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N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-2,5-dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
4-{6-[(3-fluorophenyl)methoxy]-4-(2-methylpropyl)-3-oxo-1,4-diazepane-1-carbonyl}-N,N-dimethylpiperidine-1-carboxamide
2-fluoro-N-[1-({[2-hydroxy-3-(3-methoxyphenoxy)propyl]carbamoyl}methyl)-1H-pyrazol-4-yl]benzamide
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}cyclopent-1-ene-1-carboxamide
(3S,9aR)-3-[(1R)-1-(benzyloxy)ethyl]-8-(3-methylbutyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[1-(oxolan-2-ylmethyl)piperidin-4-yl]-1-phenyl-1H-1,2,3-triazole-4-carboxamide
3-(3-fluorophenoxymethyl)-1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperidine
1-{3-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]phenyl}-1H-pyrazole
3-[(5-{1-[(1S)-2,3-dihydro-1H-inden-1-yl]-1H-imidazol-2-yl}furan-2-yl)sulfanyl]-4-methyl-4H-1,2,4-triazole
2-(2-aminoethyl)-N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}quinazolin-4-amine
4-(3-{[1-(2-methyl-6-propylpyrimidin-4-yl)piperidin-4-yl]amino}propyl)phenol
1,3-dimethyl-N-[2-(pyridin-4-yl)ethyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-({1-[4-(dimethylamino)benzoyl]piperidin-3-yl}methyl)naphthalene-1-carboxamide
1-{[2-chloro-5-methoxy-4-(propan-2-yloxy)phenyl]methyl}-4-(1-methyl-1H-imidazol-2-yl)piperidine
(1-{6-phenylimidazo[2,1-b][1,3]thiazole-3-carbonyl}piperidin-4-yl)methanol
5-[(3-aminoazepan-1-yl)methyl]-2-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-ol
3-[2-({[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}amino)ethyl]-1,3-oxazolidin-2-one
N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-2-(pyridin-4-ylsulfanyl)acetamide
5-methyl-3-(thiophen-3-ylmethyl)-5-[1-(2,4,5-trifluorobenzoyl)piperidin-4-yl]imidazolidine-2,4-dione
N-(2-methoxyethyl)-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
N-{[1-(piperidin-1-yl)cyclopentyl]methyl}-3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-(cyclohexylmethyl)-5-[ethyl(2-methylprop-2-en-1-yl)amino]-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-{4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]piperazin-1-yl}-6-methoxypyrimidin-2-amine
(2S,4R)-4-acetamido-N,N-diethyl-1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]pyrrolidine-2-carboxamide
N-[2-(6-methylpyridin-2-yl)ethyl]-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]acetamide
N-benzyl-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-(2-phenylethyl)acetamide
[(1-cyclohexylpiperidin-3-yl)methyl][(2,3-difluorophenyl)methyl](pyridin-3-ylmethyl)amine
4-[(dimethylamino)methyl]-1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]azepan-4-ol
1-[(4-fluorophenyl)methyl]-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
1-cyclopentyl-4-{5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperazin-2-one
N-(oxan-4-ylmethyl)-6-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
2-methyl-4-(2-methylphenyl)-1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperazine
(4aS,8aR)-6-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-1-propyl-decahydro-1,6-naphthyridin-2-one
1-({3-[4-(propan-2-yl)piperidine-1-carbonyl]-1,2-oxazol-5-yl}methyl)piperidin-4-ol
1-(4-{[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-2-(1H-1,2,4-triazol-1-yl)propan-1-one
2-(2-chloro-4-fluorophenyl)-N-{[5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
2-(4-benzylpiperidin-1-yl)-2-[4-(dimethylcarbamoyl)phenyl]acetic acid
(1-{[6-(dimethylamino)pyridin-3-yl]methyl}-3-(prop-2-en-1-yl)piperidin-3-yl)methanol
4-hydroxy-2-(phenoxymethyl)-N-[2-(pyridin-3-yl)ethyl]pyrimidine-5-carboxamide
3-phenoxy-N-{1-[({[3-(1H-pyrazol-1-yl)phenyl]methyl}carbamoyl)methyl]-1H-pyrazol-4-yl}propanamide
4-(2-methoxyethyl)-1-{[2-(methylsulfanyl)phenyl]methyl}piperidine
5-[1-(2-cyclopentylacetyl)piperidin-4-yl]-5-(pyridin-3-yl)-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]-N-(3-phenylpropyl)acetamide
6-[5-(3-ethyl-1,2-oxazol-5-yl)-3-(2-methoxyethyl)-1H-1,2,4-triazol-1-yl]-2-methyl-1,3-benzothiazole
N-{[4-(but-3-yn-1-yloxy)phenyl]methyl}-2-methoxy-N-(oxolan-2-ylmethyl)benzamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-2-(2-oxo-1,2-dihydroquinoxalin-1-yl)acetamide
1-[(2,3-difluorophenyl)methyl]-4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-(4-chlorophenyl)-N-{[1-(furan-3-ylmethyl)piperidin-3-yl]methyl}cyclopropane-1-carboxamide
1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-1,2,4-triazole
4-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]oxane-4-carbonitrile