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4-[1-(3-methylphenyl)-1H-pyrazol-4-yl]-N-[1-(pyridin-4-yl)propan-2-yl]pyrimidin-2-amine
N-cyclopropyl-4-fluoro-N-{[7-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}benzamide
2-(2-phenyl-1,3-thiazol-4-yl)-1-[3-(pyrimidin-4-yl)piperidin-1-yl]ethan-1-one
N-(2-methoxyethyl)-2-[1-(2-methoxyethyl)-3-(2-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-(propan-2-yl)acetamide
N-({8-[3-(2-chlorophenyl)propanoyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2-fluorobenzamide
4-(cyclopropylmethyl)-1-(2-ethoxypyridine-3-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
methyl 3-(2-chlorobenzenesulfonamido)-5-[(2-methoxyacetamido)methyl]benzoate
4-(2-chlorophenyl)-3-propyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[9-(2-methoxyethyl)-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl]pyridine-4-carbonitrile
[(3R,4S)-4-(morpholin-4-ylmethyl)-1-{[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}pyrrolidin-3-yl]methanol
4-{[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}thiomorpholine
1-{1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]piperidine-3-carbonyl}azetidin-3-ol
N-[(1-ethylcyclopropyl)methyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
methyl 3-[(3S,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl]propanoate
ethyl 2-[4-(5-fluoro-3,8-dimethylquinolin-2-yl)piperazin-1-yl]acetate
1-(1-methylpiperidin-3-yl)-3-[5-(3-oxo-3-phenylpropyl)-1,3,4-thiadiazol-2-yl]urea
N-methyl-2-[3-(2-methylphenyl)-2,5-dioxo-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]-N-(oxan-2-ylmethyl)acetamide
2-[(3-{2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidine-1-carbonyl}phenyl)amino]acetic acid
1-{[3-cyclopropyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]methyl}-4-phenylpiperidine
dimethyl({[(3S,4R)-1-(2-methylfuran-3-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl})amine
(3S,9aR)-8-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-propyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(1S,5R)-3-{2-[(cyclopropylmethyl)sulfanyl]acetyl}-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-cyclopropyl-1-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)propan-1-one
3-ethyl-1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-1,2,4-triazole
4-methyl-3-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]benzene-1-sulfonamide
4-[(5,6,7-trimethoxy-2-oxo-1,2-dihydroquinolin-3-yl)methyl]piperazine-2-carboxylic acid
1-(3,3-dimethylbutanoyl)-N-[3-(1H-indol-2-yl)phenyl]piperidine-3-carboxamide
2-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]acetamide
1-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}-4-(pyrrolidine-1-carbonyl)piperidine
N-{[7-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-phenylcyclopropane-1-carboxamide
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyridine-3-carbonitrile
5-(morpholin-4-ylmethyl)-N-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}furan-3-carboxamide
3-{[(1R,5R)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]sulfonyl}benzoic acid
(4aR,8aR)-2-(4-methyl-1,3-thiazole-5-carbonyl)-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
2-(4-{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)-N,N-dimethylacetamide
[1-({1-[(trimethylpyrazin-2-yl)methyl]piperidin-3-yl}methyl)-1H-1,2,3-triazol-4-yl]methanol
N,6-dimethyl-2-oxo-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,2-dihydroquinoline-4-carboxamide
4-({1-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}oxy)pyridine
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,1,4,6-tetramethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-(3-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenoxy)propanamide
(3S,4R)-1-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
3-(2,5-dioxoimidazolidin-4-yl)-N-{2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethyl}propanamide
N4-methyl-6-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine-2,4-diamine
8-(4-fluorobenzoyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
N-{[7-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(3-methyl-1H-pyrazol-1-yl)propanamide
2-(dimethylamino)-N-{[1-(ethoxymethyl)cyclopropyl]methyl}-2-(4-methylphenyl)acetamide
N,N,3-trimethyl-3-phenylpiperidine-1-sulfonamide
1,3-dimethyl-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
6-ethyl-N-methyl-2-oxo-N-(piperidin-4-yl)-1,2-dihydropyridine-4-carboxamide
N'-[2-(2-methoxyphenyl)ethyl]-N-[2-(methylsulfanyl)phenyl]butanediamide