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{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}[(1-methyl-1H-imidazol-2-yl)methyl](propan-2-yl)amine
(3S,4S)-1-(2-amino-6-ethyl-5-methylpyrimidin-4-yl)-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
[2-(3-fluorophenyl)ethyl]({[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
2-[4-(2H-1,3-benzodioxol-4-ylmethyl)-1-[(3,5-dimethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
N-(1-{5-propylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)acetamide
5-[1-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)pyrrolidin-2-yl]-3-phenyl-1,2,4-oxadiazole
2-(2-{[(2S,6S)-4-methyl-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}phenoxy)acetic acid
8-(2,2-dimethylpropyl)-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[1-(1-methyl-1H-indole-2-carbonyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)propanamide
4-[(2-hydroxyethyl)sulfamoyl]-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]benzamide
N-[2-(2-ethylphenoxy)ethyl]-N-methyl-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
[(4aS,8aR)-6-(2-amino-5,6,7,8-tetrahydroquinazoline-4-carbonyl)-decahydro-1,6-naphthyridin-4a-yl]methanol
2-(2-phenyl-1H-imidazol-1-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]acetamide
2-[3-(2-phenylethyl)-5-{1-[2-(propan-2-yl)-1H-imidazol-1-yl]ethyl}-1H-1,2,4-triazol-1-yl]pyridine
N1-(pyridin-3-yl)-N3-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}propane-1,3-diamine
2-butyl-1-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-2,5-dihydro-1H-pyrrole
[2-oxo-2-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)ethyl]urea
3-{[(2-methoxyethyl)(propyl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
[3-(oxolan-3-yl)-1-(quinolin-8-yl)-1H-1,2,4-triazol-5-yl]methanol
5-(3-aminopyrrolidine-1-carbonyl)-2-(4-methylphenyl)pyrimidin-4-ol
N-(2-{[4-methyl-7-(methylsulfanyl)quinolin-2-yl]amino}ethyl)acetamide
N'-(2-fluoro-5-methylphenyl)-N-[2-(1H-imidazol-1-yl)propyl]butanediamide
{3-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-oxopropyl}urea
N-(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)-3-methyl-1H-pyrazole-5-carboxamide
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(3-chlorophenyl)methyl]-4-({[3-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
1-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-phenylethane-1,2-dione
2-amino-5-methyl-4-(2-methyl-1H-imidazol-4-yl)-6-phenylpyridine-3-carbonitrile
N-phenyl-3-({[3-(1H-1,2,4-triazol-1-yl)propyl]carbamoyl}methyl)morpholine-4-carboxamide
7-[2-phenyl-2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-phenyl-1-[4-(pyridin-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]ethan-1-ol
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N-methyl-4-(1H-pyrazol-3-yl)benzamide
1-ethyl-3-[3-(1-methoxyethyl)phenyl]-N,N-dimethyl-1H-1,2,4-triazol-5-amine
(3S,9aR)-8-[(3,4-dimethylphenyl)methyl]-3-[(1R)-1-hydroxyethyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(3S,4R)-1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(3-methylthiophen-2-yl)piperidin-3-ol
1-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}-3-propylurea
N-(2,2-difluoroethyl)-2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
6-(aminomethyl)-2-(4-{[2-(4-fluorophenyl)piperidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
N-[3-hydroxy-2-(thiophen-2-ylmethyl)propyl]-4-(1H-imidazol-1-yl)benzamide
1-[3-({1-[2-(1H-imidazol-5-yl)ethyl]-3-methyl-1H-1,2,4-triazol-5-yl}methoxy)phenyl]-1H-1,2,3,4-tetrazole
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-2-methoxyacetamide
3-[(3S,4R)-1-[(3-chlorophenyl)methyl]-4-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-3-yl]-N-(oxolan-2-ylmethyl)propanamide
1-(2,3-dihydro-1H-inden-2-yl)-4-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-1,4-diazepane
(2-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl](thiophen-3-ylmethyl)amino}ethyl)dimethylamine
1-[3-(4-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}phenoxymethyl)piperidin-1-yl]-2-(1H-pyrazol-1-yl)ethan-1-one
1-ethyl-N-methyl-3-(2-methylpropyl)-N-(quinoxalin-2-ylmethyl)-1H-pyrazole-5-carboxamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[7-fluoro-2-(4-methylphenyl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)propanamide
9-(2,3-difluoro-4-methylbenzoyl)-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-({[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl](methyl)amino}methyl)-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
5-chloro-2-(2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,3-oxazole-4-carbonyl)-1,2,3,4-tetrahydroisoquinoline
13-(5-fluoro-2-methoxyphenyl)-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one