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N-{[3-methyl-7-(4-oxo-4-phenylbutanoyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(phenylsulfanyl)acetamide
2-propyl-N-[1-(thiophen-2-ylmethyl)piperidin-4-yl]-1,3-thiazole-4-carboxamide
N-[(2-chlorophenyl)methyl]-3-{1-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}propanamide
1-(2-cyclohexylethyl)-N-methyl-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-1H-1,2,3-triazole-4-carboxamide
N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-1-phenyl-1H-1,2,3-triazole-4-carboxamide
1-[(diethylcarbamoyl)methyl]-N-[3-(1H-indol-1-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
N-({7-[(2E)-3-(3,4-dimethoxyphenyl)prop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-2-carboxamide
4-methoxy-N-({3-methoxy-4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]benzamide
2-(2,2-dimethylpropanoyl)-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
5-[(adamantan-1-ylmethyl)(methyl)amino]-1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]azepan-2-one
methyl 4-[5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carbonyl]piperazine-1-carboxylate
2-[3-(2-chlorophenyl)-1-(3-methoxypropyl)-2,5-dioxopyrrolidin-3-yl]-N,N-bis(prop-2-en-1-yl)acetamide
7-cyclopentyl-2-[1-(methoxymethyl)cyclobutanecarbonyl]-2,7-diazaspiro[4.5]decan-6-one
2-(5,6-dimethoxy-1-oxo-1,2-dihydroisoquinolin-2-yl)-N-methyl-N-(oxan-4-yl)acetamide
1-[2-(2,2-dimethyloxan-4-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-(thiophen-3-ylmethyl)piperidine-3-carboxamide
3-{1-[4-(4-fluorophenyl)oxane-4-carbonyl]azetidin-3-yl}pyridine
N,N-diethyl-2-({1-[(4-methoxyphenyl)methyl]-2-oxo-4-(quinoline-6-carbonyl)-1,4-diazepan-6-yl}oxy)acetamide
1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-8-propyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-6-methylpyrimidin-2-amine
N-cyclopropyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(1H-1,2,4-triazol-3-yl)benzamide
4-[(1-ethyl-1H-pyrazol-3-yl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
2-(1-{5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-1H-pyrazole-3-carbonyl}pyrrolidin-2-yl)-1,3-thiazole
5-fluoro-N,3-dimethyl-N-[2-(2-methyl-1H-indol-1-yl)ethyl]-1H-indole-2-carboxamide
3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}-N-(thiophen-2-ylmethyl)piperidine-1-carboxamide
4-{[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]methyl}benzonitrile
N-methyl-2,4-dioxo-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1,2,3,4-tetrahydropyrimidine-5-carboxamide
2-(2-chlorophenyl)-3-methyl-N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
1-methyl-N-[1-methyl-4-(propan-2-yloxy)-1H-indazol-3-yl]piperidine-3-carboxamide
2-{1-[1-(diphenylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperidin-2-yl}pyridine
4-[(1-acetylpiperidin-4-yl)oxy]-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3-methoxybenzamide
4-({[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}amino)-5-methylthieno[2,3-d]pyrimidine-6-carboxylic acid
3-(3,4-dimethoxyphenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
2-(2,3-dihydro-1H-indol-1-yl)-1-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]ethan-1-one
3-({2-[1-(4-methoxybenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-1-(6-ethoxy-4-methylquinazolin-2-yl)piperidin-4-amine
(3R,5S)-N-cyclohexyl-5-[(2,3-dihydro-1H-inden-5-yloxy)methyl]piperidine-3-carboxamide
(4aS,7aR)-1-(5-amino-1H-pyrazole-3-carbonyl)-4-[(5-methylfuran-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl][(2E)-2-methyl-3-phenylprop-2-en-1-yl]amine
(4aS,8aR)-6-[2-(3-methyl-6-oxo-1,6-dihydropyridazin-1-yl)acetyl]-1-propyl-decahydro-1,6-naphthyridin-2-one
1-(azocan-1-yl)-3-(2-methoxy-4-{[(prop-2-en-1-yl)(prop-2-yn-1-yl)amino]methyl}phenoxy)propan-2-ol
1-[4-(furan-2-ylmethoxy)phenyl]-3-methyl-3-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}urea
4-({1-[4-(pyrrolidin-1-yl)benzoyl]piperidin-2-yl}methyl)morpholine
N'-(2,3-dimethylphenyl)-N-[3-(1H-imidazol-1-yl)propyl]propanediamide
1-[(2-ethyl-1,3-thiazol-4-yl)methyl]-4-phenyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(3-{[(2H-1,3-benzodioxol-5-ylmethyl)amino]methyl}-2-methyl-1H-indol-1-yl)acetamide
5-methyl-5-[1-(2-methylbutyl)piperidin-4-yl]imidazolidine-2,4-dione
6-chloro-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}imidazo[2,1-b][1,3]thiazole-5-sulfonamide
methyl 4-[({[2-(piperidin-1-yl)-2,3-dihydro-1H-inden-2-yl]methyl}amino)methyl]benzoate
2-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}-1,2,3,4-tetrahydroisoquinolin-4-ol
1-(4-fluorobutyl)-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one