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2-{3-[4-(benzyloxy)piperidine-1-carbonyl]piperidin-1-yl}acetamide
N-(pyridin-4-ylmethyl)-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
2-[3-({[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]amino}methyl)-2-methyl-1H-indol-1-yl]acetamide
2-(4-chlorophenyl)-2-{[1-(propan-2-yl)piperidin-4-yl]formamido}acetic acid
4-(3-fluorophenoxy)-1-[2-(pyridin-2-yl)acetyl]piperidine-4-carboxylic acid
{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]methylamine
2-methyl-4-(piperidin-4-yl)-6-{1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}pyrimidine
2,8-dimethyl-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)quinoline-4-carboxamide
N-cyclopropyl-2-(4-fluorophenyl)-N-{[5,6,7-trimethoxy-2-(2-methylphenyl)quinolin-3-yl]methyl}acetamide
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]morpholine-4-sulfonamide
1-{[3-(2-phenylethyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
5-({3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}methyl)-N-methylfuran-2-carboxamide
4-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-1-[(3-fluorophenyl)methyl]piperazin-2-one
1-({1-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)-1,4-diazepan-5-one
N-(1-{1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-4-yl}-2-phenylethyl)-N-methylthiophene-2-carboxamide
2-{1-[2-(dimethylamino)ethyl]-3-(3-fluorophenyl)-2,5-dioxopyrrolidin-3-yl}-N-(furan-2-ylmethyl)-N-methylacetamide
2-[4-chloro-2-({methyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)phenoxy]acetic acid
2-(4-methoxyphenyl)-N-({1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]piperidin-3-yl}methyl)acetamide
2-[(1-acetylpiperidin-4-yl)oxy]-N-[(dimethyl-1,2-oxazol-4-yl)methyl]-5-methoxybenzamide
(1S,5R)-3-[2-(3-chlorophenyl)acetyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(4-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}benzoyl)piperidin-3-ol
6-methoxy-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]pyrimidin-4-amine
6-cyclopropyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}pyrimidin-4-amine
2-methoxy-N-[(1-methyl-1,2,5,6-tetrahydropyridin-3-yl)methyl]-N-(prop-2-en-1-yl)acetamide
1-cyclohexyl-4-[4-(1H-pyrazol-1-yl)benzoyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
N-methyl-2-oxo-N-[2-(1H-pyrazol-4-yl)ethyl]-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-[4-(1H-1,2,3-benzotriazole-5-carbonyl)morpholin-3-yl]-N-[2-(dimethylamino)ethyl]-N-methylacetamide
(4aS,7aR)-1-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}({2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl})amine
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(propan-2-yloxy)ethan-1-one
1-(2,2-diphenylacetyl)-4-[(4-methoxyphenyl)methyl]-1,4-diazepan-5-one
(6-{8-methoxy-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2-methylpyrimidin-4-yl)methanamine
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-[(4-methoxypiperidin-1-yl)methyl]piperidin-2-one
N-{1-[(4-methylphenyl)methyl]cyclopropyl}-2-(1H-1,2,3,4-tetrazol-5-yl)acetamide
2-[1-cyclopropyl-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-(quinolin-5-ylmethyl)acetamide
5-{3-cyclopropyl-1-[2-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-5-yl}-1,2-dihydropyridin-2-one
1-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(thiophen-2-yl)ethan-1-one
{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}(methyl)(1,2-oxazol-5-ylmethyl)amine
2-[2-(4-fluorophenoxy)ethyl]benzamide
(1-{[5-(2,6-dimethoxyphenyl)-4-phenyl-1H-imidazol-1-yl]methyl}cyclobutyl)methanol
(3-{2-[1-(2-fluoro-6-methoxybenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
3-[(dimethylamino)methyl]-1-(9H-purin-2-yl)pyrrolidin-3-ol
(1S,4S)-2-(2-methoxy-5-phenylphenyl)-5-[3-(3-methyl-1H-pyrazol-1-yl)propanoyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
4-({2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}amino)-1-propylpyrrolidin-2-one
1-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-4-[2-(propan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidine
[(3-{2-[1-(furan-3-carbonyl)piperidin-2-yl]ethoxy}phenyl)methyl](methyl)(quinolin-8-ylmethyl)amine
2-(2-aminoethyl)-N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-5,6-dimethylthieno[2,3-d]pyrimidin-4-amine
[(3-fluorophenyl)methyl](methyl)({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amine
3-methyl-1-[1-(6-{pyrazolo[1,5-a]pyridin-7-yl}pyridine-3-carbonyl)piperidin-3-yl]butan-1-one
6-methoxy-N-[(5-methylpyrazin-2-yl)methyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide