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7-chloro-2-(1-methyl-1H-pyrazol-4-yl)-N-(oxan-4-yl)quinoline-4-carboxamide
1-[3-(1H-imidazol-2-yl)benzoyl]-3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
1-(2-cyclohexylethyl)-N-methyl-N-[1-(pyridin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-(1-methyl-1H-pyrazol-4-yl)-1-[4-(pyridin-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propan-1-one
methyl 2-[(3,5-dimethylphenyl)sulfamoyl]-6-(2-methylbutanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-{[3-methyl-7-(oxolane-2-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(methylsulfanyl)benzamide
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
N-[(3S,4R)-1-[2-(azepan-1-yl)-2-oxoethyl]-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
(3-{2-[1-(5-chloropyridine-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
N-({7-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-5-(methoxymethyl)furan-2-carboxamide
3-cyano-N-ethyl-5-fluoro-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
N,N-dimethyl-2-[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]aniline
N-[2-(3-methylpyridin-2-yl)ethyl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
2-[2-({[(3S,4R)-4-hydroxyoxolan-3-yl](methyl)amino}methyl)-4-(pyrazin-2-yl)phenoxy]acetic acid
4-[2-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
1-{5-[(4-ethoxyphenyl)methyl]-1H-1,2,4-triazol-1-yl}butan-2-ol
1-(4-methoxybenzenesulfonyl)-3-(naphthalene-2-carbonyl)piperidine
N-[(3S,4R)-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
1-{2-[(3-fluorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-methyl-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]piperidine-4-carboxamide
[(3R,4R)-4-(azepan-1-ylmethyl)-1-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]pyrrolidin-3-yl]methanol
{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]amine
N-(butan-2-yl)-N-cyclopentyl-2-(pyridin-2-yl)acetamide
7-chloro-N,3,5-trimethyl-N-(oxan-4-ylmethyl)-1-benzofuran-2-carboxamide
2-(4-fluorophenoxy)-1-[(3S,4S)-3-hydroxy-4-[4-(2-hydroxyethyl)piperidin-1-yl]pyrrolidin-1-yl]ethan-1-one
(3R,5S)-5-{4-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidine-1-carbonyl}pyrrolidin-3-ol
5-{1-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]piperidin-4-yl}-5-(2-methylpropyl)-3-(thiophen-2-ylmethyl)imidazolidine-2,4-dione
1-{1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-4-(4-fluorophenyl)piperazine
2-(2-fluoro-5-methoxyphenyl)-4,6-dimethoxypyrimidine
{2-[6-(4-methyl-1H-pyrazol-1-yl)pyrimidin-4-yl]phenyl}methanol
N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
N-(cyclopropylmethyl)-1,3-dimethyl-N-propyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
1-{1-[3-(4-fluorophenyl)phenyl]piperidin-4-yl}piperidine-4-carbonitrile
(3S,4S)-4-(4-fluorophenyl)-1-(isoquinoline-1-carbonyl)piperidin-3-ol
N-[2-(pyrrolidine-1-sulfonyl)ethyl]pyrazolo[1,5-a]pyridine-7-carboxamide
2-({2-[2-(pyridin-3-yl)piperidine-1-carbonyl]phenyl}amino)acetic acid
(4aS,7aR)-1-(2-ethylpyrimidine-5-carbonyl)-4-(2-methoxyacetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl(2-phenyl-1-{1-[4-(propan-2-yloxy)benzoyl]piperidin-4-yl}ethyl)(pyridin-3-ylmethyl)amine
4-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2-dihydroisoquinolin-1-one
2-{5-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)phenyl]-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
(1S,5R)-6-(dimethyl-1,3-thiazole-5-carbonyl)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
N-[(3R,4S)-1-[(2-aminopyridin-3-yl)methyl]-4-cyclopropylpyrrolidin-3-yl]oxane-4-carboxamide
5-[3-(azepan-1-yl)-3-oxopropyl]-5-[(4-methoxynaphthalen-1-yl)methyl]pyrrolidin-2-one
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-[(4-methyl-1,3-thiazol-5-yl)methyl]piperidine
(3S,4S)-1-(3-fluoropyridin-4-yl)-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
2-[7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-4-ylmethyl)acetamide
4-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperazin-2-one
5-[1-(3-chlorobenzoyl)piperidin-4-yl]-5-(2-methylpropyl)-3-(thiophen-2-ylmethyl)imidazolidine-2,4-dione
2-{1-[(5-chlorofuran-2-yl)methyl]pyrrolidin-2-yl}pyridine
{3-[(2,4-difluorophenyl)methyl]-1-(1-methyl-1H-indole-3-carbonyl)piperidin-3-yl}methanol
N-[2-(dimethylamino)ethyl]-2-methyl-N-{[7-(methylsulfanyl)-2-(thiophen-2-yl)quinolin-3-yl]methyl}-1,3-thiazole-4-carboxamide