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1-(1,3-thiazol-4-ylmethyl)-3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine
1-(2-cyclohexylethyl)-3-({[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl](methyl)amino}methyl)-3-hydroxypiperidin-2-one
methyl 3-[2-(2-methoxyphenoxy)acetyl]-7-oxo-9-(thiophen-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
3-({3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}sulfonyl)pyridine
3-(3-cyclohexyl-1H-1,2,4-triazol-5-yl)-1-(2,3-dihydro-1H-inden-2-yl)urea
N-cyclopropyl-3-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-3-yl]propanamide
5-{1-[2-(2H-1,3-benzodioxol-5-yl)acetyl]piperidin-4-yl}-5-(2-phenylethyl)imidazolidine-2,4-dione
1-[(6-methylpyridin-2-yl)methyl]-4-(3-methylpyridin-4-yl)piperazine
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]benzamide
N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1-(pyridin-3-ylmethyl)piperidin-4-amine
4-[2-(morpholin-3-yl)acetamido]-N-phenylpiperidine-1-carboxamide
3-{5-[2-(difluoromethoxy)phenyl]-1-methyl-1H,4H-pyrazolo[3,4-d]imidazol-3-yl}pyridine
5-(methoxymethyl)-N-{[3-methyl-7-(3-methylbenzoyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}furan-2-carboxamide
N-[(2-fluorophenyl)methyl]-5-methyl-4-{[3-(2-oxopyrrolidin-1-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
N-(3-hydroxypropyl)-7-(propan-2-yl)-N-(pyridin-3-ylmethyl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-2-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)butanamide
5-methyl-2-[4-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenyl]-6-(trifluoromethyl)-3,4-dihydropyrimidin-4-one
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-[2-(thiophen-3-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
1-[(1S,5R)-6-(2-chlorobenzenesulfonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
2-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-2-(2,3-dihydro-1-benzofuran-7-yl)acetic acid
6-methyl-1-[2-(methylsulfanyl)phenyl]-4-{[4-(pyrimidin-2-yloxy)phenyl]methyl}piperazin-2-one
4-[(2-ethylpyrimidin-4-yl)methyl]-1-[(4-fluorophenyl)methyl]piperazin-2-one
3-(3-fluorophenyl)-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]-1H-pyrazole-4-carboxamide
1-(oxan-4-yl)-3-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]piperidine
4-(6-methoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
4-[(2,5-dimethoxyphenyl)carbamoyl]morpholine-2-carboxylic acid
5-{[benzyl(methyl)amino]methyl}-N-{imidazo[1,2-a]pyridin-3-ylmethyl}-1,2-oxazole-3-carboxamide
4-{[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]methyl}pyridine
N-(3-acetylphenyl)-3-(4-methoxy-3,5-dimethylbenzoyl)piperidine-1-carboxamide
2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]acetamide
N,N-dimethyl-6-(3-{1-[(5-methyl-1,2-oxazol-3-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyrimidin-4-amine
3-(azepane-1-carbonyl)-1-ethyl-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-{2-oxo-4-[2-(propan-2-yl)pyrimidin-4-yl]-1,2,3,4-tetrahydroquinolin-7-yl}methanesulfonamide
5-methyl-3-({3-[3-(thiophen-2-yl)phenyl]-1H-pyrazol-1-yl}methyl)-1,2-oxazole
methyl 2-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]pyridine-3-carboxylate
9-(1-benzylpiperidine-2-carbonyl)-1,4,9-triazaspiro[5.5]undecan-5-one
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}piperidin-4-ol
N-[(3R,4S)-1-(6-methoxypyrimidin-4-yl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
(4aR,7aS)-N,N-dimethyl-6,6-dioxo-4-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N-({5-[(3-ethoxy-4-methoxyphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
1-{4-[(3-methylphenyl)methyl]piperazine-1-carbonyl}isoquinoline
2-(5-{1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-4-yl}-1H-pyrazol-3-yl)acetic acid
dimethyl[(5-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]amine
1-{1-[6-(1,4-diazepan-1-yl)pyridine-3-carbonyl]piperidin-3-yl}-3-methylbutan-1-one
(1S,5R)-3-(6-methoxypyrimidin-4-yl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(5-chloro-2-methylphenyl)-4-{[2-methanesulfonyl-1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}piperazine
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-[(1-methyl-1H-imidazol-2-yl)methyl]-N-[4-(1H-pyrazol-5-yl)phenyl]piperidine-3-carboxamide