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5-{[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]methyl}-2,1,3-benzothiadiazole
N-[3-(4-{[2-(pyridin-3-yloxy)ethyl]amino}piperidin-1-yl)phenyl]-3-(trifluoromethyl)benzamide
1-butyl-2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1H-1,3-benzodiazole
N-{1-[(4-hydroxy-6-methylquinolin-2-yl)methyl]piperidin-4-yl}methanesulfonamide
4-[(4-fluorophenyl)methyl]-1-[2-(morpholin-4-yl)-2-oxoethyl]-3-(propan-2-yl)-1,4-diazepan-5-one
3-{1-[(2-methyl-1-benzothiophen-3-yl)methyl]piperidin-3-yl}propanamide
1-ethyl-3-[3-(pyridin-3-yl)propyl]-8-{[3-(trifluoromethyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-cyclobutyl-N-(thiophen-2-ylmethyl)-1,3,4-oxadiazol-2-amine
(1s,4s)-4-[4-(3,6-dimethylpyrazin-2-yl)piperazine-1-carbonyl]cyclohexan-1-ol
3-methyl-N-{1-[1-(3-phenylprop-2-ynoyl)piperidin-4-yl]-1H-pyrazol-5-yl}butanamide
1-[1-(1-ethyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
1-[3-({[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)propyl]piperidin-3-ol
[(2S,6S)-4-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
3-(4-methyl-1,3-thiazol-5-yl)-1-[4-(thiomorpholin-4-yl)piperidin-1-yl]propan-1-one
8-[2-(morpholin-4-yl)acetyl]-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
1-({4-[(2,4-dimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)-N,N-diethylpiperidine-3-carboxamide
6-(2-chlorophenyl)-N-cyclobutyl-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-(2-methyl-5-propylpyrimidin-4-yl)piperidine-3-carboxamide
1-tert-butyl-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-1H-pyrrole-3-carboxamide
N-({1-[(3-chloro-4-hydroxy-5-methoxyphenyl)methyl]piperidin-3-yl}methyl)-4-fluorobenzamide
2-(2-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}ethoxy)ethan-1-ol
N-[(3R,4S)-4-cyclopropyl-1-(2-hydroxyethyl)pyrrolidin-3-yl]-1-ethyl-5-methyl-1H-pyrazole-4-carboxamide
8-[(2S,3R)-2-amino-3-hydroxybutanoyl]-3-[3-(4-ethylpiperazin-1-yl)propyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-(3-{[(2,3-dihydro-1H-inden-2-yl)amino]methyl}pyrrolidin-1-yl)-2-methyl-2,3-dihydropyridazin-3-one
(1S,5R)-3-[(5-propylfuran-2-yl)methyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-{3-[(dimethylamino)methyl]-3-hydroxypiperidin-1-yl}-4-phenylbutan-1-one
1-(carbamoylmethyl)-N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)piperidine-3-carboxamide
1-[2-(4-chlorophenyl)ethyl]-N-methyl-6-oxo-N-(pyrazin-2-ylmethyl)piperidine-3-carboxamide
1-[1-(5-methylhex-5-en-2-yl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
4-[1-(3,4-dimethylbenzoyl)piperidin-4-yl]-5-(2-methylphenyl)-2-(pyridin-3-yl)pyrimidine
3-[1-(furan-2-ylmethyl)-1H-pyrazol-5-yl]-1-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}urea
(3R,5R)-N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
1-[(3,5-dimethylphenyl)methyl]-4-[4-(2-oxopyrrolidin-1-yl)butanoyl]piperazin-2-one
3-(2-ethyl-1H-imidazol-1-yl)-1-[7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]propan-1-one
1-(cyclopropylmethyl)-4-(1-methyl-1H-pyrazole-3-carbonyl)-2-(propan-2-yl)-1,4-diazepane
(1R,5R)-6-benzyl-3-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-3,6-diazabicyclo[3.2.2]nonane
methyl({[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl})[(3-methylthiophen-2-yl)methyl]amine
5-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
3-{[(2,4-dimethylphenyl)methyl]amino}-5-(phenylsulfamoyl)-N-(pyridin-3-ylmethyl)benzamide
N-(3-methyl-1-{7-[(2,4,5-trimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)furan-2-carboxamide
5-[ethyl(2-methylprop-2-en-1-yl)amino]-N,N-dimethyl-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}({[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl})amine
2-(3-phenyl-1H-pyrazol-1-yl)-N-[1-(propan-2-yl)-1H-pyrazol-5-yl]acetamide
(1S,5R)-3-[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(3-methyl-1,2,4-thiadiazol-5-yl)-1-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}urea
3-{[({2-[(dimethylamino)methyl]phenyl}methyl)(methyl)amino]methyl}pyridin-2-amine
(4aS,7aR)-1-{2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]-5-methoxyphenol
N-[(3S,4R)-4-(4-methylphenyl)-1-{thieno[2,3-d]pyrimidin-4-yl}pyrrolidin-3-yl]acetamide