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(4aS,8aR)-1-(4-hydroxybutyl)-6-(1H-indol-5-ylmethyl)-decahydro-1,6-naphthyridin-2-one
1-ethyl-8-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-(pyridin-3-yl)-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one
N-methyl-2-oxo-N-[1-(1,3-thiazol-5-yl)ethyl]-1,2-dihydroquinoline-4-carboxamide
N,N-dimethyl-5-(quinoxaline-5-carbonyl)-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
N-methyl-5-(morpholin-4-ylmethyl)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}furan-3-carboxamide
4-(2H-1,3-benzodioxol-5-ylmethyl)-7-{[4-(4-fluorophenyl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
N3-(cyclohexylmethyl)-N5-cyclooctyl-1-(2-methoxyethyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
5-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-5,6,7,8-tetrahydroquinoline
5-(2-methyl-1H-imidazol-4-yl)-1-(2-phenoxyethyl)-4-phenyl-1H-imidazole
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)benzamide
2-{1-[(6-methylquinolin-5-yl)methyl]piperidin-2-yl}acetamide
5-hydroxy-N-[(1R,3S)-3-(thiomorpholine-4-carbonyl)cyclopentyl]pyrazine-2-carboxamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine
3-(benzenesulfonyl)-N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}propanamide
{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[(5-propyl-1H-pyrazol-3-yl)methyl]amine
(1R,5R)-6-(cyclobutylmethyl)-3-[1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
3-(3-hydroxy-1,2-oxazol-5-yl)-1-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]propan-1-one
4-benzyl-3-ethyl-1-(1,3-thiazol-2-ylmethyl)-1,4-diazepan-5-one
1-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-4-(4-methoxyphenyl)piperazine
N3-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-N5-ethyl-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
5-(1H-imidazol-2-yl)-2-(2-methylphenyl)-1,3-thiazole
2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-methylacetamide
3-(2-amino-1,3-thiazol-4-yl)-1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]propan-1-one
N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1-[2-(2-methoxyphenyl)ethyl]-2,6-dimethyl-4-oxo-1,4-dihydropyridine-3-carboxamide
N-cyclopropyl-4-(hydroxymethyl)-N-[(2-methoxyphenyl)methyl]benzamide
2-ethyl-5-{3-[(1-methylpiperidin-4-yl)methyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl}pyrimidine
N,N-dimethyl-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
N-cyclopropyl-3-{1-[(3,4-difluorophenyl)methyl]piperidin-3-yl}propanamide
1-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}-2-(3-hydroxypiperidin-1-yl)ethan-1-one
N-[(2-propyl-1,3-thiazol-4-yl)methyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
3,5-dimethoxy-N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1-ethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
2-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl](methyl)amino}-2-(4-fluoro-3-methylphenyl)acetic acid
1-[(2-chlorophenyl)methyl]-N-(oxan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
4-{1-[3-(2-methoxyphenyl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}morpholine
3-chloro-N-(2-methoxyethyl)-4-{[1-(1-phenoxypropan-2-yl)piperidin-4-yl]oxy}benzamide
2-[(4aR,7aS)-4-[(3,4-dimethylphenyl)carbamoyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
N-[(2-chloro-6-fluorophenyl)methyl]-5-[(4-methylpiperazin-1-yl)methyl]furan-2-carboxamide
1-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-5-(thiophene-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[(3R,4R)-1-[(2,4-dimethylphenyl)methyl]-3-hydroxypiperidin-4-yl]pyridine-4-carboxamide
5-(2-{[(4-methoxyphenyl)methyl]amino}ethyl)-1-[(3-methylphenyl)methyl]pyrrolidin-2-one
N-methyl-1-[(4-methylthiophen-2-yl)sulfonyl]-N-[2-(pyridin-2-yl)ethyl]piperidin-3-amine
[3-(cyclopropylmethyl)-1-[1-(2-fluorophenyl)cyclopropanecarbonyl]piperidin-3-yl]methanol
5-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]ethan-1-one
2-methyl-5-(3-methylphenyl)-4-[1-(5-phenoxyfuran-2-carbonyl)piperidin-3-yl]pyrimidine
N-(2-hydroxyethyl)-2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
1-(2-methoxyphenyl)-4-(1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-3-yl)piperazine