-ethylpyrimidin-2-yl)azetidin-3-yl]morpholine
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-(2-methyl-5-oxopyrrolidin-1-yl)acetamide
N-(3-hydroxypropyl)-1-(1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide
(2S,4S,5R)-1,2-dimethyl-5-phenyl-4-{[2-(pyridin-3-yl)ethyl]carbamoyl}pyrrolidine-2-carboxylic acid
N-cyclopropyl-4-fluoro-N-{[1-(2-methylprop-2-en-1-yl)-1,2,5,6-tetrahydropyridin-3-yl]methyl}benzamide
3-chloro-6-[3-(2-fluorophenyl)pyrrolidin-1-yl]pyridine-2-carboxylic acid
1-{4-[(2-methylphenyl)methyl]piperazin-1-yl}-2-(methylsulfanyl)ethan-1-one
6-methyl-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]pyridine-3-carboxamide
{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}({[1-(pyrimidin-2-yl)piperidin-3-yl]methyl})amine
1-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-propyl-1H-1,2,4-triazole
N-[1-({5-[(4-methylphenyl)sulfanyl]furan-2-yl}methyl)pyrrolidin-3-yl]acetamide
N-[2-(dimethylamino)ethyl]-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)-3-(methylsulfanyl)propanamide
(2S,4R)-N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-4-hydroxypyrrolidine-2-carboxamide
N-({8-[(3,4-dimethoxyphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2-methoxyacetamide
(4S)-1-[(1-benzyl-1H-imidazol-2-yl)methyl]-3,3,4-trimethylpiperidin-4-ol
N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
2-({4-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]phenyl}sulfanyl)ethan-1-ol
1-{5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-4-(propan-2-yl)piperazine
N-ethyl-N-[(3S,4R)-4-hydroxyoxolan-3-yl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
3-{[1-(ethanesulfonyl)piperidin-4-yl]methyl}benzoic acid
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)cyclopentanecarboxamide
5-(cyclohexylamino)-1-methyl-N-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(3R,5S)-5-[(2,3-dihydro-1H-inden-5-yloxy)methyl]-1-(2-methylpropyl)-N-[3-(morpholin-4-yl)propyl]piperidine-3-carboxamide
1-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}-4-methylpiperazine
4-(1-benzofuran-2-yl)-7-[(dimethylsulfamoyl)amino]-1,2,3,4-tetrahydroquinolin-2-one
N-{[8-(naphthalen-1-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}oxane-4-carboxamide