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7-[(3-methylphenyl)methyl]-2-(1H-pyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-methyl-3-(2-methylphenyl)-3-phenyl-N-(1,3-thiazol-2-ylmethyl)propanamide
2-[2-(4-carbamoylphenyl)pyrimidin-4-yl]pyridine-4-carboxylic acid
N-[1-(cyclohex-1-en-1-yl)ethyl]-2-methoxyquinoline-4-carboxamide
2-methyl-7-{4-[4-(propan-2-yl)phenyl]butanoyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(2S,4R)-1-cyclopentyl-N,N-diethyl-4-[2-(3-methyl-1,2-oxazol-5-yl)acetamido]pyrrolidine-2-carboxamide
(1s,4s)-4-[4-(2,3-dihydro-1H-isoindole-2-carbonyl)-1H-1,2,3-triazol-1-yl]cyclohexan-1-amine
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-8-fluoroquinoline-2-carboxamide
1-(7-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-3-(thiophen-2-yl)propan-1-one
5-(2,6-dimethylphenoxymethyl)-N-(3-phenylpropyl)-1,2-oxazole-3-carboxamide
N-(1-benzylpyrrolidin-3-yl)-3-{1-[(dimethylcarbamoyl)methyl]piperidin-4-yl}propanamide
4-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-5-methyl-N-[2-(pyridin-2-yl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
2-amino-6-(2-amino-4-methyl-1,3-thiazol-5-yl)-4-(cyclohex-3-en-1-yl)pyridine-3-carbonitrile
[3-(1H-imidazol-1-yl)propyl](pyridin-4-ylmethyl)(quinolin-4-ylmethyl)amine
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-{2-[(dimethylcarbamoyl)amino]acetyl}pyrrolidine-3-carboxylic acid
(1S,5R)-3-(4,6-dimethylpyridine-3-carbonyl)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(2-methoxy-6-{[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]methyl}phenoxy)propanoic acid
N-[4-(2-methoxyphenyl)-1,3-dimethyl-1H-pyrazol-5-yl]-3,4-dihydro-2H-1-benzopyran-2-carboxamide
2-[6-(1-hydroxyethyl)pyridin-2-yl]-6-methoxy-N,N-bis(propan-2-yl)benzamide
8-[(2-aminopyridin-3-yl)methyl]-2-[(4-chlorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
4-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1λ6-thiomorpholine-1,1-dione
2-[5-(1-{pyrazolo[1,5-a]pyridine-3-carbonyl}pyrrolidin-2-yl)-1,2,4-oxadiazol-3-yl]pyridine
2-(2-{1-[2-(pyrimidin-2-ylsulfanyl)acetyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-5-phenyl-1,2-oxazole-3-carboxamide
N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1,2-oxazole-3-carboxamide
{[1-(cyclohexylmethyl)-2-methanesulfonyl-1H-imidazol-5-yl]methyl}(methyl)[1-(trimethyl-1H-pyrazol-4-yl)ethyl]amine
1-{3-[3-(4-methylpiperazin-1-yl)-3-oxopropyl]piperidin-1-yl}-3-(methylsulfanyl)propan-1-one
N-[(5-methylthiophen-2-yl)methyl]-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
1-[6-(2,3-dimethoxyphenyl)-1,2,3,4-tetrahydroquinolin-1-yl]ethan-1-one
1-(oxolan-2-ylmethyl)-4-[2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]piperazine
4-(3-ethoxypropanoyl)-5-methyl-1-(2-methylphenyl)piperazin-2-one
3-methyl-N-[2-(3-{[methyl(quinolin-8-ylmethyl)amino]methyl}phenoxy)ethyl]thiophene-2-carboxamide
N-(1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}piperidin-4-yl)methanesulfonamide
3-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-1-[4-methyl-3-(propan-2-yl)phenyl]urea
N-[(2-phenoxypyridin-3-yl)methyl]-2-(propan-2-yl)pyrimidine-5-carboxamide
2-(2-methoxyphenyl)pyridine-3-carbonitrile
2-(2,6-dimethoxyphenyl)-5,6-dimethylpyridine-3-carboxamide
(1S,4S)-5-[1-(4-chlorophenyl)cyclopropanecarbonyl]-2-(2-methoxy-5-methylphenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
N'-({1-[(4-methoxy-2,5-dimethylphenyl)methyl]piperidin-3-yl}methyl)ethanediamide
N-(2-{3-[3-(4-fluorophenyl)oxolan-3-yl]-1,2,4-oxadiazol-5-yl}propan-2-yl)aniline
5-methyl-4-{methyl[2-(pyridin-2-yl)ethyl]amino}-N-(3-methylbutyl)thieno[2,3-d]pyrimidine-6-carboxamide
3-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-triene-4-carbonyl]-2-methyl-4,5,6,7-tetrahydro-1-benzofuran-4-one
2-[3-(pyrrolidin-1-yl)piperidine-1-carbonyl]-1,4-dihydroquinolin-4-one
N-(1-methylpiperidin-4-yl)-2-(2-oxo-1,2-dihydropyridin-1-yl)-N-(2-phenylethyl)acetamide
N-[(3S,7S,8aS)-3-[(benzyloxy)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-tert-butyl-1-methyl-1H-pyrazole-5-carboxamide
N-[3-chloro-2-(4-ethylpiperazin-1-yl)phenyl]-2-(pyrrolidin-1-yl)acetamide
3-[2-(4-cyclohexyl-3-oxopiperazin-1-yl)-2-oxoethyl]-1-methyl-3-(4-phenylphenyl)pyrrolidine-2,5-dione
2-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}acetic acid
2-(3,5-dimethylphenyl)-2-{methyl[3-(morpholin-4-yl)propyl]amino}acetic acid