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3-(3-phenyl-1,2,4-oxadiazol-5-yl)-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]propanamide
1-(1H-imidazol-4-ylmethyl)-4-(1H-1,2,3-triazol-4-ylmethyl)-1,4-diazepane-6-carboxylic acid
9-(2-methoxyethyl)-1-methyl-4-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
2-[(6-{[(4-fluorophenyl)methyl](methyl)amino}pyridazin-3-yl)oxy]-N-{[2-(trifluoromethyl)phenyl]methyl}acetamide
3-(2-methyl-1H-1,3-benzodiazol-1-yl)-5-(morpholine-4-sulfonyl)benzoic acid
2-(3-hydroxypropyl)-9-(2-methoxy-5-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(2,3-dihydro-1H-inden-2-yl)-2-(pyridin-3-yl)acetamide
4-(5-chloro-6-oxo-1,6-dihydropyridine-3-carbonyl)-3-methyl-1-(2-methylpropyl)piperazin-2-one
N-(2H-1,3-benzodioxol-5-yl)-6-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-6-azaspiro[2.5]octane-1-carboxamide
(4aS,7aR)-N-(3,4-dimethylphenyl)-4-(2-methylpropyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propanamide
N4-[1-(2,5-dimethoxyphenyl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
2-chloro-6-methoxy-4-{[propyl(pyridin-3-ylmethyl)amino]methyl}phenol
1-{1-[(2-methoxyphenyl)methyl]piperidin-4-yl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
7-fluoro-3-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-benzofuran-2-carboxamide
4-[2-(4-acetylphenoxy)acetyl]-1-(3-methoxyphenyl)-6-methylpiperazin-2-one
1-[2-amino-6-(cyclopropylamino)pyrimidin-4-yl]-1,4-diazepan-5-one
N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
2-methyl-4-(4-{7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decane-2-carbonyl}phenyl)but-3-yn-2-ol
1-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}-2,3,4,9-tetrahydro-1H-carbazole
3-({[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl](methyl)amino}methyl)-6-methoxy-1,2-dihydroquinolin-2-one
methyl 2-[4-(thiophen-2-ylmethyl)-1,4-diazepane-1-carbonyl]piperidine-1-carboxylate
ethyl 4-{1-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]piperidin-3-yl}piperazine-1-carboxylate
4-methoxy-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
1-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]-3-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propan-1-one
N-[(1R,3R)-3-aminocyclopentyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
methyl 3-(1H-indole-6-carbonyl)-7-oxo-9-[2-(thiophen-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(4-chlorophenyl)-N-{1-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}cyclobutane-1-carboxamide
4-[(methylsulfanyl)methyl]-N-[4-(oxolan-2-ylmethoxy)phenyl]piperidine-1-carboxamide
2-(2-methoxyethyl)-N-[2-(piperidin-1-yl)ethyl]-1,3-benzoxazole-6-carboxamide
3-[(4-methanesulfonylphenyl)methyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran
4-[3-(2-cyclopentylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1-(propan-2-yl)-1H-pyrazole
1-amino-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}cyclopropane-1-carboxamide
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-one
N-(1-{1-[(3,4-dimethoxyphenyl)methyl]piperidin-4-yl}-2-phenylethyl)-N,1,3-trimethyl-1H-pyrazole-5-carboxamide
(2E)-3-(2-fluorophenyl)-N-{[3-methyl-7-(4-phenylbutanoyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}prop-2-enamide
1-[2-(3,4-dimethoxyphenyl)ethyl]-5-(2-{[(3-methoxyphenyl)methyl]amino}ethyl)pyrrolidin-2-one
1-methyl-N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-(3-methoxybenzenesulfonyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
(2S,4R)-1-{[3-(benzyloxy)phenyl]methyl}-N-[(4-methylphenyl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
1-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
3-(1H-imidazol-1-ylmethyl)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine
(1S,5R)-6-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-{1-[2-(difluoromethoxy)benzoyl]piperidin-4-yl}piperidin-4-ol
3-(2-ethylphenoxy)-1-(5-fluoro-2-methoxybenzoyl)azetidine
3-[3-(3-methoxypropyl)piperidine-1-carbonyl]-6-(trifluoromethyl)pyridin-2-ol
1-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-3-yl]-2-(4-methoxyphenoxy)ethan-1-one
3-[(5,8-dimethoxy-4-methylquinolin-2-yl)(methyl)amino]propan-1-ol
1-[(5-chloro-2,4-dimethoxyphenyl)methyl]-3-ethylpiperidine-3-carboxylic acid
N-methyl-N-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}oxolan-3-amine