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benzyl 3-({[(1,3,4-thiadiazol-2-yl)carbamoyl]amino}methyl)piperidine-1-carboxylate
(1R,5S)-6-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}-6-azabicyclo[3.2.1]octane
4-[(2-benzylmorpholin-4-yl)methyl]-5-tert-butylfuran-2-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)imidazo[1,2-a]pyridine-3-carboxamide
2-[({[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]-6-methylphenol
N-[5-(morpholin-4-yl)pentyl]-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
N-{2-[(5-acetylthiophen-3-yl)methyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}-3-(2-methoxyphenyl)propanamide
2-cyclopropyl-N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-4-methylpyrimidine-5-carboxamide
3-(2,5-dioxoimidazolidin-4-yl)-N-[(2-phenoxypyridin-3-yl)methyl]propanamide
{1-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-3-(2-phenylethyl)piperidin-3-yl}methanol
5-ethyl-5-{1-[(5-ethylfuran-2-yl)methyl]piperidin-4-yl}-3-[2-(4-methoxyphenyl)ethyl]imidazolidine-2,4-dione
5-methyl-4-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-1-(3-methylphenyl)piperazin-2-one
5-benzyl-5-[1-(quinolin-6-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione
3-(2-methoxyethyl)-1-[6-(trifluoromethyl)pyridin-2-yl]piperidine-3-carboxylic acid
3-cyclopropyl-N-(1H-imidazol-2-ylmethyl)-N-methyl-1H-pyrazole-5-carboxamide
(4aR,7aS)-1-(1H-imidazol-4-ylmethyl)-4-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(cyclohexylmethyl)-3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
N-[(4-methoxyphenyl)methyl]-6-methyl-2-(4-methylphenoxymethyl)-4-oxo-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-ethoxyethan-1-one
methyl 8-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
4-fluoro-N-({1-[(4-hydroxy-3,5-dimethylphenyl)methyl]piperidin-3-yl}methyl)benzamide
2-[(3R,4S)-3-(3,5-difluoropyridine-2-amido)-4-propylpyrrolidin-1-yl]acetic acid
(4-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-1,4-oxazepan-6-yl)methanol
N-[(1R,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
N-[1-(furan-2-ylmethyl)piperidin-4-yl]-1-(2-hydroxyethyl)-1H-1,3-benzodiazole-5-carboxamide
(1H-1,3-benzodiazol-2-ylmethyl)({1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
1-methyl-3-[4-(2-phenylpyrimidin-4-yl)piperidine-1-carbonyl]-1,4-dihydroquinolin-4-one
1-(2-methoxyethyl)-3-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)-1-(1,3-thiazol-2-ylmethyl)urea
2-(3-fluorophenyl)-1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]piperidine
5-fluoro-2-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-6-oxo-1,6-dihydropyridine-2-carboxamide
N-ethyl-3,5-dimethyl-N-[2-(1H-pyrazol-1-yl)ethyl]-1H-indole-2-carboxamide
4-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-1-(2-methoxyphenyl)-2,2-dimethylpiperazine
3-(2-fluorophenoxy)-1-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}azetidine
5-{1-[(2-hydroxy-3-methoxyphenyl)methyl]piperidin-4-yl}-5-[(3-methoxyphenyl)methyl]-3-methylimidazolidine-2,4-dione
3-(2-oxo-2-{4-[(4-phenyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}ethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(3-{[3-(methanesulfonylmethyl)piperidin-1-yl]methyl}phenoxy)acetamide
2-[3-(3-phenylphenyl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-2-azabicyclo[2.2.1]heptane
3-{2-[4-(3-chlorophenyl)piperazin-1-yl]-2-oxoethyl}-4-methylpiperazin-2-one
N-cyclohexyl-3-{[(3,5-dimethoxyphenyl)formamido]methyl}piperidine-1-carboxamide
2-methoxy-5-[(4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidin-1-yl)methyl]pyridine
1-[(4-fluorophenyl)methyl]-4-(2-methoxypyridine-4-carbonyl)-1,4-diazepane
4-[(2-fluoro-4-methoxyphenyl)methyl]-3-(2-oxo-2-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-yl}ethyl)piperazin-2-one
2-ethoxy-5-[2-({1-oxaspiro[4.4]nonan-3-yl}amino)pyrimidin-4-yl]benzoic acid
N-cyclohexyl-N-[2-(ethylsulfanyl)ethyl]-2-(1H-imidazol-2-yl)benzamide
7-(2,6-dimethoxyphenyl)-9-methoxy-4-{[4-(trifluoromethyl)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(6-chloro-1,3-benzothiazol-2-yl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-(4-methoxyphenyl)-1-(1-methylcyclohexanecarbonyl)piperidin-3-amine
2-{2-[1-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
2,5-dimethyl-N-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine