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2-(2-chlorophenyl)-3-methyl-N-[2-(1,3-thiazol-2-yl)ethyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
3-(3-chlorobenzoyl)-1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidine
6-({methyl[2-(pyridin-2-yl)ethyl]amino}methyl)-2-oxo-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,2-dihydropyridine-3-carboxamide
5-tert-butyl-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-1,3,4-oxadiazol-2-amine
7-fluoro-1-(2-methoxyethyl)-3-({methyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)-1,2-dihydroquinolin-2-one
6-methyl-3-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidine-1-carbonyl}pyridin-2-ol
N-(3,4-dihydro-2H-1-benzopyran-3-yl)-2-(ethylamino)-4-methyl-1,3-thiazole-5-carboxamide
4-[(4-fluorophenyl)methyl]-1-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]-3-(propan-2-yl)-1,4-diazepan-5-one
(4aS,8aR)-6-[2-(methylamino)pyridine-4-carbonyl]-1-[3-(methylsulfanyl)propyl]-decahydro-1,6-naphthyridin-2-one
N-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}-2,7-dimethylimidazo[1,2-a]pyridine-3-carboxamide
(3S,4R)-3-[(dimethylsulfamoyl)amino]-N-(furan-2-ylmethyl)-4-(propan-2-yl)pyrrolidine-1-carboxamide
2-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]-6-methoxy-1,2,3,4-tetrahydroisoquinoline
2-(4-chloro-2-methylphenoxy)-1-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)ethan-1-one
N,N-diethyl-1-{5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-1,2-oxazole-3-carbonyl}pyrrolidin-3-amine
5-[(4-chlorophenyl)methyl]-5-{3-[4-(2-methoxyphenoxy)piperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
N-methyl-3-(3-methylpiperidin-1-yl)-N-{[3-(methylsulfanyl)phenyl]methyl}propanamide
1-{[1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxylic acid
N-{[2-(dimethylamino)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)-2-(thiophen-3-yl)acetamide
1-[(2-chloro-4-fluorophenyl)methyl]-N-methyl-N-(pyridin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
4-[(dimethylamino)methyl]-1-[2-(1H-imidazol-2-yl)benzoyl]azepan-4-ol
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-[(1-ethyl-1H-imidazol-2-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
6-fluoro-N-[2-(2-methyl-1H-indol-1-yl)ethyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-(4,6-dimethylpyrimidin-2-yl)-N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]piperidin-4-amine
{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)(oxolan-2-ylmethyl)amine
1-methyl-N-[(4-oxo-3,4-dihydrophthalazin-1-yl)methyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-butyl-4-oxo-N-(3-phenylprop-2-yn-1-yl)-3,4-dihydroquinazoline-2-carboxamide
1-(2-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)ethan-1-one
N-benzyl-5-{[4-(pyrazin-2-yl)piperazin-1-yl]methyl}pyrimidin-2-amine
1-methyl-3-[1-(1-phenylethyl)-1H-pyrazol-5-yl]-1-(thian-4-yl)urea
{2-[(1-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)oxy]ethyl}dimethylamine
(2S,4S)-N-ethyl-1-(naphthalen-1-ylmethyl)-4-{[(3-phenoxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
3-cyclohexyl-1-[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]propan-1-one
4-hydroxy-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-phenylpyrimidine-5-carboxamide
N-[2-(4-{[2-(cyclohex-1-en-1-yl)acetamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]oxolane-2-carboxamide
2-(4-chlorophenyl)-1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]ethan-1-one
N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-2-(pyridin-2-yl)acetamide
3-(trifluoromethyl)-2-(3,4,5-trimethoxyphenyl)pyridine
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-[2-(trimethyl-1H-pyrazol-1-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
N-[3-(4-fluorophenyl)phenyl]-1-[3-(methylsulfanyl)propanoyl]piperidine-3-carboxamide
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-methyl-2-(pyridin-4-yl)quinoline-4-carboxamide
3-(2H-1,3-benzodioxol-5-yl)-1-{3-[4-(3,4-difluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}propan-1-one
N-[2-methyl-1-(morpholin-4-yl)propan-2-yl]-9-oxo-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraene-10-carboxamide
1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-4-(4-methoxyphenyl)butane-1,4-dione
1-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)-4-[(2-fluorophenyl)methyl]piperidine
1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-4-(pyrimidin-2-yl)piperazine-2-carboxylic acid
8-cycloheptyl-1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-[(1-methyl-1H-pyrazol-4-yl)methyl]benzamide
1-[4-(2-methylphenyl)-3-oxopiperazin-1-yl]-2-phenylethane-1,2-dione
1-[3-(3-fluorophenyl)benzoyl]-4-(4H-1,2,4-triazol-4-yl)piperidine
3-[5-(morpholine-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]-1-(pyrrolidin-1-yl)propan-1-one