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8-chloro-2-({cyclopropyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)quinolin-4-ol
N-({7-[(2E)-3-(2,6-difluorophenyl)prop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-ethyl-1-methyl-1H-pyrazole-5-carboxamide
methyl (2S,3S)-2-{[5-(2-chloro-4-methoxyphenoxymethyl)-1,2-oxazol-3-yl]formamido}-3-methylpentanoate
(4aS,8aR)-6-(thiophen-3-ylmethyl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
2-[(2,3-dimethoxyphenyl)methyl]-4-[4-(2-oxo-2H-chromene-3-carbonyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
(1R,5R)-6-(2,4-dimethoxybenzoyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-[2-(1H-imidazol-4-yl)ethyl]-N-methyl-3-oxo-N-phenyl-2,9-diazaspiro[5.5]undecane-9-carboxamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-{[4-(dimethylamino)-1-methylpiperidin-4-yl]methyl}-5-methylpiperidin-2-one
5-chloro-N-(1-methylpiperidin-4-yl)-6-oxo-N-(2-phenylethyl)-1,6-dihydropyridine-3-carboxamide
(3S,4R)-4-(3-methylthiophen-2-yl)-1-(quinolin-2-ylmethyl)piperidin-3-ol
4-{[1-(4-hydroxy-3-methylbenzoyl)pyrrolidin-3-yl]methyl}benzoic acid
3-(3-methoxyphenoxymethyl)-1-(1-methyl-1H-pyrazole-4-carbonyl)piperidine
4-ethyl-6-(2-methoxyethyl)-2-(piperidin-1-yl)pyrimidine
N-{[7-chloro-5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(3,4-difluorophenyl)acetamide
1-[3-(2-methoxyphenyl)-1H-pyrazole-5-carbonyl]-2-(1-methyl-1H-pyrazol-3-yl)piperidine
N-[2-(2-chloro-6-methylphenoxy)ethyl]-3-(4-hydroxyphenyl)-1H-pyrazole-5-carboxamide
1-(6-hydroxy-1,4-oxazepan-4-yl)-3-(3-methoxyphenyl)propan-1-one
N-[(3-chlorophenyl)methyl]-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidine-3-carboxamide
N-[3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)propyl]-1H-pyrazole-4-carboxamide
1-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-3-[1-methyl-3-(pyridin-3-yl)-1H-pyrazol-5-yl]urea
N-methyl-3-(pyrrolidine-1-carbonyl)-N-(thian-4-yl)benzene-1-sulfonamide
N-[(2-chlorophenyl)methyl]-1-ethyl-N-(prop-2-en-1-yl)-1H-pyrazole-4-carboxamide
1-(1-methyl-1H-imidazole-2-carbonyl)-3-(4H-1,2,4-triazol-3-yl)piperidine
N-[2-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-6-hydroxypyridine-3-carboxamide
1-[2-methyl-5-oxo-4-(2-phenylphenyl)piperazine-1-carbonyl]cyclopropane-1-carboxamide
[(4-cyclopropyl-5-{1-[(3-fluoro-2-methylphenyl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
N-methyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
8-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[3-(2-phenylpropyl)-1,2-oxazole-5-carbonyl]piperidine
N-{[5-fluoro-7-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-oxo-2,3-dihydro-1H-indene-1-carboxamide
2-methyl-N-[(2R,3R)-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
[3-ethyl-1-(2-methylpyridin-4-yl)piperidin-3-yl]methanol
N-{2-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}acetamide
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(3-methyl-1,2-oxazol-5-yl)acetamide
1-{2-[4-(1-hydroxy-3-methylbutyl)piperidin-1-yl]-2-oxoethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
N-cyclopropyl-N-(1-{1-[(4-fluorophenyl)methyl]piperidin-4-yl}-2-phenylethyl)pyridine-2-carboxamide
1-{4-[hydroxy(thiophen-2-yl)methyl]piperidin-1-yl}-2-({6-[4-(pyridin-2-yl)piperazin-1-yl]pyridazin-3-yl}oxy)ethan-1-one
4-[3-({2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propyl]-1,3-thiazol-2-amine
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
3-(8-chloro-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-1-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]urea
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-1-ethyl-3-methyl-1H-pyrazole-5-carboxamide
N-[5-({4-[2,5-dioxo-1-(oxolan-2-ylmethyl)-4-propylimidazolidin-4-yl]piperidin-1-yl}methyl)thiophen-2-yl]acetamide
[9-(1H-imidazol-2-ylmethyl)-3-[(2E)-3-phenylprop-2-en-1-yl]-3,9-diazaspiro[5.5]undecan-1-yl]methanol
1-{3-[7-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]phenyl}pyrrolidin-2-one
4-(2,4-difluoro-3-methoxyphenyl)-1-[(dimethyl-1,2-oxazol-4-yl)methyl]-1H-1,2,3-triazole
1-[(1-methanesulfonylpiperidin-3-yl)methyl]-3-[1-(propan-2-yl)-1H-pyrazol-5-yl]urea
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-[5-(pyrrolidin-2-yl)thiophene-2-carbonyl]piperazine
1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
3-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-5-phenyl-1,2-oxazole