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1-methyl-4-{4-[4-(4H-1,2,4-triazol-4-yl)piperidine-1-carbonyl]phenyl}piperazine
N-(1-cycloheptylpiperidin-3-yl)-4,4,4-trifluorobutanamide
5-[5-(3-fluorophenyl)-1,2,4-oxadiazol-3-yl]-6-methyl-2-[(4-methyl-1H-imidazol-5-yl)methyl]-1,2,3,4-tetrahydro-2,7-naphthyridine
N-{3-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]propyl}acetamide
7-fluoro-2-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-propylquinoline-4-carboxamide
5-cyclopropyl-1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1H-pyrazole-4-carboxamide
N-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3,5-dichlorobenzamide
3-{2-[(4aS,8aR)-decahydroisoquinolin-2-yl]-2-oxoethyl}-1-ethyl-3-[3-(trifluoromethyl)phenyl]pyrrolidine-2,5-dione
N-[(2R)-pyrrolidin-2-ylmethyl]-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-2-(1H-pyrazol-1-yl)benzamide
N,N-diethyl-1-{1-[2-(naphthalen-2-yl)acetyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
N-{[7-chloro-2-(4-hydroxypiperidin-1-yl)quinolin-3-yl]methyl}-N-[2-(4-fluorophenyl)ethyl]pent-4-enamide
2-{[(3S,5S)-5-[4-(adamantan-2-yl)piperazine-1-carbonyl]-1-[(2E)-2-methylbut-2-en-1-yl]pyrrolidin-3-yl]sulfanyl}pyrimidine
2-{4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-[(2-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
3-(cyclopropylmethyl)-1-[3-(pyridin-4-yl)propanoyl]piperidine-3-carboxylic acid
3-[(2R,5S)-2,5-dimethylpyrrolidine-1-carbonyl]-5-(3-fluorophenoxymethyl)-1H-pyrazole
3-{[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl)amino}pyrazine-2-carbonitrile
N-(2,4-dimethylphenyl)-N'-[(2S)-1-hydroxy-3-phenylpropan-2-yl]propanediamide
methyl 3-{[(4-tert-butylphenyl)formamido]methyl}-5-[2-(1H-pyrazol-1-yl)acetamido]benzoate
4-(1-methylpiperidine-2-carbonyl)-1-phenylpiperazin-2-one
5-(2-chlorophenyl)-N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}furan-2-carboxamide
3-(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]propanamide
N-(prop-2-en-1-yl)-N-(pyridin-2-ylmethyl)piperidin-3-amine
5-({[(3-ethoxyphenyl)methyl](2-hydroxyethyl)amino}methyl)-2-hydroxybenzoic acid
5-methoxy-1-methyl-2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1H-indole
7-chloro-4-(furan-3-ylmethyl)-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(cyclopropylmethyl)-2-oxo-3-(oxolan-2-ylmethyl)-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
1-{4-[(6-chloropyridin-3-yl)methyl]piperazin-1-yl}-2-(dimethylamino)-2-(4-methylphenyl)ethan-1-one
2-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
(1S,3R)-3-amino-N-(4-phenylquinolin-8-yl)cyclopentane-1-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-8-(1H-indol-2-ylmethyl)-1-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(2-ethoxyethyl)-N-[(3-methylphenyl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
1-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-3-(pyridin-4-yl)propan-1-one
1-[7-(1,3-benzothiazol-2-yl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(pyridin-2-ylsulfanyl)ethan-1-one
3-methyl-N-[3-(methylcarbamoyl)-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-1-propyl-1H-pyrazole-4-carboxamide
5-cyclopropyl-N-[2-(dimethylamino)ethyl]-N-ethyl-1-[4-(2-fluorophenyl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
(5-{[1-(2-chloro-6-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}furan-2-yl)methanol
3-methoxy-1-[3-(4-methoxyphenoxymethyl)piperidin-1-yl]propan-1-one
3-cyano-N-{4-[ethyl(phenyl)carbamoyl]phenyl}piperidine-1-carboxamide
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]cyclopropanesulfonamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-3-propyl-1H-pyrazole-5-carboxamide
3-(2,3-dihydro-1H-isoindol-2-ylmethyl)-6-ethoxy-1,2-dihydroquinolin-2-one
N-[2-(1H-imidazol-1-yl)ethyl]-5-(1-pentanoylpyrrolidin-2-yl)thiophene-2-carboxamide
2,5-dimethoxy-N-[(5-{[(3-methylphenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]benzamide
(3R,5S)-N-[2-(dimethylamino)ethyl]-5-[(4-methylpiperazin-1-yl)methyl]piperidine-3-carboxamide
N-({1-[(6-chloropyridin-2-yl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)butanamide
4-(2-methoxyphenyl)-6-methyl-5-{2-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}-1,2,3,4-tetrahydropyrimidin-2-one
4-({4-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperazin-1-yl}methyl)benzoic acid
4-(5-chloro-2,3-dihydro-1H-indole-2-carbonyl)piperazine-1-sulfonamide
N-[3-(2-chlorophenoxy)propyl]-2-(ethylamino)-N-methylpyrimidine-5-carboxamide