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3-hydroxy-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}benzamide
2-[5-cyclobutyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-3-yl]pyridine
4-(4-ethyl-6-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}pyrimidin-2-yl)morpholine
3-{2-[4-(2-fluorophenyl)piperazin-1-yl]-2-oxoethyl}-1-methyl-3-(4-phenylphenyl)pyrrolidine-2,5-dione
2-[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]pyridine-4-carboxamide
1-(2H-1,3-benzodioxol-4-ylmethyl)-4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]piperidine
2-methyl-7-({2-[(oxolan-2-ylmethyl)amino]pyrimidin-5-yl}methyl)-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
2-[9-methoxy-7-(6-methoxypyridazin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pyridine-3-carboxamide
1-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}cyclobutan-1-amine
(3S)-3-ethyl-4-[(6-methoxy-2H-chromen-3-yl)methyl]morpholine
4-(2-methyl-5-propylpyrimidin-4-yl)phenol
methyl 3-[2-(2-acetamidoethyl)piperidine-1-carbonyl]-5-methoxybenzoate
(3S,4R)-1-(ethylcarbamoyl)-4-phenylpyrrolidine-3-carboxylic acid
5-acetyl-3-[1-(2-hydroxyethyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]-6-methyl-1,2-dihydropyridin-2-one
[(3,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl){[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}amine
(1R,5S,6S)-6-({4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-3-azabicyclo[3.1.0]hexane
4-{4-[(2,4-dimethoxyphenyl)methyl]piperazin-1-yl}-2-{[4-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindole-1,3-dione
(2E)-N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]-3-(pyridin-2-yl)prop-2-enamide
4-chloro-2-{[3-(2-hydroxyethyl)-4-(thiophen-2-ylmethyl)piperazin-1-yl]methyl}phenol
1-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)-4-(4-methoxybenzoyl)piperazine
(2S,4S)-N-methyl-4-(4-{4-[(4-methyl-1,4-diazepan-1-yl)methyl]phenyl}-1H-1,2,3-triazol-1-yl)pyrrolidine-2-carboxamide
ethyl({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(quinolin-8-ylmethyl)amine
[4-(oxan-2-ylmethyl)-1-{[4-(pyrimidin-2-yloxy)phenyl]methyl}piperidin-4-yl]methanol
N-butyl-2-(3-chloro-6-oxo-1,6-dihydropyridazin-1-yl)-N-[(2-fluorophenyl)methyl]acetamide
4-benzyl-1-(4-chloro-1-methyl-1H-pyrazole-5-carbonyl)-3-ethyl-1,4-diazepan-5-one
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-[(pyridin-2-ylmethyl)amino]pyridine-3-carboxamide
4-(3-{[1-(5-cyclopropyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]oxy}benzoyl)morpholine
[(3-ethyl-4-methyl-1H-pyrazol-5-yl)methyl](methyl)[2-(morpholin-4-yl)ethyl]amine
(3S,4R)-1-(5-chlorofuran-2-carbonyl)-4-methylpiperidine-3,4-diol
5-(2-{[(4-fluorophenyl)methyl]amino}ethyl)-1-[(2-methylphenyl)methyl]pyrrolidin-2-one
N-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-5-methoxy-2-(1H-1,2,3,4-tetrazol-1-yl)aniline
[(2-fluoro-4-methoxyphenyl)methyl]({[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
2-[(2-{[4-(3-hydroxypiperidin-1-yl)pyrimidin-2-yl]amino}ethyl)amino]-6-methyl-3,4-dihydropyrimidin-4-one
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-{[4-(methylsulfanyl)phenyl]methyl}piperazin-2-yl}ethan-1-ol
4-[3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]-6-(propan-2-yl)pyrimidin-2-amine
1-methyl-8-(quinoxalin-2-yl)-1,8-diazaspiro[4.5]decane
2-[2-(1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperidin-4-yl)-1H-imidazol-1-yl]acetamide
4-(naphthalen-2-yloxy)-1-(5-propyl-1,3,4-thiadiazol-2-yl)piperidine-4-carboxylic acid
N-[2-(dimethylamino)ethyl]-1,3-dimethyl-N-(oxolan-2-ylmethyl)-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
3-[(1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperidin-4-yl)oxy]pyridine
2-methoxy-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-5-methyl-N-(pyridin-3-ylmethyl)-1H-pyrazole-4-carboxamide
(9aS)-N-{4-[(2-methoxyethyl)carbamoyl]phenyl}-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carboxamide
(1S,5R)-3-(5-propylthiophene-3-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[5-cyclopropyl-4-(4-ethylpiperazine-1-carbonyl)-1H-pyrazol-1-yl]-4-(3-methoxyphenyl)pyrimidine
ethyl 2-[1-(4-fluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]acetate
2-(dimethylamino)-N-methyl-2-(3-methylphenyl)-N-[3-(1H-pyrazol-1-yl)propyl]acetamide
methyl 4-{[({4-[3-(diethylamino)-2-hydroxypropoxy]-3-methoxyphenyl}methyl)amino]methyl}benzoate
6-(2-chlorophenyl)-8-oxo-N-(oxolan-3-ylmethyl)-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-8-(pyridin-2-yl)-1,8-diazaspiro[4.5]decane