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N-(cyclopropylmethyl)-N-propyl-2-(1H-pyrazole-3-carbonyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
1-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
N-(1-{1-[(3-ethoxy-4-hydroxyphenyl)methyl]piperidin-4-yl}-2-phenylethyl)-N-methylthiophene-2-carboxamide
N-cyclobutyl-3-{[2-(2-methoxyethyl)piperidin-1-yl]sulfonyl}benzamide
3-(5-{[2-(difluoromethoxy)phenyl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanoic acid
1-(3-chlorophenyl)-4-{2-[4-(propan-2-yl)morpholin-2-yl]acetyl}piperazin-2-one
methyl 9-[2-(2-fluorophenyl)ethoxy]-3-[(4-fluorophenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(2-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoethyl)pyrrolidin-2-one
N-[(2R,3R)-2-methoxy-1'-(4,4,4-trifluorobutanoyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide
6-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methyl-1-{7-methyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carbonyl}piperidine
1-[(3-fluorophenyl)methyl]-4-[(4,4,4-trifluorobutyl)amino]pyrrolidin-2-one
1-{3-[(diethylamino)methyl]phenyl}-3-methyl-3-[1-(4-methylpyridin-2-yl)propan-2-yl]urea
2-(2-methyl-1H-pyrrole-3-carbonyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
4-(6-ethoxy-2,3-dihydro-1H-inden-5-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
7a-[2-(4H-1,2,4-triazol-4-yl)ethyl]-hexahydro-1H-pyrrolizine
N-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
2-[(1-acetylpiperidin-4-yl)oxy]-5-methoxy-N-[3-(methylsulfanyl)propyl]benzamide
(4aS,8aR)-6-[2-(dimethylamino)-6-ethylpyrimidin-4-yl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
methyl 4-[(4aS,7aR)-6,6-dioxo-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-1-carbonyl]benzoate
5-(3-chlorophenyl)-3-[4-(4-fluorophenyl)piperazin-1-yl]-1,2,4-triazine
methyl 3-({[4-(3-fluorophenyl)phenyl]formamido}methyl)-5-[2-(1H-pyrazol-1-yl)acetamido]benzoate
N-[(3R,4S)-1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
3-cyclopropyl-N-({2-[3-(2-methoxyacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-1H-pyrazole-5-carboxamide
8-{[6-(dimethylamino)pyridin-3-yl]methyl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-[3-(4-phenylbenzoyl)piperidine-1-carbonyl]pyridine
3-hydroxy-3-({[2-(1H-imidazol-2-yl)ethyl]amino}methyl)-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
3-{1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]piperidin-4-yl}-1,3-oxazolidin-2-one
6-ethyl-4-(4-methanesulfonylpiperazine-1-carbonyl)-1,2-dihydropyridin-2-one
[2-(diethylamino)ethyl](ethyl){[3-(3-methylbutyl)-1,2,4-oxadiazol-5-yl]methyl}amine
2-amino-6-butanoyl-4-(5-tert-butyl-1H-pyrazol-3-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
8-[(2,3-dimethoxyphenyl)methyl]-3-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl 9-(cyclopentyloxy)-3-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[1-(4-fluorophenyl)piperidin-4-yl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
1-(4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}-1,4-diazepan-1-yl)-2-methoxyethan-1-one
3-benzyl-N-[(2-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
3-[2-(ethanesulfonyl)ethyl]-1-[4-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]urea
1-({3-[2-(pyridin-2-yl)piperidine-1-carbonyl]-1,2-oxazol-5-yl}methyl)piperidin-4-ol
2-{4-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-1,2-oxazole-3-carbonyl]morpholin-3-yl}-1-(pyrrolidin-1-yl)ethan-1-one
4-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}phthalazin-1-ol
N-(3-{pyrazolo[1,5-a]pyrimidin-3-yl}phenyl)acetamide
3-[({2-[3-(azepan-1-yl)-2-hydroxypropoxy]-5-chlorophenyl}methyl)(methyl)amino]propanamide
N-{[5-chloro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-methylpiperidine-4-carboxamide
2-{4-[2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)acetyl]-2-oxopiperazin-1-yl}benzonitrile
N3-(cyclopropylmethyl)-N5-[1-(furan-2-yl)ethyl]-4-oxo-1-(propan-2-yl)-N3-propyl-1,4-dihydropyridine-3,5-dicarboxamide
methyl 4-{3-[(4-fluorophenyl)amino]piperidine-1-carbonyl}benzoate
1-[2-(dimethylamino)ethyl]-N-{[4-(methylsulfanyl)phenyl]methyl}-6-oxopiperidine-3-carboxamide
N-[(3-fluorophenyl)methyl]-7-(3-methoxypropyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
6-methoxy-2-oxo-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-1,2,3,4-tetrahydroquinoline-4-carboxamide
3-[1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-1-(4-phenylpiperazin-1-yl)propan-1-one