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7-(thiophen-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
N-cyclopentyl-4-[4-(4-methoxyphenyl)-3-oxopiperazin-1-yl]-4-oxobutanamide
2-benzyl-9-(2-propoxyacetyl)-2,9-diazaspiro[5.5]undecan-3-one
6-[2-(furan-2-yl)pyrrolidine-1-carbonyl]-1,3-benzothiazole
N-(furan-2-ylmethyl)-N-{[2-(4-hydroxypiperidin-1-yl)-7-(methylsulfanyl)quinolin-3-yl]methyl}-3-(2-methoxyphenyl)propanamide
1-(2-methanesulfonylethyl)-2-(4-methoxynaphthalen-1-yl)-1H-imidazole
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-({[2-(5-methylfuran-2-yl)ethyl]amino}methyl)piperidin-2-one
N2,6-dimethyl-N4-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]pyrimidine-2,4-diamine
6,8-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)-4-(2-methylpyrrolidine-1-carbonyl)quinoline
3-({4-[4-(2-ethoxyethyl)piperazin-1-yl]-6-methylpyrimidin-2-yl}amino)phenol
{4-[(2-chlorophenyl)methyl]-1-[4-(piperidin-1-yl)benzoyl]piperidin-4-yl}methanol
7-[(2,3-dimethoxyphenyl)methyl]-2-[(2E)-3-phenylprop-2-en-1-yl]-2,7-diazaspiro[4.5]decan-6-one
5-ethyl-N-({5-[4-(methylsulfanyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-1,2-oxazole-3-carboxamide
6-(1-ethyl-1H-pyrazole-3-carbonyl)-N-methyl-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[9-methoxy-7-(quinolin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
N-[(5-methylpyrazin-2-yl)methyl]-1-(oxan-4-yl)piperidine-4-carboxamide
2-(2-hydroxypropyl)-9-[(1-methyl-1H-imidazol-5-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(3-fluorophenyl)-1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
2-(2,3-dihydro-1-benzofuran-7-yl)-2-{methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}acetic acid
(2S,4S)-4-amino-1-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-N-methylpyrrolidine-2-carboxamide
N-(3-ethoxypropyl)-3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-(carbamoylmethoxy)-N-cyclopropyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]benzamide
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-4-(4H-1,2,4-triazol-4-yl)benzamide
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-3-(1-methylcyclopropyl)propanamide
1-{1-[3-(furan-2-yl)-1-(4-methoxyphenyl)-1H-1,2,4-triazol-5-yl]ethyl}-4-methylpiperazine
(4aS,8aR)-1-(4-hydroxybutyl)-6-[5-(hydroxymethyl)furan-2-carbonyl]-decahydro-1,6-naphthyridin-2-one
methyl 3-(2H-1,3-benzodioxol-5-ylmethyl)-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
2-[2,5-dioxo-3-phenyl-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]-N-methyl-N-(quinoxalin-6-ylmethyl)acetamide
(1R,3S)-3-methoxy-7-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-7-azaspiro[3.5]nonan-1-ol
4-(4-chlorophenyl)-1-[5-(naphthalen-1-yl)-1,2,4-triazin-3-yl]piperidin-4-ol
3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methyl-1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidine
3-acetyl-N-[(2-chlorophenyl)methyl]-N-(2-methoxyethyl)-1H-pyrazole-5-carboxamide
5-[2-(4-fluorophenyl)azetidine-1-carbonyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole
(3S,5R)-5-(azepane-1-carbonyl)-N-(4-methylphenyl)piperidine-3-carboxamide
N-[(1-ethylpyrrolidin-3-yl)methyl]-1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}piperidine-4-carboxamide
N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-4-(pyridin-4-yl)pyrimidin-2-amine
N-(1-{1-[(dimethylcarbamoyl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}ethyl)-N,3,5-trimethyl-1,2-oxazole-4-carboxamide
(2S,4R)-1-{[4-(benzyloxy)phenyl]methyl}-N-[2-(2-methoxyphenyl)ethyl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
(4aS,7aR)-1-(1,3-benzothiazole-6-carbonyl)-4-(cyclopropylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-cyclopropyl-3-({1-[(4-ethylphenyl)methyl]piperidin-4-yl}oxy)-4-methoxybenzamide
6-{9-ethyl-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}pyrazine-2-carboxylic acid
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-phenylpyrimidine-5-carboxamide
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-3-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
4-({5-[3-(3-fluorophenyl)-1H-pyrazol-4-yl]-1,2,4-oxadiazol-3-yl}methyl)morpholine
(1R,2S)-N-[(5-methyl-2-{3-[3-(pyridin-3-yl)propanamido]phenyl}-1,3-oxazol-4-yl)methyl]-2-propylcyclopropane-1-carboxamide
N,N-dimethyl-3-(3-phenylpropanoyl)piperidine-1-sulfonamide
4-[2-(4-aminopiperidin-1-yl)-2-oxoethyl]-1-methyl-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
2,2-dimethyl-N-{1-[1-(1-methyl-1H-indole-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}propanamide
N-ethyl-4-[2-(2-hydroxyphenoxy)acetamido]piperidine-1-carboxamide