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N-[(5-methyl-2-{3-[3-(pyridin-3-yl)propanamido]phenyl}-1,3-oxazol-4-yl)methyl]-5-(2-methylpropyl)-1,2-oxazole-3-carboxamide
N-(2-{7-[(5-ethylfuran-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclobutanecarboxamide
1-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-4-phenylazepane
(1S,5R)-6-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-[2-(azepan-1-yl)-2-phenylethyl]-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
S-[2-(2,2-dimethylpropanoyl)-1,2,3,4-tetrahydroisoquinolin-6-yl]-3-hydroxybutane-1-sulfonamido
(1R,2R)-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-2-phenylcyclopropane-1-carboxamide
1-(cyclohexylmethyl)-5-[4-(hydroxymethyl)piperidine-1-carbonyl]piperidin-2-one
N-[1-(2-chlorophenyl)ethyl]-1-methyl-4-oxo-1,4-dihydroquinoline-3-carboxamide
3-hydroxy-1-(2-phenylethyl)-3-({[2-(1H-1,2,3,4-tetrazol-5-yl)ethyl]amino}methyl)piperidin-2-one
(2S,4R)-4-cyclobutaneamido-N,N-diethyl-1-(1-methyl-1H-pyrrole-2-carbonyl)pyrrolidine-2-carboxamide
N,N-dimethyl-6-({1-[methyl(pyridin-3-ylmethyl)amino]hex-5-en-2-yl}oxy)pyridazin-3-amine
N-[(3,4-difluorophenyl)methyl]-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
4-ethyl-N-[(5-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-1,2,3-thiadiazole-5-carboxamide
1-methyl-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-2-(1H-pyrazol-1-yl)acetamide
2-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)-N,N-dimethylaniline
1-methyl-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-6-oxo-1,6-dihydropyridazine-3-carboxamide
4-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-4-oxobutanamide
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-2-(2-oxopyrrolidin-1-yl)propanamide
methyl[3-(1H-pyrazol-1-yl)propyl]{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}amine
N-[(3-chlorophenyl)methyl]-3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
(3-{2-[1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
6-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carbonitrile
1-(2-phenoxyethyl)-4-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
1-(1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}piperidin-4-yl)-2-(methoxymethyl)-5-(trifluoromethyl)-1H-1,3-benzodiazole
8-methoxy-2-{[3-(3-methoxybenzoyl)piperidin-1-yl]methyl}quinoline
{2-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]-2-oxoethyl}urea
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-methyl-N-[2-(4-methylphenoxy)ethyl]propanamide
1-[2-(dimethylamino)benzoyl]-N-(4-fluorophenyl)piperidin-3-amine
5-({3-oxo-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-9-yl}methyl)-1,2,4-oxadiazole-3-carboxamide
N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-2-methylbenzamide
9-methoxy-3-[(3-methylthiophen-2-yl)methyl]-7-oxo-N-[3-(1H-pyrazol-1-yl)propyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4-[(1,2-oxazol-3-ylmethyl)sulfamoyl]-N-(pyridin-3-yl)benzamide
N,N-dimethyl-1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]azepan-4-amine
3-(1-{1-[2-(2-methoxyphenyl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(2-methylphenyl)urea
{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
2,8-dimethyl-N-[4-(pyridin-2-yl)butyl]quinoline-4-carboxamide
N,1-dimethyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrrole-2-carboxamide
(2S,4R)-4-(dimethylamino)-N-(2,5-dimethylphenyl)-2-(hydroxymethyl)pyrrolidine-1-carboxamide
methyl 4-{[2-(aminomethyl)piperidine-1-carbonyl]amino}-2-chlorobenzoate
3-(4-ethyl-1H-pyrazol-5-yl)-1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]piperidine
6-methoxy-N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
({5-[1-(2,5-dimethylfuran-3-carbonyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
methyl 6-(1-methylcyclopropanecarbonyl)-2-[(3-methylphenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[3-(azepan-1-yl)propyl]-N-methylpyrimidin-4-amine
1-(methoxymethyl)-N-{[3-(trifluoromethoxy)phenyl]methyl}cyclobutane-1-carboxamide
methyl 1-(2-{[cyclohexyl(prop-2-yn-1-yl)amino]methyl}-6,7-dimethoxyquinazolin-4-yl)piperidine-4-carboxylate
N-[2-({[1-(2-carbamoylethyl)-1H-indol-3-yl]methyl}amino)ethyl]pyridine-3-carboxamide
4-{[1-(4-cyclobutyl-6-methylpyrimidin-2-yl)piperidin-4-yl]methyl}morpholine