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2-[2-(dimethylamino)phenyl]-5-fluoro-N,N-dimethylpyrimidin-4-amine
1-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-3-(2-chlorophenyl)propan-1-one
N-[(3,4-dimethoxyphenyl)methyl]-N-(pyridin-3-ylmethyl)propanamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-(1,2,3-thiadiazole-4-carbonyl)piperidin-3-amine
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1,3-thiazol-2-ylmethyl)piperidine
4-phenyl-5-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]pyrimidin-2-amine
N-(cyclopropylmethyl)-3-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}benzamide
(1S,9S)-11-{1H-pyrrolo[2,3-b]pyridin-6-yl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
4-phenyl-1-(prop-2-yn-1-yl)-5-(thiophen-3-yl)-1H-imidazole
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-2-(trifluoromethyl)-1H-1,3-benzodiazole-5-carboxamide
3-[1-(adamantan-2-yl)piperidin-4-yl]-N-(3-methoxyphenyl)propanamide
5-oxo-1-(propan-2-yl)-N-[1-(pyridine-4-carbonyl)piperidin-4-yl]pyrrolidine-3-carboxamide
(1S,5R)-6-[(4-methoxypyridin-2-yl)methyl]-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
3-(2-fluorophenoxymethyl)-1-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
[4-({1-[3-(4-fluorophenyl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-yl}methyl)phenyl]methanol
4-[3-(1H-pyrazol-4-yl)benzoyl]thiomorpholine
(2,1,3-benzoxadiazol-5-ylmethyl)({[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl})methylamine
3-(1-methylpiperidin-2-yl)-1-[4-(pyrimidin-2-yl)piperazin-1-yl]propan-1-one
ethyl 3-[5-(2,1,3-benzoxadiazol-4-yl)-4-phenyl-1H-imidazol-1-yl]propanoate
2-[4-(1H-imidazol-2-ylmethyl)piperazin-1-yl]pyridine-3-carbonitrile
1-[(2-cyanophenyl)methyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
2-methyl-9-[6-(trifluoromethyl)pyridin-2-yl]-2,9-diazaspiro[5.5]undecan-3-one
2-cyclopropyl-9-(4-propylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
1-cyclopropanecarbonyl-4-(6-methoxypyrimidin-4-yl)-1,4-diazepane
N,N-dimethyl-3-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine-1-carbonyl}piperidine-1-carboxamide
8-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(2S,4R,6S)-2-benzyl-6-(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)oxan-4-yl]acetamide
3-(2,3-dihydro-1H-inden-2-yl)-8-[3-(5-methylfuran-2-yl)butyl]-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-ethyl-3-{1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{5-[(2-ethylphenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}benzonitrile
3-cyclopentyl-N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
2-(3-butyl-4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)acetamide
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-5-(1H-pyrazol-1-ylmethyl)furan-2-carboxamide
4-(1,3-benzothiazol-2-yl)-2-({[(4-methoxyphenyl)methyl]amino}methyl)phenol
2-(1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}piperidin-2-yl)acetamide
(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-6-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-(5-fluoro-2-methoxyphenyl)-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
N-methyl-N-{2-phenyl-1-[1-(1-phenyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]ethyl}-2-(1H-pyrazol-1-yl)acetamide
1-[(4-hydroxyphenyl)methyl]-N-[3-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
3-[2-oxo-2-(4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidin-1-yl)ethyl]-1,3-oxazolidin-2-one
3-{2-amino-4-[(3S,4S)-3-hydroxy-4-(morpholin-4-yl)pyrrolidin-1-yl]-6-methylpyrimidin-5-yl}propanoic acid
1-[5-(methoxymethyl)thiophene-2-carbonyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
3-(8-fluoro-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-1-[2-(2,4,6-trimethylphenoxy)ethyl]urea
4-chloro-3-{[4-(2-methoxyethoxy)piperidin-1-yl]methyl}-1-methyl-1H-indazole
4-{2-methylthieno[2,3-d]pyrimidin-4-yl}-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-{[4-(2,6-dimethylpyrimidine-4-carbonyl)-2-oxo-1-(2-phenylethyl)-1,4-diazepan-6-yl]oxy}-N,N-diethylacetamide
methyl 3-[(2-cyclohexylacetamido)methyl]-5-(furan-2-amido)benzoate
N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
(2S,4S)-4-amino-N-ethyl-1-{2-[4-(2-oxoimidazolidin-1-yl)phenyl]acetyl}pyrrolidine-2-carboxamide
2-(cyclohex-1-ene-1-carbonyl)-7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decane