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2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(3,4-dimethoxyphenyl)methyl]acetamide
5-oxo-1-{4-[2-(pyridin-2-yl)ethyl]phenyl}pyrrolidine-3-carboxylic acid
N-{1-[({[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}carbamoyl)methyl]-1H-pyrazol-4-yl}pyridine-2-carboxamide
6-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-2-methyl-2,3-dihydropyridazin-3-one
3-({[3-(dimethyl-1,3-thiazol-2-yl)propyl]amino}methyl)piperidin-3-ol
N-ethyl-5-[5-(1-ethyl-5-methyl-1H-pyrazol-4-yl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine-2-carboxamide
5-oxo-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carboxamide
5-cyclopropanecarbonyl-3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-(2-methoxyethyl)-3-{[1-(1H-1,2,4-triazole-5-carbonyl)piperidin-4-yl]oxy}benzamide
3-[4-(3-methylphenyl)piperazin-1-yl]-N-(oxolan-2-ylmethyl)propanamide
(6S)-6-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]piperidin-2-one
N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-6-(1H-pyrazol-3-yl)pyridine-3-carboxamide
2-benzyl-9-[(5-methylthiophen-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
3-(2-chlorophenyl)-1-[2-(dimethylamino)ethyl]-3-{2-[4-(morpholin-4-yl)piperidin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
7-fluoro-4-(4-methanesulfonylpiperazine-1-carbonyl)-1,2-dihydroquinolin-2-one
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[(1-methyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl]-1,3-dimethyl-1H-pyrazole-4-carboxamide
3-{1-[1-(2-methylpentyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-1-ol
6-[(3-methoxypyrrolidin-1-yl)methyl]naphthalen-2-ol
1-(2-methoxy-5-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}phenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
ethyl 4-({[3-(1,3-oxazol-5-yl)phenyl]carbamoyl}amino)piperidine-1-carboxylate
4-(cyclopropylmethyl)-1-{imidazo[1,2-a]pyridine-2-carbonyl}-1,4-diazepan-5-one
3-[4-(5-chloropyridin-2-yl)piperazine-1-carbonyl]-1,2,5,6,7,8-hexahydroquinolin-2-one
(1S,6R)-9-(4-ethyl-5-methylthiophene-3-carbonyl)-3,9-diazabicyclo[4.2.1]nonane
N-[(3R,4S)-4-cyclopropyl-1-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]pyrrolidin-3-yl]cyclopentanecarboxamide
1-cyclopentyl-4-{[methyl({[2-(propan-2-yl)pyrimidin-5-yl]methyl})amino]methyl}pyrrolidin-2-one
2-{[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]methyl}-1H-imidazole
ethyl 4-({ethyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]carbamoyl}amino)benzoate
[(3-methoxyphenyl)methyl][(4-methyl-1H-imidazol-5-yl)methyl](prop-2-en-1-yl)amine
1-ethyl-N-[(4-methoxyphenyl)methyl]-5-[2-(morpholin-4-yl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(benzylsulfamoyl)({[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl})amine
N-{4-[2-(3-acetylphenyl)-1H-imidazol-1-yl]-2-methoxyphenyl}methanesulfonamide
(2S,4R)-4-amino-N,N-diethyl-1-[(2-ethyl-1-benzofuran-3-yl)methyl]pyrrolidine-2-carboxamide
3-[4-(1H-indol-5-yl)-3,5-dimethyl-1H-pyrazol-1-yl]propanamide
1-{3-[2-(4-chlorophenyl)morpholin-4-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
7-[(5-methyl-1,2-oxazol-4-yl)sulfonyl]-N-(prop-2-en-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-(2-methyl-2H-1,2,3-triazol-4-yl)-2-[5-(5-methylfuran-2-yl)-1H-indol-1-yl]acetamide
3-(2-aminoethyl)-N-(2-{[(2-fluorophenyl)methyl]sulfanyl}phenyl)piperidine-1-carboxamide
2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}-N-[2-(pyridin-2-yl)ethyl]acetamide
2-(benzyloxy)-1-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]ethan-1-one
4-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-yl]-6-methyl-2-phenylpyrimidine
N-[2-(1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperidin-3-yl)ethyl]acetamide
2-(4-methoxyphenyl)-N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]acetamide
2-{4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[(1S,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]ethan-1-one
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-3-(2-fluorophenyl)-1H-pyrazole-5-carboxamide
N-[2-(2-oxoimidazolidin-1-yl)ethyl]-5-[1-(piperidin-1-yl)ethyl]furan-2-carboxamide
3-[4-(3-methylphenyl)piperazin-1-yl]-N-(thiolan-3-yl)propanamide
1-[3-(azepane-1-carbonyl)phenyl]-3-[2-(2-oxoimidazolidin-1-yl)ethyl]urea
N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-2,5-dimethylfuran-3-carboxamide
(1S,5R)-3-benzyl-6-{[3-(morpholin-4-yl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane