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{6-[4-(adamantan-1-yl)piperazin-1-yl]-2-methylpyrimidin-4-yl}methanamine
2-{1-[(4-ethoxyphenyl)methyl]-4-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]-N-{[3-(trifluoromethoxy)phenyl]methyl}acetamide
(1S,6R)-9-{3-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]propanoyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
N-[(3-methyl-1-benzofuran-2-yl)methyl]-2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
3-{[(3,5-dimethoxyphenyl)methyl]amino}-N-[(1S)-1-phenylethyl]-5-[(propan-2-yl)sulfamoyl]benzamide
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
2-amino-4-(2-ethylpyrimidin-5-yl)-6-phenyl-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
3-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-5-{1-[(4-ethoxyphenyl)methyl]piperidin-4-yl}-5-ethylimidazolidine-2,4-dione
N-methyl-2-(2-methyl-1,3-thiazol-4-yl)-N-(1,2-oxazol-5-ylmethyl)acetamide
5-methyl-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-1,3,4-oxadiazol-2-amine
2-(2H-1,3-benzodioxol-5-yl)-2-[4-(pyridin-2-yl)piperazin-1-yl]acetic acid
4-[1-(5-methyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]-5-phenyl-2-(trifluoromethyl)pyrimidine
(3R,4R)-1-(4-methoxybenzoyl)-4-{[2-(3-methylpyridin-2-yl)ethyl]amino}pyrrolidin-3-ol
1-{4-[3-(2-hydroxyethyl)-4-[(4-methoxy-3-methylphenyl)methyl]piperazin-1-yl]piperidin-1-yl}ethan-1-one
4-(2,4-dioxoimidazolidin-1-yl)-N-methyl-N-[1-(thiophen-2-yl)ethyl]benzamide
methyl 3-[2-(naphthalen-1-ylmethyl)morpholin-4-yl]propanoate
(3R,4R)-1-[(6-chloro-2H-chromen-3-yl)methyl]-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
2-[1-(4-fluorophenyl)cyclopropanecarbonyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one
7-(cyclopropylmethyl)-2-(dimethyl-1,2-oxazole-4-carbonyl)-2,7-diazaspiro[4.5]decane
(2S,4R)-4-amino-1-(dimethyl-1,3-thiazole-5-carbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-(4-{[(2,3-difluorophenyl)methyl]amino}piperidin-1-yl)benzamide
(3aR,6aR)-2-cyclopentyl-5-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
methyl 8-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-[(4-methylphenyl)(pyridin-4-yl)methyl]propanamide
N-[(2R,3R)-1'-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]furan-2-carboxamide
[1-(2,3-dimethylbenzoyl)-3-[(4-fluorophenyl)methyl]piperidin-3-yl]methanol
(1S,6R)-N-(2-fluoro-5-methanesulfonamidophenyl)-3-methyl-4-oxo-3,9-diazabicyclo[4.2.1]nonane-9-carboxamide
ethyl 4-{5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-6-yl}piperidine-1-carboxylate
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-5-(3-fluorophenoxymethyl)-N-methyl-1H-pyrazole-3-carboxamide
2-[2-(1H-imidazol-4-yl)ethyl]-8-(1-methyl-1H-pyrazole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-(4-phenylpiperidin-1-yl)acetamide
2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-N-[2-(methylamino)ethyl]-1,3-oxazole-4-carboxamide
6-fluoro-4-[4-(3-oxo-3,4-dihydropyrazin-2-yl)piperazine-1-carbonyl]-1,2-dihydroquinolin-2-one
[(2S)-1-[4-(azocan-1-yl)-5-methylthieno[2,3-d]pyrimidine-6-carbonyl]pyrrolidin-2-yl]methanol
1-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]-2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidine
[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl][1-(morpholin-4-yl)propan-2-yl]amine
(2S)-N-{[4-fluoro-3-(trifluoromethyl)phenyl]methyl}-1-(piperidin-4-yl)pyrrolidine-2-carboxamide
3-(4-methyl-4H-1,2,4-triazol-3-yl)-N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]propanamide
3-fluoro-N-[(2R,3R)-2-methoxy-1'-(1,2-oxazole-5-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]benzamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(3-tert-butyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
2-(4-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl)ethan-1-ol
6-(3-chlorophenyl)-N-(2-hydroxyethyl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-[4-(4-{[3-(propan-2-yloxy)propyl]amino}piperidin-1-yl)benzoyl]piperidin-3-ol
3-[5-(5-methyl-1,2-oxazol-3-yl)-1,3,4-oxadiazol-2-yl]-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-1-methylazepane-2-carboxamide
5-(azetidin-1-ylmethyl)-2-(2-methoxyphenyl)-1,3-thiazole
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[2-(pyrrolidine-1-carbonyl)piperazin-1-yl]ethan-1-one
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-{3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}propan-1-one
1-(3-methyl-1H-pyrazole-5-carbonyl)-4-[(3-methylpyridin-2-yl)methyl]piperazine