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3-hydroxy-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]pyridine-2-carboxamide
1-(2-chloro-6-fluoro-3-methylbenzoyl)-4-(1H-imidazol-2-yl)piperidine
(1S,5R)-3-(2,8-dimethylquinoline-3-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
ethyl 4-{2-[1-(3-methylbut-2-en-1-yl)-3-oxopiperazin-2-yl]acetamido}piperidine-1-carboxylate
5-(4-chloro-2-methoxyphenoxymethyl)-N-[(1-hydroxycyclohexyl)methyl]-1,2-oxazole-3-carboxamide
1-(4-chlorophenyl)-N-({4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)cyclobutane-1-carboxamide
N,4-dimethyl-N-[2-(pyrrolidin-1-yl)ethyl]quinazolin-2-amine
6-{5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}pyridine-2-carbonitrile
N-methyl-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-4,5,6,7-tetrahydro-1,3-benzothiazole-2-carboxamide
ethyl 2-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-1,3-oxazole-4-carboxylate
N-benzyl-N-(cyclobutylmethyl)-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
4-benzyl-3-ethyl-1-[2-(2-hydroxyphenyl)acetyl]-1,4-diazepan-5-one
N-{[7-chloro-5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-(4-fluorophenyl)-4-oxobutanamide
N,5,6-trimethyl-N-[(2E)-3-phenylprop-2-en-1-yl]pyridine-3-carboxamide
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}but-2-ynamide
3-{1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]piperidin-3-yl}-N-[4-(trifluoromethyl)phenyl]propanamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-3-(piperidin-4-ylmethyl)benzamide
ethyl 3-[(2-fluorophenyl)methyl]-1-(isoquinoline-1-carbonyl)piperidine-3-carboxylate
1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
4-[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl]-1,4-oxazepan-6-ol
1-[4-(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-1H-pyrazole-4-carbonyl)piperazin-1-yl]ethan-1-one
N-{1-[1-(3-methoxybenzoyl)piperidin-4-yl]-2-phenylethyl}-N,2-dimethylfuran-3-carboxamide
(1S,5R)-N-[3-(methylsulfanyl)phenyl]-7-oxo-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-(5-{[4-(4-methoxyphenoxy)piperidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)pyridine
6-(3-fluoro-4-methoxyphenyl)-N-methyl-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-methyl-3-[2-({[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]carbamoyl}amino)phenyl]propanamide
methyl[1-(4-methylpyridin-2-yl)propan-2-yl]{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}amine
3-(but-2-yn-1-yl)-5-{1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-5-(3-phenylpropyl)imidazolidine-2,4-dione
2-[1-(3-methylbutyl)-4-(pyridin-3-ylmethyl)piperazin-2-yl]ethan-1-ol
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(5-ethyl-1,2,4-oxadiazol-3-yl)piperidine
4-ethyl-7-[(1-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}-1-oxopropan-2-yl)oxy]-2H-chromen-2-one
4-(cyclopropylmethyl)-1-(6-methylpyridazin-3-yl)-3-(propan-2-yl)-1,4-diazepan-5-one
4-[4-(2-chlorophenyl)piperidin-4-yl]-N-cyclopropylpyrimidin-2-amine
methyl 3-{[3-(1H-indol-2-yl)phenyl]carbamoyl}piperidine-1-carboxylate
3-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
2-chloro-N-(2-{[2-(methylamino)pyridin-4-yl]formamido}ethyl)benzamide
2-(3-ethyl-1,2-oxazole-5-carbonyl)-7-(pyrrolidine-1-sulfonyl)-1,2,3,4-tetrahydroisoquinoline
(1S,5R)-6-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
methyl (2S,4S,5R)-5-(2-chlorophenyl)-1,2-dimethyl-4-[(pyridin-4-ylmethyl)carbamoyl]pyrrolidine-2-carboxylate
1-cyclopentyl-N-[(2,4-dimethoxyphenyl)methyl]-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
4-(2-chloropyridine-4-carbonyl)-6-[(3-methoxyphenyl)methoxy]-1-(2-phenylethyl)-1,4-diazepan-2-one
(1S,5R)-3-methyl-6-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
1-methyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-2-oxo-1,2-dihydroquinoline-4-carboxamide
1-[2-(dimethylamino)ethyl]-N-{1-[(2-methylphenyl)methyl]cyclopropyl}-5-oxopyrrolidine-3-carboxamide
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(1-methyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
5-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-3-(phenoxymethyl)-1,2,4-oxadiazole
N-(4-chloro-3-methylphenyl)-2-{[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]amino}acetamide
(3R,5S)-5-[4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]pyrrolidin-3-ol
7-(1-benzofuran-5-carbonyl)-N-ethyl-N-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine