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N-[(3S)-2-oxoazepan-3-yl]-4-{4-[(thiophen-2-ylmethyl)amino]piperidin-1-yl}benzamide
5-cyclobutyl-3-{[5-(1-ethyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-1,2,4-oxadiazole
8-[2-(pyridin-4-yl)ethanesulfonyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
dimethyl[2-(2-{1-[1-(4-methylphenyl)cyclopropanecarbonyl]piperidin-3-yl}-1H-imidazol-1-yl)ethyl]amine
2-(4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl)-N,N-diethylacetamide
4-chloro-1-methyl-3-({4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}methyl)-1H-indazole
2-(3-chloro-4-fluorophenyl)-2-[2-(1-ethylpiperidin-4-yl)acetamido]acetic acid
(2R,3S,6R)-3-phenyl-5-(pyrimidin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(2-methoxyethyl)-2-(3-methyl-1H-pyrazole-5-carbonyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
3-{[methyl(1,2-oxazol-5-ylmethyl)amino]methyl}-N-(6-methylpyridazin-3-yl)benzamide
3-[(3-hydroxyphenyl)methyl]-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
[(3R,4R)-1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
2-{[(1-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-3-yl)oxy]methyl}pyridine
N-[2-(4-methoxyphenyl)ethyl]-2-(morpholin-3-yl)-N-(pyridin-4-ylmethyl)acetamide
N-{[2-(trifluoromethoxy)phenyl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethyl-5,6,7,8-tetrahydroquinazolin-2-amine
N-methyl-N-[4-(morpholin-4-yl)butyl]-1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
(2S,4S)-N-ethyl-1-(prop-2-en-1-yl)-4-[2-(3,4,5-trifluorophenyl)acetamido]pyrrolidine-2-carboxamide
1-(4-fluorophenyl)-2-(thiophene-3-carbonyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
2-{4-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}-1,3-benzothiazole
2-(2-oxopyrrolidin-1-yl)-N-[(3R,4S)-4-propyl-1-(pyrimidin-2-ylmethyl)pyrrolidin-3-yl]acetamide
1-{3-[2-methyl-5-(3-methylphenyl)pyrimidin-4-yl]piperidin-1-yl}-2-(morpholin-4-yl)-2-(pyridin-3-yl)ethan-1-one
6-(3-methoxy-2-methylbenzoyl)-2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
3-chloro-4-[1-(1-cyclopropylethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]phenol
(2S,4R)-N-(2-methoxyethyl)-4-[(naphthalen-1-ylmethyl)amino]-1-(propan-2-yl)pyrrolidine-2-carboxamide
N-[(1-hydroxycyclohexyl)methyl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
1-ethyl-5-{1-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-4-phenyl-1H-imidazol-5-yl}-1H-1,2,4-triazole
(3S,4S)-4-methyl-1-{[3-(pyridin-2-ylmethoxy)phenyl]methyl}piperidine-3,4-diol
6,6-dimethyl-5-oxo-N-[(5-phenyl-1H-pyrazol-3-yl)methyl]-N-(propan-2-yl)thiomorpholine-3-carboxamide
5-(dimethylamino)-2-(2-oxo-2-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethyl)-2,3-dihydropyridazin-3-one
7-(2-methoxyphenyl)-2-[(1-methyl-1H-1,2,4-triazol-5-yl)methyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-(azepan-1-yl)-N-{imidazo[1,2-a]pyridin-2-ylmethyl}pyridine-2-carboxamide
2-(2-chlorophenyl)-N-{[8-(furan-3-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
1-[(2,6-dimethoxyphenyl)methyl]-3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)urea
N-{1-oxaspiro[4.4]nonan-3-yl}-3-(pyridin-3-yl)propanamide
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
N-cyclopropyl-1-[1-(5-cyclopropyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
N-[(3R,4S)-1-(4-chlorobenzenesulfonyl)-4-propylpyrrolidin-3-yl]acetamide
1-[1-(4-propylpyrimidine-5-carbonyl)piperidin-4-yl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
4-methoxy-N-{[1-(6-methylpyridine-2-carbonyl)piperidin-3-yl]methyl}benzene-1-sulfonamide
2,5-dioxo-6-[2-(propan-2-ylsulfanyl)ethyl]-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-{3-[4-phenyl-1-(2-propoxypropyl)-1H-imidazol-5-yl]phenoxy}ethan-1-ol
3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]propanamide
2-cyclobutanecarbonyl-1-(4-ethylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
3-[3-(pyrrolidine-1-carbonyl)pyridin-2-yl]phenol
3-[(3R,5R)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidine-1-carbonyl]-6-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
N-methyl-N-(2-methylpropyl)-3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-methyl-N-[(4-methylphenyl)(pyridin-4-yl)methyl]-1H-pyrazole-4-carboxamide
N-methyl-2-[methyl(pyridin-4-ylmethyl)amino]-N-[(1-phenylpyrrolidin-3-yl)methyl]acetamide
ethyl(methyl){[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}amine