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(7-methoxy-3,7-dimethyloctyl)[5-(morpholin-4-yl)pentyl]amine
6-{3-[(1S,3R)-3-hydroxy-1-methoxy-1-methyl-7-azaspiro[3.5]nonan-7-yl]-3-oxopropyl}-2,3-dihydropyridazin-3-one
4-(2-methylpropyl)-3-{2-oxo-2-[4-(pyridin-2-yl)piperazin-1-yl]ethyl}piperazin-2-one
3,5-difluoro-2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
3-{[2-(aminomethyl)morpholin-4-yl]methyl}-6,8-dimethyl-1,2-dihydroquinolin-2-one
N-cyclopropyl-N-{[4-(methylsulfanyl)phenyl]methyl}-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carboxamide
2-benzyl-8-[(4-hydroxyphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
2-methyl-4-(2-methylphenyl)-1-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]piperazine
5-methoxy-2-[5-(propane-1-sulfonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]-1H-1,3-benzodiazole
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}({[4-(2-methylpropyl)phenyl]methyl})(pyridin-4-ylmethyl)amine
2-methoxy-6-({3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)phenol
1-(1-{1-[(4-methoxy-2,5-dimethylphenyl)methyl]piperidin-4-yl}ethyl)-4-methylpiperazine
N-(2-{[(3-chlorophenyl)methyl]sulfanyl}ethyl)-2-methylpyrimidine-5-carboxamide
[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl](methyl){4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}amine
5-[1-(4-tert-butylbenzoyl)piperidin-4-yl]-5-propyl-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amine
4-(3-methyl-1H-1,2,4-triazol-5-yl)-1-{[5-(oxan-2-yl)thiophen-2-yl]methyl}piperidine
ethyl 1-[(2-methyl-1,3-thiazol-5-yl)methyl]-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
N-benzyl-N-(4-hydroxybutyl)-2-[(prop-2-en-1-yl)amino]benzamide
5-methoxy-1-methyl-N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]-1H-indole-2-carboxamide
7-amino-4-{3-[3-(dimethylamino)propoxy]phenyl}-1,2,3,4-tetrahydro-1,8-naphthyridin-2-one
1-(3-{2-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]-1H-imidazol-1-yl}piperidin-1-yl)-2-methylpropan-1-one
5-(2,4-difluorophenoxymethyl)-N-(furan-2-ylmethyl)-N-methyl-1H-pyrazole-3-carboxamide
2,4-dimethyl-5-[4-(pyridin-2-yl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]pyrimidine
[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]({1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl})amine
3-(1H-pyrazol-1-yl)-N-[1-(thian-4-yl)piperidin-4-yl]benzamide
3-{[1-(furan-3-ylmethyl)piperidin-4-yl]oxy}-N-(pyridin-2-ylmethyl)benzamide
(2S,4R)-4-amino-1-[2-(2-phenyl-1,3-thiazol-4-yl)acetyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
methyl 5-[(2R,3R)-3-acetamido-2-(pyridin-2-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-5-oxopentanoate
4-(3-{2-[(4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanoyl)-1-[(3-methylphenyl)methyl]piperazin-2-one
5-ethyl-1'-(2-methoxypyridine-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[4-(3-methoxyphenyl)phenyl]-1-[(2-propylpyrimidin-5-yl)methyl]piperidine-3-carboxamide
1-{2-[1-(2-fluorophenyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}-4-methylpiperazine
[1-({methyl[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}methyl)cyclobutyl]methanol
(1S,5R)-6-[4-(methylsulfanyl)benzoyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-(3-hydroxyquinoxalin-2-yl)-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)propanamide
1-(7-methoxy-4-methylquinazolin-2-yl)-N-(2-methoxyethyl)-N-(propan-2-yl)piperidine-3-carboxamide
N-ethyl-2-(morpholin-4-yl)-6-{8-thiatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-yl}pyridine-3-carboxamide
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-methyl-N-(1H-pyrazol-3-ylmethyl)acetamide
5-oxo-1-(pyridin-3-ylmethyl)-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyrrolidine-3-carboxamide
8-(4-chloro-1H-pyrazole-3-carbonyl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-(furan-3-carbonyl)-N-[3-(3-methylphenyl)phenyl]piperidine-3-carboxamide
2-{4-[6-(aminomethyl)pyridin-3-yl]phenyl}-N,N-dimethylacetamide
4-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-2-(morpholin-4-ylmethyl)-1,4-oxazepane
[(1R,3S,3aS,6aR)-3-{4-[(dimethylamino)methyl]thiophen-2-yl}-5-methyl-1-(2-methylpropyl)-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
2-(dimethylamino)-2-(2-fluorophenyl)-N-[3-(methylamino)propyl]acetamide
5-(4-fluorophenyl)-4-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-2-methylpyrimidine
3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}-N-methyl-N-(2-methylpropyl)propanamide