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N-(2-{[4-hydroxy-2-(4-methylphenyl)pyrimidin-5-yl]formamido}ethyl)-2-methylpropanamide
5-(methoxymethyl)-N-[(2-methoxyphenyl)methyl]-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
ethyl 1-(1-benzofuran-2-ylmethyl)-3-(2-methoxyethyl)piperidine-3-carboxylate
N4-[1-(4-ethoxy-3-fluorophenyl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
2-[3-(furan-2-yl)-5-[(2S)-1-methanesulfonylpyrrolidin-2-yl]-1H-1,2,4-triazol-1-yl]-6-methylpyridine
3-(1H-imidazol-1-yl)-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}propanamide
1-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-3-(2-ethyl-1H-imidazol-1-yl)propan-1-one
3-(2-methoxyethyl)-3-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-(2,3,4-trifluorophenyl)urea
1-[2-(methoxymethyl)piperidin-1-yl]-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propan-1-one
2-amino-4-[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]-6-(1-methyl-1H-pyrrol-3-yl)pyridine-3-carbonitrile
3-(4-methyl-1,3-thiazol-5-yl)-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]propanamide
6-(1-methyl-1H-imidazol-2-yl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}pyridazin-3-amine
5-(2,4-dimethoxyphenyl)-N-{[2-(trifluoromethoxy)phenyl]methyl}-1,2,4-triazin-3-amine
4,4,4-trifluoro-N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)butanamide
4-(3-hydroxy-3-methylbutyl)-N-[2-(pyridin-2-ylsulfanyl)ethyl]benzamide
3-(2-methyl-1H-imidazol-1-yl)-1-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
9-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-2-cyclopropyl-2,9-diazaspiro[5.5]undecan-3-one
N-{[5-methyl-7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(1H-pyrazol-1-ylmethyl)benzamide
3-fluoro-N-({7-[(2-fluoro-5-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzamide
2-(cyclopent-2-en-1-yl)-1-[4-(4-hydroxypiperidin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]ethan-1-one
2-[(4-methoxyphenyl)methyl]-N-(propan-2-yl)-1,3-benzoxazole-6-carboxamide
2-({[5,8-dimethoxy-2-(3-methylphenyl)quinolin-3-yl]methyl}(methyl)amino)ethan-1-ol
methyl 2-(3-{[benzyl(methyl)amino]methyl}-7-chloro-2-oxo-1,2-dihydroquinolin-1-yl)acetate
2-{2-[(dimethylamino)methyl]phenyl}-N,6-dimethylpyrimidin-4-amine
{4-[(1-{[3-(morpholin-4-yl)phenyl]methyl}pyrrolidin-3-yl)methyl]phenyl}methanol
1-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-1-methyl-3-(3-phenyl-1,2,4-thiadiazol-5-yl)urea
3-[1-(1-cyclopropylethyl)-1H-pyrazol-5-yl]-1-methyl-1-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}urea
2-(1-methyl-1H-imidazol-2-yl)-1-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-1-cyclohexyl-1H-1,2,3-triazole-4-carboxamide
(4S,4aS,8aR)-1-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}-4-phenyl-decahydroquinolin-4-ol
(3S,4R)-N,N-dimethyl-4-propyl-1-(3,5,7-trimethyl-1H-indole-2-carbonyl)pyrrolidin-3-amine
4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-methyl-N-[2-(oxan-2-yl)ethyl]benzamide
2-cyclopropyl-9-(3-methoxypropanoyl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
dimethyl[3-(2-{[3-(piperidin-1-yl)pyrrolidin-1-yl]methyl}phenoxy)propyl]amine
1-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-(2-methoxyphenyl)propan-1-one
2-(furan-2-yl)-1-(morpholine-4-sulfonyl)azepane
N-{1-[2-(1,2-oxazolidin-2-yl)-2-oxoethyl]-1H-pyrazol-4-yl}benzamide
N-(propan-2-yl)-1-[1-(propan-2-yl)piperidin-4-yl]piperidine-4-carboxamide
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]piperidin-3-ol
3-(1H-1,3-benzodiazol-1-yl)-1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
2-[1-(5-chlorothiophene-2-carbonyl)pyrrolidin-2-yl]-1-methyl-1H-1,3-benzodiazole
methyl 3-(3,5-dimethyl-1H-pyrrole-2-carbonyl)-9-[3-(1-methyl-1H-pyrazol-4-yl)propoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N4,6-dimethyl-N4-[(3-methylpyridin-4-yl)methyl]pyrimidine-2,4-diamine
1-(1,3-oxazole-5-carbonyl)-N-[4-(1H-pyrazol-5-yl)phenyl]piperidine-3-carboxamide
8-[2-(2,3-dihydro-1H-inden-5-yloxy)-2-methylpropanoyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-[2-(2-ethoxyethoxy)benzoyl]-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
5-(2,3-dihydro-1H-isoindole-2-carbonyl)-2-(pyridin-2-yl)pyrimidin-4-ol
(1S,5R)-3-(4-methylpyrimidin-2-yl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[2-(4-{[2-(2-fluorophenyl)acetamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]-3-phenoxypropanamide
1-{4-[3-(4-chlorobenzoyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one